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1-(2-methoxyethyl)-4-[4-(pyridin-4-ylmethyl)-1,4-diazepane-1-carbonyl]pyrrolidin-2-one
2-ethoxy-4-{[3-(pyrrolidin-1-yl)piperidin-1-yl]methyl}phenol
3-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-5-methyl-1,2-oxazole
N-{[2-(4-acetylpiperazin-1-yl)-7-methoxyquinolin-3-yl]methyl}-N-(2-methoxyethyl)thiophene-2-carboxamide
2-[3-(phenoxymethyl)-5-[4-(4H-1,2,4-triazol-4-yl)phenyl]-1H-1,2,4-triazol-1-yl]ethan-1-ol
3-(4-methoxyphenyl)-1-[4-(1,2,4-oxadiazol-3-yl)piperidin-1-yl]-3-phenylpropan-1-one
6-methyl-2-{[(2-methyl-6-propylpyrimidin-4-yl)amino]methyl}-3,4-dihydropyrimidin-4-one
9-methoxy-7-(4-methylphenyl)-4-(2-methylpropyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-[(3-methoxyphenyl)sulfanyl]-1-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
2-[2-(piperidin-1-ylmethyl)-1,4-oxazepane-4-carbonyl]quinoline
(2S)-2-amino-2-methyl-3-phenyl-1-[4-(thiomorpholin-4-yl)piperidin-1-yl]propan-1-one
N-[2-(2-ethylphenoxy)ethyl]-N-methyl-3-(1,2-oxazinan-2-yl)propanamide
(3aS,7aR)-5-methyl-2-(4-phenoxybutanoyl)-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
4-(benzyloxy)-1-(piperidin-3-ylmethyl)piperidine
2-{[2-({2-[(4-methylpyridin-2-yl)amino]ethyl}carbamoyl)phenyl]amino}acetic acid
1-[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-(thiophene-3-carbonyl)piperidine
3-[2-(4,4-diphenylpiperidin-1-yl)-2-oxoethyl]-1,3-oxazolidin-2-one
1-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
methyl({[2-(5-methylfuran-2-yl)phenyl]methyl})[3-(1H-pyrazol-1-yl)propyl]amine
N-[2-(7-{[3-(4-chlorophenoxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]furan-3-carboxamide
(1R,5S,6R)-3-[(3,5-dimethyl-1-benzofuran-2-yl)methyl]-N-(2-hydroxyethyl)-3-azabicyclo[3.1.0]hexane-6-carboxamide
3-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-[(2-fluorophenyl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
8-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-1-oxa-8-azaspiro[4.5]decane
2-(dimethyl-1,2-oxazol-4-yl)-2-[4-(2-ethoxyphenyl)piperazin-1-yl]acetic acid
2-(adamantan-1-yl)-N-[1-(pyridin-4-yl)propan-2-yl]acetamide
(1S,9S)-11-[2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetyl]-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
(2-methoxyethyl)[(2-methoxypyrimidin-5-yl)methyl][(3-methylthiophen-2-yl)methyl]amine
3-[1-(adamantane-1-carbonyl)piperidin-4-yl]-1-(morpholin-4-yl)propan-1-one
[(3R,4R)-1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
8-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-ethyl-N-{[1-(2-phenylethyl)piperidin-4-yl]methyl}pyrimidine-5-carboxamide
3-[5-({[1-(pyrimidin-2-yl)piperidin-3-yl]amino}methyl)thiophen-3-yl]prop-2-yn-1-ol
2-[2-(1H-imidazol-4-yl)ethyl]-8-(4,4,4-trifluorobutanoyl)-2,8-diazaspiro[5.5]undecan-3-one
2-amino-4-(3-hydroxyphenyl)-6-(3-methylphenyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
1-(2-methoxyphenyl)-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-1H-pyrazole-4-carboxamide
N-(3-cyclohexyl-1H-1,2,4-triazol-5-yl)-2-phenylazetidine-1-carboxamide
6-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decane-4-carbonyl]-3-ethyl-3H-imidazo[4,5-b]pyridin-2-amine
N-[2-(diethylamino)ethyl]-1-ethyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
5-methyl-N-[(1-methyl-1,2,5,6-tetrahydropyridin-3-yl)methyl]-3-phenyl-1,2-oxazole-4-carboxamide
5-[(3R,4S)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidine-1-carbonyl]-1,2-dihydropyridin-2-one
1-{4-[(dimethylamino)methyl]-4-hydroxyazepan-1-yl}-3-(2-methyl-1H-indol-1-yl)propan-1-one
5-(1H-indazol-1-yl)-N-(pyridin-3-yl)furan-2-carboxamide
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxy-N-(prop-2-en-1-yl)benzamide
3-[(cyclohexylamino)methyl]-3-hydroxy-1-(2-methoxyethyl)piperidin-2-one
1-{1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-phenylpiperidin-4-yl}ethan-1-one
(3R,4R)-1-(3-chloro-4-fluorobenzoyl)-3-methyl-4-(oxan-4-yl)piperidin-4-ol
2-{4-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-1H-1,2,3-triazol-1-yl}ethan-1-amine
4-[2-(azepan-1-yl)propanoyl]-1-(4-methylphenyl)piperazin-2-one
3-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]-3,9-diazaspiro[5.5]undecane