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6-[3-(morpholin-4-yl)propyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
6-{1-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]piperidin-3-yl}pyrimidin-4-ol
1-[4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-2-(pyridin-2-yl)ethan-1-one
3-[(dimethylamino)methyl]-1-[2-methyl-6-(1H-pyrazol-1-yl)pyrimidin-4-yl]piperidin-3-ol
(1R,3S,5S)-3-(4-fluoro-3-methylphenyl)-8-(pyridin-2-ylmethyl)-8-azabicyclo[3.2.1]octane
N-(2-hydroxy-1-phenylethyl)-2-methyl-4-phenylpyrimidine-5-carboxamide
1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-4-(4-fluorophenyl)-1,4-diazepane
4-{[4-(3-methyl-1,2,4-oxadiazol-5-yl)furan-2-yl]methyl}morpholine
N-methyl-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}-2-{2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl}acetamide
3-[(2-{1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]piperidin-4-yl}-1H-imidazol-1-yl)methyl]pyridine
2-(2-methyl-1,3-thiazol-4-yl)-1-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
1-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]-3-(3-hydroxy-1,2-oxazol-5-yl)propan-1-one
6-(2,5-dimethylfuran-3-yl)-2-(2-ethylpyrrolidine-1-carbonyl)-7-methyl-7H,8H-imidazo[1,2-a]pyrazin-8-one
1-(3-chlorophenyl)-5-methyl-4-pentanoylpiperazin-2-one
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-3-(3-fluorophenyl)-1H-pyrazole-4-carboxamide
3-methoxy-5-methyl-N-[4-(methylamino)butyl]thiophene-2-carboxamide
N-[2-(2-chlorophenyl)ethyl]-5-(2-methylphenyl)-1,2,4-triazin-3-amine
[(4-methanesulfonylphenyl)methyl](methyl)[(1-phenylpyrrolidin-3-yl)methyl]amine
N,7,8-trimethyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-2-(1-methyl-1H-pyrazol-4-yl)quinoline-4-carboxamide
2-methyl-N-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
8-[2-(5-amino-3-methyl-1H-pyrazol-1-yl)acetyl]-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[4-carboxy-4-(2-methylphenoxy)piperidin-1-yl]-6-methylpyridine-3-carboxylic acid
(3S,9aR)-3-benzyl-8-(3,5-dichlorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]pyridine
5-(1H-pyrazol-1-ylmethyl)-3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazole
1-methyl-4-({6-[4-(1H-pyrazol-5-yl)phenyl]pyridin-3-yl}methyl)piperazine
(3S,4S)-1-[5-(propan-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl]-4-(propan-2-yloxy)pyrrolidin-3-ol
5-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-2-methylphenol
6-({4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}methyl)-1,4-oxazepan-6-ol
N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}acetamide
1-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-{4-[1-(2-hydroxybutyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}ethan-1-one
2-(1-benzylpiperidin-4-yl)-2,7-diazaspiro[4.5]decane
2-[3-cyclopropyl-5-(3-methylphenoxymethyl)-1H-1,2,4-triazol-1-yl]pyridine
3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-(1,3-thiazole-4-carbonyl)piperidine
4-[(dimethylamino)methyl]-1-{2-methylimidazo[1,2-a]pyridine-6-carbonyl}azepan-4-ol
3-{2-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]-2-oxoethyl}-4-(pyridin-3-ylmethyl)piperazin-2-one
N-ethyl-N-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]thiophene-2-carboxamide
1-(3-methylbutyl)-3-(2-methylpropyl)-8-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(6-{[1-(pyrrolidin-1-yl)hex-5-en-2-yl]oxy}pyrazine-2-carbonyl)morpholine
4-[4-(8-methyl-4-oxo-1,4-dihydroquinoline-3-carbonyl)-2-oxopiperazin-1-yl]benzonitrile
2-{1-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-1,4-diazepan-6-yl}acetic acid
1-(4-{3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}piperidin-1-yl)ethan-1-one
1-(3,4-dihydro-2H-1,4-benzoxazin-4-yl)-2-[(3R,4S)-3-(3-hydroxypropyl)-4-(morpholin-4-yl)piperidin-1-yl]ethan-1-one
{[7-chloro-2-(thiophen-3-yl)quinolin-3-yl]methyl}[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]amine
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N-methyl-1H-pyrazole-3-carboxamide
2-(1H-indol-1-yl)-N-[1-(propan-2-yl)-1H-1,2,3-triazol-4-yl]acetamide
2-(dimethylamino)-N-methyl-2-(3-methylphenyl)-N-(thiophen-3-ylmethyl)acetamide
3-chloro-N-cyclopentyl-4-[(1-methylpiperidin-4-yl)oxy]benzamide
3-[1-(1-acetylpiperidin-4-yl)-1H-pyrazol-5-yl]-1-(2-methylphenyl)urea