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[3-(4-methoxyphenyl)propyl](methyl)[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]amine
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-cyclopentanecarbonylpyrrolidine-3-carboxylic acid
1-ethyl-3-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
6-(morpholin-4-yl)-N4-(1-propylpiperidin-3-yl)pyrimidine-2,4-diamine
N-{[5-(benzylsulfanyl)-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl]methyl}-5-methylthiophene-2-carboxamide
9-(5-ethyl-1,3-oxazole-4-carbonyl)-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-(2-methoxyacetyl)-N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-3-carboxamide
1-[(2-fluorophenyl)methyl]-N-{[1-(2-phenylethyl)piperidin-4-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
(4aS,7aR)-1-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(4S)-1-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-3,3,4-trimethylpiperidin-4-ol
5-[(3-methyl-3-phenylpiperidin-1-yl)sulfonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[5-(3-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]azocane
N,N-dimethyl-6-{4-[1-(piperidin-1-yl)ethyl]phenyl}pyridazin-3-amine
1-(6-aminopyrimidin-4-yl)-4-(quinolin-6-yloxy)piperidine-4-carboxylic acid
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1-(2-methoxyethyl)piperidine
(5S,9aS,9bS)-5-[4-(4-hydroxybut-1-yn-1-yl)phenyl]-2-(2-methoxyphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(4-methyl-1H-pyrazol-1-yl)propan-1-one
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-3,5-dimethyl-1,2-oxazole-4-carboxamide
1-benzoyl-2-[3-(2,6-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]piperidine
1-[4-({[4-(pyridin-4-yl)pyrimidin-2-yl]amino}methyl)phenyl]pyrrolidin-2-one
[3-methyl-5-(3,4,5-trimethoxyphenyl)-1H-indol-2-yl]methanol
(2S,4R)-4-amino-N-ethyl-1-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]pyrrolidine-2-carboxamide
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-2-(4,6,7-trimethyl-1-benzofuran-3-yl)acetamide
4-methoxy-6-[4-(pyridin-4-yl)piperidin-1-yl]pyrimidin-2-amine
(1R,5R)-3-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-6-propyl-3,6-diazabicyclo[3.2.2]nonane
[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]({[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl})amine
5-(2-methoxyphenoxymethyl)-N-[(3-methyloxetan-3-yl)methyl]-1H-pyrazole-3-carboxamide
4-[(3,4-dimethoxyphenyl)methyl]-3-[2-(1,2-oxazinan-2-yl)-2-oxoethyl]piperazin-2-one
4-{[6-(morpholin-4-yl)pyridin-3-yl]sulfonyl}morpholine-2-carboxylic acid
3-[3-({[2-(pyridin-3-yloxy)propyl]amino}methyl)-1H-indol-1-yl]propanamide
2-[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]-1H-1,3-benzodiazole-5-carbonitrile
1-(1-benzofuran-2-ylmethyl)-N-phenylpiperidin-3-amine
3-{[(1R,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}pyridin-2-amine
1,3-dimethyl-2,6-dioxo-N-[3-(2-propoxyphenyl)propyl]-1,2,3,6-tetrahydropyrimidine-4-carboxamide
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-phenylprop-2-ynamide
N,N-dimethyl-3-oxo-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecane-9-sulfonamide
1-(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepin-3-yl)-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
1-[(4-fluorophenyl)methyl]-2-methyl-3-[2-oxo-2-(piperazin-1-yl)ethyl]-4,5,6,7-tetrahydro-1H-indol-4-one
(1-{[5-chloro-2-(prop-2-en-1-yloxy)phenyl]methyl}pyrrolidin-3-yl)methanamine
3-{[3-(cyclopropylmethyl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]methyl}phenol
2-(3-methoxypropyl)-9-(2-methyl-6-propylpyrimidin-4-yl)-2,9-diazaspiro[5.5]undecan-3-one
2-(3-hydroxypropyl)-8-{[2-(methylsulfanyl)phenyl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
1-(8-fluoro-4-oxo-1,4-dihydroquinoline-2-carbonyl)-4-hydroxypiperidine-4-carboxylic acid
5-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
N-methyl-6-oxo-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1-(pyridin-2-ylmethyl)piperidine-3-carboxamide
3-(4-hydroxyphenyl)-1-[2-(3-methoxypropyl)piperidin-1-yl]propan-1-one
2-(3-methoxypropyl)-8-(pyridin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
N-[2-(pyridin-3-yloxy)phenyl]-1-(1,3-thiazol-2-yl)piperidine-3-carboxamide
1-({6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-4-(3-methylpyridin-4-yl)-1,4-diazepane
1-[3-(azepane-1-carbonyl)phenyl]-3-ethyl-3-[(3S,4R)-4-hydroxyoxolan-3-yl]urea