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6-{[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]methoxy}-1,2-benzoxazole
3-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}propanamide
(3aR,6aS)-5-({4-[2-(dimethylamino)ethoxy]phenyl}methyl)-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(1-benzyl-1H-1,2,4-triazol-5-yl)-1,5,6-trimethyl-1,2-dihydropyridin-2-one
(1S,5R)-3-(dimethyl-1,3-thiazole-5-carbonyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
5-benzyl-5-(1-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperidin-4-yl)imidazolidine-2,4-dione
(4aS,8aR)-6-(ethanesulfonyl)-1-[3-(1H-imidazol-1-yl)propyl]-decahydro-1,6-naphthyridin-2-one
(3S,4R)-4-(hydroxymethyl)-1-[4-(1H-pyrazol-1-yl)benzenesulfonyl]piperidin-3-ol
1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine
1-(1,4-dimethyl-3-phenyl-1H-pyrazol-5-yl)-3-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)urea
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(9H-purin-6-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
3-amino-1-[(2-hydroxy-6-methoxyquinolin-3-yl)methyl]pyrrolidine-3-carboxylic acid
2-[2-(benzenesulfonyl)ethyl]-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one
N-[(1-cyclopropanecarbonylpiperidin-4-yl)methyl]-2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
N-(2-methylpropyl)-N-(thiophen-3-ylmethyl)-4-(4H-1,2,4-triazol-4-yl)benzamide
1-(2-hydroxyethyl)-5-(2-methyl-1,2,3,4-tetrahydroisoquinoline-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-(pyrrolidin-3-ylmethyl)-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
3-[(3-hydroxyazetidin-1-yl)sulfonyl]-N-[1-(pyridin-2-yl)propan-2-yl]benzamide
8-{[6-(dimethylamino)pyridin-3-yl]methyl}-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
2-(4-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)-1,3-benzothiazole
(4aR,8aR)-7-[(3-cyanophenyl)methyl]-4a-hydroxy-N,N-dimethyl-decahydro-2,7-naphthyridine-2-sulfonamide
2-({4-[2-(methylsulfanyl)ethyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)quinolin-8-ol
ethyl 2-[(4-{[5-(hydroxymethyl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}piperidine-1-carbonyl)amino]propanoate
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-2-phenylacetamide
1-{7-[(4-acetylpiperazin-1-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-2-(3-fluorophenyl)ethan-1-one
1-[1-(furan-2-carbonyl)piperidin-4-yl]-3-(5-methyl-1,3,4-thiadiazol-2-yl)urea
2-[4-(2H-1,3-benzodioxol-5-yl)-3-(methoxymethyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-(propan-2-yl)acetamide
7-[3-(2-methoxyphenoxy)propyl]-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-methyl-6-{[(3-methyl-1,2-oxazol-5-yl)methyl]amino}pyridine-3-carboxamide
2-amino-6-(2,4-dichlorophenyl)-4-(pyridin-3-yl)pyridine-3-carbonitrile
6-(3-fluoro-4-methoxyphenyl)-1H-1,3-benzodiazole
N-{1-[2-(pyrrolidin-3-yl)benzoyl]piperidin-4-yl}pyrimidin-2-amine
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-[4-(methylsulfanyl)phenyl]acetamide
2-methoxy-4-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}phenol
N-[1-(2-phenylethyl)piperidin-3-yl]-2-(pyridin-2-ylsulfanyl)acetamide
2-({4-[(3R,4R)-3-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidine-1-carbonyl]phenyl}sulfanyl)ethan-1-ol
1-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-4-(1,2,4-oxadiazol-3-yl)piperidine
5-[(benzyloxy)methyl]-1-[(1-ethyl-1H-imidazol-5-yl)methyl]-4-phenyl-1H-imidazole
5-[(2S)-1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}pyrrolidin-2-yl]-3-(2-methoxyethyl)-1,2,4-oxadiazole
N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-2-(1H-pyrazol-1-yl)butanamide
6-methyl-3-[(4-oxo-3,4-dihydrophthalazin-1-yl)methyl]-3,4-dihydroquinazolin-4-one
N-(3,4-dihydro-2H-1-benzopyran-3-yl)-2,3-dimethylquinoxaline-6-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[2-(1H-pyrazol-1-yl)benzoyl]piperazine
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-(4-methoxyphenoxy)-N-({5-methyl-2-[2-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)acetamide
1-[1-(hydroxymethyl)-9-propyl-3,9-diazaspiro[5.5]undecan-3-yl]-2-(trimethyl-1H-pyrazol-1-yl)ethan-1-one
(1R,5R)-3-cyclobutanecarbonyl-6-{[4-(methylsulfanyl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonane
2-(2-methoxyethyl)-3-oxo-N-[(1R)-1-phenylethyl]-2,9-diazaspiro[5.5]undecane-9-carboxamide
ethyl 2-{4-[(6-hydroxy-1,4-oxazepane-4-carbonyl)amino]phenyl}-1,3-oxazole-4-carboxylate