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6-methyl-N-[(4-methylphenyl)(pyridin-4-yl)methyl]-2-oxo-1,2-dihydropyridine-4-carboxamide
2-(2-hydroxyethyl)-N-[2-(2-methoxyphenoxy)phenyl]-3-oxopiperazine-1-carboxamide
4-({methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}methyl)-1H-pyrazole-3-carboxylic acid
(1S,5R)-6-(cyclobutylmethyl)-3-[4-(methylsulfanyl)benzoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[1-(1H-pyrazole-3-carbonyl)piperidin-4-yl]-3-(pyrrolidine-1-carbonyl)piperidine
2-({cyclopropyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)-6-methoxyphenol
3-chloro-4-fluoro-N-{3-[(pyridin-3-yl)amino]propyl}-1-benzothiophene-2-carboxamide
2-{4-[2-(3-fluorophenyl)azepane-1-carbonyl]piperidin-1-yl}acetamide
1-methyl-8-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
8-[(4-methyl-1H-imidazol-5-yl)methyl]-1-(3-methylbutyl)-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}-N,N-diethylacetamide
1-(1-ethyl-2-methyl-1H-indol-5-yl)-3,3-dimethylurea
4-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-1,4-oxazepane
4-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-5-ethyl-2-methylpyrimidine
methyl 2-{8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-(2-methoxyethyl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl}acetate
5-benzyl-4-(2-hydroxyacetyl)-1-(2-phenylphenyl)piperazin-2-one
7-[1-(2,3-dimethylphenyl)piperidin-4-yl]-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-[(1R,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-2-(1H-1,2,4-triazol-3-yl)benzamide
N-(3-hydroxy-3-phenylpropyl)-N-methyl-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamide
3-{[ethyl({[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl})amino]methyl}-5-methyl-1H-indole-2-carboxylic acid
4-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]benzene-1-sulfonamide
3-{2-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
N-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2-methylimidazo[1,2-a]pyrimidine-3-carboxamide
1-{3-fluoro-7-methylimidazo[1,2-a]pyridine-2-carbonyl}-N-(furan-2-ylmethyl)piperidine-4-carboxamide
4-cyclopropanecarbonyl-9-[(1-methylpiperidin-3-yl)methoxy]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-{1-[(4-ethoxyphenyl)methyl]-4-(1-propylpiperidin-4-yl)piperazin-2-yl}ethan-1-ol
(1R,3S)-N1,N1,2,2,3-pentamethyl-N3-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}cyclopentane-1,3-dicarboxamide
2-({4-[2-methoxy-5-(propan-2-yl)phenyl]-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl}oxy)acetic acid
3-(1,3-benzothiazol-2-yl)-3,9-diazaspiro[5.6]dodecan-10-one
N-{[2-(4-acetylpiperazin-1-yl)pyridin-3-yl]methyl}-2-(2-methyl-1H-indol-3-yl)acetamide
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-2-(1H-pyrazol-1-yl)acetamide
1-(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidin-1-yl)-3-(methylsulfanyl)propan-1-one
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
2-{[4-(1-{[(2-methyl-2H-1,2,3-triazol-4-yl)carbamoyl]methyl}-1H-pyrazol-4-yl)phenyl]sulfanyl}acetamide
1-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]-4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidine
1-(4-hydroxy-1,2,3,4-tetrahydroisoquinolin-2-yl)-4-(1H-1,2,4-triazol-1-yl)butan-1-one
2-[3-(dimethylamino)propyl]-9-[(2-methylpyrimidin-5-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
2-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-N-[3-methyl-1-(2-methylpropyl)-1H-pyrazol-5-yl]morpholine-4-carboxamide
2-(3-fluoro-4-methylphenyl)-N-methyl-N-[(3-methylthiophen-2-yl)methyl]acetamide
(1R,5R)-3-benzoyl-6-(2-propoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
N-[3-(dimethylcarbamoyl)-5-({[1-(2-fluorophenyl)propan-2-yl]amino}methyl)phenyl]pyridine-2-carboxamide
methyl[(1-methyl-1H-imidazol-2-yl)methyl]{[8-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}amine
N,N-dimethyl-3-(2-{[(1H-1,2,3,4-tetrazol-5-ylmethyl)carbamoyl]amino}phenyl)propanamide
N-methyl-6-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)pyridine-2-carboxamide
4-{[(3R,4S)-3-(dimethylamino)-4-propylpyrrolidin-1-yl]methyl}-1,5-dimethyl-1H-pyrrole-2-carbonitrile
3-cyclohexyl-N-methyl-N-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-1H-pyrazole-4-carboxamide
(4aS,8aS)-2-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-decahydroisoquinolin-4a-ol
4-[(4aR,8aS)-6-[4-(trifluoromethyl)benzoyl]-decahydro-1,6-naphthyridine-1-carbonyl]-1,2-dihydrophthalazin-1-one
2-{[(5-cyclopropyl-1H-pyrazol-3-yl)methyl](methyl)amino}-2-(2-fluoro-5-methoxyphenyl)acetic acid
1-[3-(4-fluorophenoxymethyl)piperidin-1-yl]-2-(4-methyl-1,4-diazepan-1-yl)ethan-1-one