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N-(2-methoxyethyl)-4-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-phenylpyrimidine-5-carboxamide
1-[4-(4-methoxyphenoxy)piperidin-1-yl]-2-methyl-3-(1H-pyrazol-1-yl)propan-1-one
1-[2-(4-methylpentyl)morpholin-4-yl]-3-(1,2-oxazolidin-2-yl)propan-1-one
N-cyclohexyl-N-methyl-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-[2-(2-fluorophenyl)-1-{1-[3-(prop-2-en-1-yloxy)benzoyl]piperidin-4-yl}ethyl]-N-methyl-3-(methylsulfanyl)propanamide
(3S,4R)-1-[(5-acetylthiophen-3-yl)methyl]-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
1-[(3-methylphenyl)methyl]-4-(oxane-2-carbonyl)piperazine
1-(6-aminopyridine-3-carbonyl)-4-phenoxypiperidine-4-carboxylic acid
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[(6-chloropyridin-3-yl)methyl]piperidin-3-ol
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-N-methyl-2-[(4S)-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]acetamide
[(3R,4R)-1-(5-ethyl-2-methylpyrimidin-4-yl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
1-(2-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-pyrazol-3-yl]phenyl}phenyl)ethan-1-one
5-{3-[2-(2,3-dimethoxyphenyl)-1H-imidazol-1-yl]propyl}-4-methyl-1,3-thiazole
2-(pyrrolidin-1-yl)-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)pyrimidine-5-carboxamide
(1S,5R)-3-benzyl-6-[(3-methyl-1,2-oxazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
3-[(2H-1,3-benzodioxol-4-ylmethyl)amino]-N-(1,3-dihydro-2-benzofuran-5-yl)-5-[(propan-2-yl)sulfamoyl]benzamide
3-butanamido-N-methyl-N-(quinoxalin-2-ylmethyl)benzamide
5-methyl-N-{[8-(3-methylbut-2-en-1-yl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}-1,3-oxazole-4-carboxamide
2-(5-{1-[2-(propan-2-ylsulfanyl)ethyl]pyrrolidin-2-yl}-1,2,4-oxadiazol-3-yl)pyridine
8-(2-methylpyrimidin-4-yl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
(4aR,7aS)-1-(2-methoxyethyl)-4-(3-propyl-1H-pyrazole-4-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[(1S,5R)-7-oxo-6-propyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-1,3-thiazole-4-carboxamide
N-[(3R,4S)-1-[(3-chloro-4-methoxyphenyl)methyl]-4-cyclopropylpyrrolidin-3-yl]-2-methoxyacetamide
methyl 3-[(cyclopropylformamido)methyl]-5-(2,3-dihydro-1,4-benzodioxine-6-sulfonamido)benzoate
N-ethyl-8-methyl-2-(1-methyl-1H-pyrazol-4-yl)-N-(pentan-3-yl)quinoline-4-carboxamide
N-[cyclopropyl(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-6-ethyl-2-methylquinoline-4-carboxamide
4-methyl-2-(1-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperidin-4-yl)-1H-1,3-benzodiazole
N-[2-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)ethyl]-2-(dimethylamino)-2-(2-fluorophenyl)acetamide
2,6-dimethyl-N-{2-[(pyridin-3-yl)amino]ethyl}imidazo[1,2-a]pyridine-3-carboxamide
N-ethyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-1-(pyridin-3-ylmethyl)piperidin-4-amine
1-(2H-1,3-benzodioxol-5-ylmethyl)-5-(5-methyl-1,3-oxazol-4-yl)-1H-1,2,4-triazole
2-methyl-4-{3-[(4-methyl-1,2,3,6-tetrahydropyridin-1-yl)sulfonyl]benzoyl}-1,4-oxazepane
1-benzyl-5-(4-cyclohexylpiperazine-1-carbonyl)-N-ethyl-4-oxo-1,4-dihydropyridine-3-carboxamide
3-(2-hydroxyphenyl)-N-[1-(3-methylphenyl)piperidin-4-yl]-1H-pyrazole-5-carboxamide
1-{4-[(2S)-2-(methoxymethyl)pyrrolidine-1-carbonyl]phenyl}imidazolidine-2,4-dione
3-(6-methoxy-2H-1,3-benzodioxol-5-yl)-1-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]urea
4-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)thiomorpholine
(3S,4R)-1-[1-(7-fluoroquinazolin-2-yl)piperidin-4-yl]-N,N-dimethyl-4-propylpyrrolidin-3-amine
2-cyclohexyl-5-{[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}pyrimidine
N-methyl-3-(3-phenyl-1,2,4-oxadiazol-5-yl)-N-[1-(pyrimidin-4-yl)ethyl]propanamide
N-[2-(2-fluorophenoxy)ethyl]-N-(2-methoxyethyl)-1-methylpiperidine-2-carboxamide
(2,1,3-benzoxadiazol-5-ylmethyl)(methyl)({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amine
N-(2-{2-[3-(cyclopentyloxy)phenyl]-1H-imidazol-1-yl}ethyl)acetamide
benzyl({[5-(1H-pyrazol-5-yl)furan-2-yl]methyl})(1,3-thiazol-2-ylmethyl)amine
(1-{1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-2-phenylethyl)(2-methoxyethyl)(pyridin-2-ylmethyl)amine
1-(2,2-diethylcyclopropanecarbonyl)-2-[2-(1H-imidazol-1-yl)ethyl]piperidine
(3aR,5R,6S,7aS)-2-[1-(4-methoxyphenyl)piperidin-4-yl]-octahydro-1H-isoindole-5,6-diol
N-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-N,7-dimethyl-2-(1H-pyrazol-4-yl)quinoline-4-carboxamide
N-[3-(6-methyl-1,3-benzoxazol-2-yl)propyl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
4-[3-(2-hydroxyethyl)-4-methylpiperazin-1-yl]-2-methoxypyridine-3-carbonitrile