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ethyl 3-[(3-chlorophenyl)methyl]-1-(2-oxo-2-phenylacetyl)piperidine-3-carboxylate
{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amine
(3R,5S)-N3-(2-methoxyethyl)-N3-methyl-N5-(4-methylphenyl)piperidine-3,5-dicarboxamide
3-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-methyl-6-(4H-1,2,4-triazol-4-yl)pyridine
1-[4-(1H-indol-2-yl)phenyl]-N-(1-methoxypropan-2-yl)piperidin-4-amine
3-phenyl-5-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-1,2-oxazole
2-methoxy-6-{[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]methyl}-5-oxo-5,6-dihydro-1,6-naphthyridine-3-carbonitrile
1-{2-hydroxy-3-[2-methoxy-4-({[2-methyl-2-(morpholin-4-yl)propyl]amino}methyl)phenoxy]propyl}piperidin-4-ol
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-N'-(2,4-dimethylphenyl)ethanediamide
1-cyclopentyl-N,N-bis(1,3-oxazol-4-ylmethyl)-5-oxopyrrolidine-3-carboxamide
5-ethyl-4-[4-(thiomorpholin-4-yl)piperidin-1-yl]pyrimidin-2-amine
(2R,3R,6R)-5-(2-ethylpyrimidine-5-carbonyl)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-{1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carbonyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
N-(furan-2-ylmethyl)-2-[1-methyl-10-oxo-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-4-yl]acetamide
(3R,4R)-4-ethyl-1-(9H-fluorene-9-carbonyl)piperidine-3,4-diol
methyl 3-[1-(4-chlorophenyl)cyclopropaneamido]-5-[(pyridin-3-ylformamido)methyl]benzoate
3-methyl-7-(2-phenylquinoline-4-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
4-(3-{2-methyl-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}propoxy)benzamide
N-(2-methoxyethyl)-3-[1-(quinolin-8-ylmethyl)piperidin-4-yl]propanamide
8-(2-methoxypyridine-4-carbonyl)-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
1-[(2E)-hex-2-en-1-yl]-4-[3-(piperidine-1-carbonyl)pyridin-2-yl]piperazine
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-phenylbenzamide
ethyl 2-{2-oxo-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}-1,3-oxazole-4-carboxylate
1-[(2-fluoro-3-{furo[3,2-c]pyridin-4-yloxy}phenyl)methyl]pyrrolidine
1-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
3-[3-(4-methoxyphenoxymethyl)piperidine-1-carbonyl]benzonitrile
1-[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]-4-[(3-methoxyphenyl)methyl]-1,4-diazepan-5-one
5-[(3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)methyl]-1,2,4-oxadiazole-3-carboxamide
1-(butan-2-yl)-3-[3-methyl-1-(3-methylbutyl)-1H-pyrazol-5-yl]-1-(pyridin-4-ylmethyl)urea
1-(2-aminoethyl)-N-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
5-chloro-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
4-methoxy-3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]benzene-1-sulfonamide
5-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-1-(4-methoxyphenyl)-3-(oxan-4-yl)-1H-1,2,4-triazole
2-{[(3S)-1-benzylpyrrolidin-3-yl]amino}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-(3,5-dimethylphenyl)-4-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}piperazin-2-one
4-methoxy-6-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyrimidin-2-amine
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-2-methyl-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
(3S,4R)-1-(1H-imidazol-2-ylmethyl)-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-(1-methyl-2-oxoimidazolidine-4-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
N3-[(4-methylphenyl)methyl]-4-oxo-N5-[2-(propan-2-yloxy)ethyl]-1-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
2-{4-[6-(piperidin-3-yl)pyrimidin-4-yl]piperazin-1-yl}-1,3-benzoxazole
1-[2-(dimethylamino)-6-methyl-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-4-yl]piperidin-4-ol
2-[4-(benzyloxy)butanoyl]-7-ethyl-2,7-diazaspiro[4.5]decan-6-one
3-(2-ethylphenoxy)-1-(furan-2-ylmethyl)azetidine
2-[3-(difluoromethyl)-5-methyl-1H-pyrazol-1-yl]-N-[(5-ethylpyridin-2-yl)methyl]-N-methylacetamide
4-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,2-dihydroquinolin-2-one
1-{[4-chloro-2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-N-(4-fluorophenyl)piperidin-3-amine
1-[(1R,5S,6R)-6-({4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}methyl)-3-azabicyclo[3.1.0]hexan-3-yl]butan-1-one
N-methyl-4-[4-(2-phenylethyl)piperidine-1-carbonyl]-1,3-thiazol-2-amine
2-(4-{[3-(cyclopentyloxy)phenyl]methyl}piperazin-1-yl)pyridine-3-carboxamide