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4-[2-(2-methyl-4-oxo-1,4-dihydroquinolin-1-yl)acetyl]-1λ6-thiomorpholine-1,1-dione
(3S,4S)-4-(propan-2-yl)-1-(1,3-thiazol-2-yl)pyrrolidine-3-carboxylic acid
N-(1-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}piperidin-4-yl)methanesulfonamide
2-(4-{7-cyclopropanecarbonyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}morpholin-2-yl)ethan-1-amine
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-[(4-methoxy-2,5-dimethylphenyl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-5-(morpholin-4-ylmethyl)furan-3-carboxamide
5-[3-(4-fluorophenoxymethyl)piperidine-1-carbonyl]-2-methoxyphenol
1-(3-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}phenyl)imidazolidin-2-one
N-(1-benzylcyclopropyl)-3-[(4-fluorophenyl)formamido]propanamide
1-(4-{[(5-methyl-1H-pyrazol-3-yl)methyl]amino}-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
(1S,5R)-6-[(2-butyl-1H-imidazol-4-yl)methyl]-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-(piperidin-1-yl)-3-[(3S,4R)-1-(pyridin-2-ylmethyl)-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]propan-1-one
4-(1-ethyl-1H-1,3-benzodiazol-2-yl)-3-(furan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-[2-(furan-2-yl)-2-(pyrrolidin-1-yl)ethyl]-3-(3-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-5-yl)urea
1-(2-{[2-(4-methanesulfonylphenyl)-1H-imidazol-1-yl]methyl}phenyl)-1H-1,2,4-triazole
(3S,4R)-4-(hydroxymethyl)-1-(1H-indole-7-carbonyl)piperidin-3-ol
6-[1-methyl-10-oxo-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-4-yl]pyrazine-2-carboxamide
2-{[2-(1-{imidazo[1,2-a]pyridine-2-carbonyl}piperidin-4-yl)-1H-imidazol-1-yl]methyl}pyridine
(1-{[5-(2-fluorophenyl)furan-2-yl]methyl}piperidin-4-yl)(1-methyl-1H-imidazol-2-yl)methanol
4-({[6-methyl-2-(pyridin-3-yl)pyrimidin-4-yl]amino}methyl)benzene-1-sulfonamide
4-[(1-{[1-(3-chloropyridin-2-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]piperazin-2-one
2-(furan-2-yl)-5-({4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}methyl)pyrimidine
4-[(1-{[1-(cyclohex-3-ene-1-carbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]piperazin-2-one
5-methyl-4-[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]thieno[2,3-d]pyrimidine-6-carboxylic acid
2-amino-N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)acetamide
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
1-[1-(4,6-dimethylpyrimidin-2-yl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
1-[(2-fluorophenyl)methyl]-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-4-carboxamide
N-[(2,5-dimethylphenyl)(pyridin-3-yl)methyl]-5-methyl-1,3,4-oxadiazole-2-carboxamide
1-(2-{4-[(dimethylamino)methyl]phenyl}pyrrolidin-1-yl)-2-(pyridin-3-yloxy)ethan-1-one
2-(1-{[4-(furan-2-yl)phenyl]methyl}pyrrolidin-2-yl)ethan-1-ol
2-{N-methyl-1-[1-(propan-2-yl)-1H-pyrazol-4-yl]formamido}-2-(thiophen-2-yl)acetic acid
N-[(2-amino-1,3-thiazol-4-yl)methyl]-2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
1-(2-aminoethyl)-N-{3-[(4-chlorophenyl)sulfanyl]propyl}-1H-1,2,3-triazole-4-carboxamide
2-(4-{[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]methyl}phenyl)acetic acid
4-phenyl-N-{1-[1-(2-phenylethyl)piperidin-4-yl]-1H-pyrazol-5-yl}butanamide
N-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-bromobenzamide
N-[2-(dimethylamino)-2-(2-methylphenyl)ethyl]-2-(piperidin-4-yl)acetamide
3-[(3S,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-fluorophenyl)urea
(2S,4R)-4-cyclobutaneamido-N-ethyl-1-[(6-methylpyridin-2-yl)methyl]pyrrolidine-2-carboxamide
4-{[2-(quinolin-8-yl)-1H-imidazol-1-yl]methyl}benzene-1-sulfonamide
(2R,3R)-1'-(2-amino-6-hydroxypyrimidin-4-yl)-3-(pyrrolidin-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
4-(3-fluorophenyl)-3-(1H-pyrazol-5-yl)-4H-1,2,4-triazole
1-(furan-2-ylmethyl)-4-[4-methyl-6-(methylamino)pyrimidin-2-yl]-1,4-diazepane-6-carboxylic acid
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[2-(2-fluorophenyl)ethyl]piperidine-3-carboxamide
3-phenyl-N-[4-(4-{[1-(pyridin-2-yl)propan-2-yl]amino}piperidin-1-yl)phenyl]propanamide
(2-{2-[1-(2-ethoxybenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
N-cyclobutyl-3,6,7-trimethyl-1-benzofuran-2-carboxamide
5-(2-hydroxypropyl)-11-methyl-8-thia-3,5,10-triazatricyclo[7.4.0.02,7]trideca-1(13),2(7),3,9,11-pentaen-6-one
1-(4-{3-[2-(3-methoxyphenyl)ethyl]piperidin-1-yl}piperidin-1-yl)ethan-1-one