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N-[7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]-3-methylbutanamide
ethyl 2-(1-{5-[3-(trifluoromethyl)phenoxymethyl]-1,2-oxazole-3-carbonyl}piperidin-2-yl)acetate
4-({methyl[1-(methylcarbamoyl)propan-2-yl]amino}methyl)-N-(1,2,4-thiadiazol-5-yl)benzamide
2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]-N-[2-(2-oxopiperidin-1-yl)ethyl]acetamide
5-hydroxy-6-[(4S)-4-hydroxy-3,3,4-trimethylpiperidine-1-carbonyl]-2-(4-methylphenyl)-2,3-dihydropyridazin-3-one
(2,1,3-benzoxadiazol-5-ylmethyl)(methyl){[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}amine
2-phenoxy-N-[4-(4-{[2-(1H-pyrazol-1-yl)ethyl]amino}piperidin-1-yl)phenyl]acetamide
5-fluoro-2-(4-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperazin-1-yl)pyrimidine
(4aS,8aR)-1-(3-methoxypropyl)-6-[2-(phenylsulfanyl)acetyl]-decahydro-1,6-naphthyridin-2-one
5-[3-(1-benzyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-4-methylpyrimidine
3-(4-hydroxyphenyl)-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]propanamide
5-hydroxy-N-[(3R,4S)-1-methanesulfonyl-4-propylpyrrolidin-3-yl]pyrazine-2-carboxamide
4-{3-oxo-1H,2H,3H,4H,5H,6H,7H,8H-pyrazolo[3,4-d]azepine-6-carbonyl}-1,2-dihydroquinolin-2-one
4-{[5-(6-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)-1,2,4-oxadiazol-3-yl]methyl}-1-methylpiperidine
5-(1-{[5-(pyridin-2-yl)thiophen-2-yl]methyl}pyrrolidin-2-yl)thiophene-2-carboxamide
3-amino-1-[(3-fluoro-5-methylphenyl)methyl]pyrrolidine-3-carboxylic acid
5-oxo-N-[(1-phenylcyclohexyl)methyl]-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
3-chloro-N-(2-methoxyethyl)-4-[(1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)oxy]benzamide
2-({[(3R,4R)-1-[(3,5-dimethylphenyl)methyl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
1-[(4-chlorophenyl)methyl]-N-{[4-(dimethylamino)-1-methylpiperidin-4-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
(2S,4R)-4-amino-1-(2H-1,3-benzodioxole-5-carbonyl)-N,N-diethylpyrrolidine-2-carboxamide
3-(4-methoxypiperidine-1-carbonyl)-N-(1,2-oxazol-3-ylmethyl)benzene-1-sulfonamide
4-({5-[1-(3,3-dimethylbutyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)morpholine
2-{1-[(2-ethoxyphenyl)methyl]-4-{[5-(hydroxymethyl)furan-2-yl]methyl}piperazin-2-yl}ethan-1-ol
1-(1-tert-butyl-1H-pyrrole-3-carbonyl)-4-(2-phenoxyethyl)piperazine
1-{3,9-diazaspiro[5.6]dodecan-9-yl}-2-[(2-ethyl-6-methylpyridin-3-yl)oxy]ethan-1-one
3-{2-[2,2-bis(prop-2-en-1-yl)pyrrolidin-1-yl]-2-oxoethyl}-4-(2-phenylethyl)piperazin-2-one
N-(2-ethoxyphenyl)-3-[2-(3-methyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]-3-oxopropanamide
3-[(2-hydroxyethyl)(methyl)sulfamoyl]-N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]benzamide
4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(propane-1-sulfonyl)piperidine
1-[1-(1-cycloheptanecarbonylpiperidin-4-yl)-1H-1,2,3-triazol-4-yl]propan-2-ol
2-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]-N,N-dimethylpyridine-3-carboxamide
3-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-7-methyl-3H,4H-thieno[3,2-d]pyrimidin-4-one
2-[(2-methyl-1,3-thiazol-5-yl)methyl]-2,8-diazaspiro[4.5]decane
6-methyl-3-[1-(3-methylpyridin-4-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]-4H-pyrido[1,2-a]pyrimidin-4-one
2-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
N-[1-(6-chloropyridazin-3-yl)piperidin-4-yl]-5-(oxolan-2-yl)thiophene-2-carboxamide
(3aR,6aS)-5-[(2,3-dimethoxyphenyl)methyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(2-methylpyridin-4-yl)-4-(pyrrolidin-3-ylmethyl)-1,4-diazepane
5-{[1-(2,5-difluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-2-(methylsulfanyl)pyrimidine
4-methyl-2-[1-(1-methyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]-1H-1,3-benzodiazole
3-[(3R,4S)-1-[(5-fluoro-3-methyl-1H-indol-2-yl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
1-[4-({[(3,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)-2-methoxyphenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
1-[(3,5-dimethoxyphenyl)methyl]-N-phenylpiperidin-3-amine
2-[(4,6-dimethylpyrimidin-2-yl)sulfanyl]-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(2-methylpropyl)propanamide
N-propyl-N-(pyridin-2-ylmethyl)-4-[(pyridin-2-ylsulfanyl)methyl]benzamide
(4aS,8aR)-1-(3-hydroxypropyl)-6-[(1-methyl-1H-pyrazol-4-yl)methyl]-decahydro-1,6-naphthyridin-2-one
5,8-dimethoxy-N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-4-methylquinolin-2-amine
3-(2-methoxyphenyl)-N-[2-(4-methyl-5-{[2-(morpholin-4-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)ethyl]propanamide