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N-[3-(2,3-dihydro-1H-isoindol-2-yl)propyl]-6-fluoro-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
1-methyl-4-(1-{1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}ethyl)piperazine
7-[2-(2-chlorophenoxy)acetyl]-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
[3-(cyclopropylmethyl)-1-[(dimethyl-1,3-thiazol-4-yl)methyl]piperidin-3-yl]methanol
N-methyl-3-(1,2-oxazinan-2-yl)-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}propanamide
1-{imidazo[1,2-a]pyrimidine-2-carbonyl}-2-(3-methoxyphenyl)piperidine
4-{[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]amino}-5-methyl-N-(1,3-thiazol-2-ylmethyl)thieno[2,3-d]pyrimidine-6-carboxamide
N-[3-(2-methyl-5-oxopyrrolidin-1-yl)phenyl]-4-[(methylsulfanyl)methyl]piperidine-1-carboxamide
1-methyl-5-[4-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1H-1,3-benzodiazole
3-{3-benzyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}-1-ethyl-6-methyl-1,2-dihydropyridin-2-one
N-[(3R,4S)-1-acetyl-4-cyclopropylpyrrolidin-3-yl]-2-chloro-6-methylbenzene-1-sulfonamide
N-{2-[(2-cyclohexyl-1,3-benzoxazol-6-yl)formamido]ethyl}acetamide
(2R,6S)-4-[5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]-2,6-dimethylmorpholine
1-{4-[(4-fluorophenyl)methyl]piperidin-1-yl}-2-(morpholin-2-yl)ethan-1-one
2,2,6,6-tetramethyl-4-{[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
1-(butane-1-sulfonyl)-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
1-(1-phenoxypropan-2-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
3-[3-(1-methoxyethyl)phenyl]-N,N-dimethylpyrazin-2-amine
4-acetyl-N-(1,2,3-thiadiazol-5-yl)piperazine-1-carboxamide
6-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]pyrimidin-4-amine
(2S,4S)-1-[(4-chlorophenyl)methyl]-4-{[(2,4-dimethoxy-3-methylphenyl)methyl]amino}-N-ethylpyrrolidine-2-carboxamide
1-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-(1H-pyrazol-1-yl)butan-1-one
(1S,5R)-3-(1,3-benzoxazol-2-yl)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-{6-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl}morpholine
1-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
(4-{[(3,4-difluorophenyl)methyl]amino}quinazolin-2-yl)methanol
2-cyclopropanecarbonyl-8-(3-hydroxybenzoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
methyl 3-(2,1,3-benzothiadiazol-5-ylmethyl)-9-(oxan-2-ylmethoxy)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[(1S,2R)-2-(cyclohexylamino)cyclobutyl]-3-(trimethyl-1H-pyrazol-1-yl)propanamide
N-(4-{[methyl({[4-(oxolan-2-ylmethyl)-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl})amino]methyl}phenyl)acetamide
4-methyl-N-(3-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)-3,4-dihydro-2H-1,4-benzoxazine-7-carboxamide
1-(3-cyanopyridin-2-yl)-N-[2-(pyridin-3-yloxy)phenyl]piperidine-3-carboxamide
N-[3-(2-fluorophenyl)propyl]-4-(piperidin-1-yl)butanamide
5-[2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
1-[(2-amino-5-methylpyrimidin-4-yl)amino]-3-(piperidin-1-yl)propan-2-ol
(2S)-2-{[(5-{1-[(4-methyl-1,3-thiazol-5-yl)methyl]-1H-pyrazol-3-yl}thiophen-2-yl)methyl]amino}butan-1-ol
(1S,5R)-6-[(1-methyl-1H-pyrazol-4-yl)sulfonyl]-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
N-[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
7-(5-methylthiophen-2-yl)-4-(thiophen-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
methyl 2-{[(4-chlorophenyl)methyl]sulfamoyl}-6-cyclobutanecarbonyl-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-(methoxymethyl)-6-[(E)-2-[4-(trifluoromethyl)phenyl]ethenyl]pyrimidine
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-2-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
4-({3-[4-(pyrrolidine-1-carbonyl)pyridin-2-yl]phenyl}methyl)morpholine
{[(3S,4R)-1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl}dimethylamine
1-[(3-{[1-(5-methylthiophene-2-carbonyl)piperidin-4-yl]oxy}phenyl)methyl]-4-(pyridin-3-ylmethyl)piperazine
N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2-(3-methyl-2-oxo-1,2-dihydroquinoxalin-1-yl)acetamide
N-[4-(2-fluorophenoxy)phenyl]-1-(2-oxopropanoyl)piperidine-4-carboxamide
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-2-propyl-1,3-thiazole-4-carboxamide
(1R,3S)-3-[4-(3-chlorophenoxy)piperidine-1-carbonyl]cyclopentane-1-carboxylic acid
2-{3,9-diazaspiro[5.6]dodecan-9-yl}pyridine-3-carboxylic acid