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ethyl 1-[7-(2-methoxyacetamido)-1-(2-phenylethyl)-1H-1,3-benzodiazole-5-carbonyl]piperidine-3-carboxylate
3-amino-1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propan-1-one
4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1-[2-(propan-2-yloxy)acetyl]-1,4-diazepan-5-one
1-{5,7-dimethyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carbonyl}-4-phenyl-1,4-diazepane
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-N,1-dimethyl-1H-indole-2-carboxamide
N-[3-(morpholin-4-yl)propyl]-2-(1H-pyrazol-1-yl)butanamide
[(2E)-3-(furan-2-yl)prop-2-en-1-yl][(2-methoxyphenyl)methyl](pyridin-3-ylmethyl)amine
8-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
6-methyl-N-[1-(thian-4-yl)piperidin-4-yl]imidazo[1,2-a]pyridine-2-carboxamide
1-{4-[(3-cyclopropyl-1H-pyrazol-5-yl)methyl]-6-hydroxy-1,4-diazepan-1-yl}-2-(1H-pyrazol-1-yl)ethan-1-one
1-[(6-ethoxy-2,3-dihydro-1H-inden-5-yl)methyl]-4-[(3-methylpyridin-2-yl)methyl]piperazine
4-{methyl[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]sulfamoyl}-N-[(3S)-pyrrolidin-3-yl]benzamide
{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}({2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl})amine
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-5-oxo-2,5-dihydro-1H-pyrazole-3-carboxamide
N-[(4,6-dimethylpyridin-2-yl)methyl]-N,1-dimethyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-[3-(2-chlorophenyl)-1H-pyrazol-5-yl]-1-(1H-imidazol-2-ylmethyl)piperidine
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-[3-(1H-pyrazol-1-yl)azetidin-1-yl]pyridine-3-carboxamide
N-cyclopropyl-1-[(3-methoxyphenyl)methyl]-5-(1H-pyrazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(2S,4S,5R)-5-(3-chlorophenyl)-4-[(2-methoxyethyl)carbamoyl]-1-methylpyrrolidine-2-carboxylic acid
2-methyl-6-{[3-(pyridin-4-yl)azetidin-1-yl]sulfonyl}-1,3-benzothiazole
4-(1H-imidazol-1-yl)-1-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}piperidine-4-carboxylic acid
8-[(8-fluoro-4-hydroxyquinolin-2-yl)methyl]-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
1-(4-benzylpiperazin-1-yl)-3-{1-[2-(3,5-dimethyl-1H-pyrazol-1-yl)acetyl]piperidin-3-yl}propan-1-one
8-(2-amino-4-methyl-1,3-thiazole-5-carbonyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
2-(cyclohex-1-en-1-yl)-1-[3-(hydroxymethyl)-3-(2-phenylethyl)piperidin-1-yl]ethan-1-one
N-cyclopropyl-4-[(2-hydroxy-2-phenylethyl)sulfamoyl]benzamide
1-[1-(3-chlorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-(morpholin-4-yl)propan-1-one
(3R,5S)-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
(3aR,7aS)-2-{[5-(1H-pyrazol-5-yl)furan-2-yl]sulfonyl}-2,3,3a,4,7,7a-hexahydro-1H-isoindole
3-{1-[2-(2-ethyl-1,3-thiazol-4-yl)ethyl]-1H-imidazol-2-yl}pyridine
5-(4-methoxy-2-methylphenyl)-4-phenyl-1-(prop-2-yn-1-yl)-1H-imidazole
N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide
(2S,4S)-N-ethyl-1-(furan-3-ylmethyl)-4-[2-(thiophen-3-yl)acetamido]pyrrolidine-2-carboxamide
1-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}-3-(4,5,6,7-tetrahydro-2H-indazol-3-yl)propan-1-one
1-(2-methylphenyl)-4-[4-(1H-pyrazol-1-yl)benzoyl]-1,4-diazepane
N-benzyl-4-(4H-1,2,4-triazol-4-yl)piperidine-1-sulfonamide
3-[(2,4-difluorophenyl)methyl]-1-(5,6-dimethylpyrimidin-4-yl)piperidine-3-carboxylic acid
4-[(1-cyclopentylpiperidin-4-yl)oxy]-3-methoxy-N-[(6-methylpyridin-2-yl)methyl]benzamide
N-[(2,4-dimethoxyphenyl)methyl]-3-ethyl-4-methyl-1H-pyrazole-5-carboxamide
3-cyclopropyl-N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]-1H-pyrazole-5-carboxamide
N-methyl-5-phenyl-N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-1,2-oxazole-4-carboxamide
N,N-dimethyl-2-[methyl(2-phenylethyl)amino]-2,3-dihydro-1H-indene-2-carboxamide
(1R,9S)-5-amino-12-methyl-3-[2-(methylsulfanyl)pyrimidin-5-yl]-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
3-[(dimethylamino)methyl]-1-(2,2-dimethylpropyl)-3-hydroxypiperidin-2-one
5-cyclopropyl-N-[2-(4-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-3-methyl-1H-pyrazole-4-carboxamide
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-{[1-(hydroxymethyl)cyclopropyl]methyl}-5-methylpiperidin-2-one
2-[2-(hydroxymethyl)piperidin-1-yl]-N,N-bis(prop-2-en-1-yl)acetamide
(3aS,6aR)-3-[3-(4-methoxyphenyl)propyl]-N,N-dimethyl-2-oxo-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazole-5-sulfonamide
[(5-cyclopropyl-1,2-oxazol-3-yl)methyl][(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]methylamine
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(1-methylpiperidin-4-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane