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2-[4-(2-amino-6-methylpyrimidin-4-yl)-1-[(4-methoxy-3-methylphenyl)methyl]piperazin-2-yl]ethan-1-ol
4-(2-{3-[(4,4-difluoropiperidin-1-yl)methyl]phenoxy}ethyl)morpholine
1-{3-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-oxopropyl}-6-methyl-1,2-dihydropyridin-2-one
5-[4-(hydroxymethyl)piperidine-1-carbonyl]-1-[2-(4-methoxyphenyl)ethyl]piperidin-2-one
({3-[(2R,5S)-2,5-dimethylpyrrolidine-1-carbonyl]pyrazolo[1,5-a]pyrimidin-6-yl}methyl)diethylamine
(1R,3S)-3-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}cyclopentan-1-amine
2-{4-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1-(thiophen-3-ylmethyl)piperazin-2-yl}ethan-1-ol
4-{[2-(3,4-dimethoxyphenyl)ethyl]amino}-N,5-dimethyl-N-(propan-2-yl)thieno[2,3-d]pyrimidine-6-carboxamide
4-[(2-methoxyphenyl)methyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-(4-methoxyphenyl)-4-{[2-(piperidin-1-yl)pyrimidin-5-yl]methyl}piperazin-2-one
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-[2-(methylsulfamoyl)ethyl]acetamide
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-{2-[(2-methoxyethyl)(methyl)amino]acetyl}pyrrolidine-3-carboxylic acid
5-{[(2-fluorophenyl)methyl]amino}-N,N-dimethyl-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-hydroxy-3-methyl-N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]benzamide
2-{3-[(2-fluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}-1,3-thiazole-4-carboxamide
N-[2-methyl-2-(morpholin-4-yl)propyl]-3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-2-methylpyrrolidine
(1S,4S)-2-{5-chloro-2-[(1-cyclopentylpiperidin-4-yl)oxy]benzoyl}-2-azabicyclo[2.2.1]heptane
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
1-[(2,3-difluorophenyl)methyl]-3-hydroxy-3-{[methyl(2-methylprop-2-en-1-yl)amino]methyl}piperidin-2-one
6-(4-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)pyridine-3-carbonitrile
9-[(2R)-2-hydroxy-3-methylbutanoyl]-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
(8R,9aS)-2-(2,2-diphenylethyl)-8-hydroxy-octahydro-1H-pyrido[1,2-a]piperazine-1,4-dione
3-{1-[2-(cyclohex-1-en-1-yl)acetyl]piperidin-3-yl}-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
3-(2-hydroxyphenyl)-N-(4-phenylbutyl)-1H-pyrazole-5-carboxamide
4-(4-methoxyphenoxy)-1-[(2S)-pyrrolidine-2-carbonyl]piperidine
8-[2-(3-methoxyphenoxy)ethyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-4-methyl-2-(pyridin-3-yl)pyrimidine-5-carboxamide
2-(2-methoxyphenyl)-4-[(6-methylpyridin-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-(1-methylazepane-2-carbonyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
(2S,4S)-4-(3,4-difluorobenzamido)-N-ethyl-1-[(2E)-2-methylbut-2-en-1-yl]pyrrolidine-2-carboxamide
N-{3-[(4aS,8aR)-1-(2-aminoethyl)-2-oxo-decahydro-1,6-naphthyridin-6-yl]-3-oxopropyl}methanesulfonamide
1-(2-methyl-1-benzofuran-5-carbonyl)-2-propylpyrrolidine
1-{4-[hydroxy(1-methyl-1H-imidazol-2-yl)methyl]piperidin-1-yl}-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propan-1-one
3-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-1-(pyrrolidin-1-yl)propan-1-one
[(4-fluorophenyl)methyl](pyridin-2-ylmethyl)(pyridin-4-ylmethyl)amine
7-(6-ethyl-2-methylquinoline-4-carbonyl)-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
N-[2-(N-methylmethanesulfonamido)ethyl]-2-propylpyridine-4-carboxamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-4-(2,4-dioxoimidazolidin-1-yl)benzamide
1-(4-hydroxy-3-methylbenzoyl)-4-(hydroxymethyl)azepan-4-ol
(4aR,7aS)-1-[(4-methyl-1H-imidazol-5-yl)methyl]-4-(4,4,4-trifluorobutanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(2H-1,3-benzodioxol-5-yl)-N-[(1-propylpiperidin-3-yl)methyl]acetamide
6-chloro-2-methyl-N-[2-(1-methylpiperidin-3-yl)ethyl]imidazo[1,2-a]pyridine-3-carboxamide
N-benzyl-3-({[1-(1,3-dimethyl-1H-pyrazol-4-yl)ethyl]amino}methyl)-N-methylimidazo[1,2-a]pyridine-2-carboxamide
7-(1,3-benzothiazol-2-yl)-4-[(5-methylthiophen-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
[(8-methoxyquinolin-5-yl)methyl](methyl)({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)amine
N-(5-methyl-1,3,4-thiadiazol-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carboxamide
2-[2-(pyridin-2-yl)ethyl]-9-(1,3-thiazole-4-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
3-cyclohexyl-4-(prop-2-en-1-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one