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N-{[3-(cyclohex-3-en-1-ylmethoxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)furan-2-carboxamide
methyl 4-({9-methoxy-7-[4-(methylsulfanyl)phenyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}methyl)benzoate
4-(3-fluorophenoxy)-1-[2-(pyridin-3-yl)acetyl]piperidine-4-carboxylic acid
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
7-fluoro-N,2-dimethyl-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]quinoline-4-carboxamide
1'-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-cyclopentyl-4-{2-methoxy-4-[3-(methoxymethyl)pyrrolidine-1-carbonyl]phenoxy}piperidine
1-methanesulfonyl-4-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-1,4-diazepane
1-[4-(2-ethoxyphenyl)piperazin-1-yl]-3-(1-methyl-1H-pyrazol-5-yl)propan-1-one
1-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-methyl-2-phenylpropan-1-one
2-(2-phenyl-1H-imidazol-1-yl)-1-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]ethan-1-one
N-(1-ethyl-1H-1,2,3-triazol-4-yl)-2-[4-(4-methyl-1,4-diazepan-1-yl)-6-oxo-1,6-dihydropyridazin-1-yl]acetamide
2-amino-4-(4-ethoxy-3-methoxyphenyl)-6-(1-methyl-1H-pyrrol-3-yl)pyridine-3-carbonitrile
N-(1-methyl-1H-1,2,4-triazol-3-yl)-3-{[4-(1H-pyrazol-1-ylmethyl)piperidin-1-yl]methyl}benzamide
4-(1-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}azetidin-3-yl)pyridine
1-(2-methylpropyl)-N,N-bis(prop-2-en-1-yl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-[1-(4-cyclohexylpiperazine-1-carbonyl)-6-azaspiro[2.5]octane-6-carbonyl]-4,5,6,7-tetrahydro-1-benzofuran-4-one
(3S,4S)-1-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}-4-(piperidin-1-yl)pyrrolidin-3-ol
3-[(4-fluorophenyl)methyl]-5-[1-(5-methylthiophene-2-carbonyl)piperidin-4-yl]-5-(pyridin-3-yl)imidazolidine-2,4-dione
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-4-sulfamoylbenzamide
5-[2-(6-methoxynaphthalen-2-yl)morpholine-4-carbonyl]-2,3-dihydro-1H-pyrazol-3-one
N-(oxolan-2-ylmethyl)-4-({[3-(4H-1,2,4-triazol-4-yl)propyl]carbamoyl}amino)benzamide
2-{2-[3-(thiophen-3-ylmethyl)-1,2,4-oxadiazol-5-yl]ethyl}pyrazine
5-{1-methyl-2-oxo-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}-5-oxopentanamide
3-{2-[(4-chlorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}-N-(propan-2-yl)propanamide
3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)propanamide
4-benzyl-1-(3-chloro-4-hydroxybenzoyl)-3-ethyl-1,4-diazepan-5-one
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-5-methanesulfonyl-2-methylpyrimidin-4-amine
2-[7-(3,6-dimethylpyrazin-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetic acid
2-(4-fluorophenoxymethyl)-N-[2-(methylsulfanyl)ethyl]-1,3-oxazole-4-carboxamide
3-[4-(1-benzyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1λ6-thiolane-1,1-dione
N-{1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-phenylacetamide
N-ethyl-4-({1-[(2-oxo-2H-chromen-7-yl)oxy]propan-2-yl}amino)piperidine-1-carboxamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methyl-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
2-hydroxy-1-(4-{[3-(1H-imidazol-1-yl)propyl]amino}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl)ethan-1-one
3-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-[1-(thiophen-2-yl)propan-2-yl]benzamide
(4aR,7aS)-1-acetyl-4-(5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{[2-(diethylamino)pyridin-3-yl]methyl}-2-(2-methyl-1H-imidazol-1-yl)propanamide
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-4-cyano-N,1-dimethyl-1H-pyrrole-2-carboxamide
methyl[(6-methylpyridin-2-yl)methyl][(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]amine
3-[2-(3-methoxyphenyl)azetidine-1-carbonyl]-1,4,6-trimethyl-1,2-dihydropyridin-2-one
(3aS,6aR)-3-cyclopentyl-5-(pyridin-2-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-{1-[(1-phenyl-1H-pyrazol-4-yl)methyl]pyrrolidin-2-yl}-1,3-thiazole
N-cycloheptyl-4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperazine-1-carboxamide
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-4-(2,4-dioxoimidazolidin-1-yl)benzamide
2-(1H-pyrazol-1-yl)-N-{[5-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-3-yl]methyl}butanamide
5-[2-oxo-2-(pyridin-3-yl)acetyl]-N-phenyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
6-[(4aR,8aR)-7-cyclopentanecarbonyl-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]pyridine-2-carboxamide
1-[(2-methylphenyl)methyl]-4-(2-propyl-1,3-thiazole-4-carbonyl)piperazine
2-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl}-1-methyl-1H-indole