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5-cyclopentyl-2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
1-[4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]-4-(oxolane-2-carbonyl)-1,4-diazepane
N-[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
(1S,5R)-3-{[2-(methylamino)-1,3-thiazol-4-yl]methyl}-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
5-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidine-1-carbonyl}-1H-indole
2-[2-methyl-4-(pyrrolidin-1-ylmethyl)phenoxy]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
2-(2-hydroxyethyl)-9-[3-(2-methoxyphenyl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
[(3R,4R)-1-(6-methylpyridazin-3-yl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
4-[4-(1-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]piperidine
1-{1-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-1-oxopropan-2-yl}pyrrolidin-2-one
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
(1S,5R)-3-[2-(3-chlorophenoxy)acetyl]-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
methyl[1-(4-methylpyridin-2-yl)propan-2-yl]{[5-(1H-pyrazol-5-yl)furan-2-yl]methyl}amine
8-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)-3-(2-ethylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-3-cyclopentaneamido-4-methylbenzamide
N-[(5-amino-1H-1,2,4-triazol-3-yl)methyl]-4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}benzamide
8-(3-hydroxypropanoyl)-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
(2S)-N-[4-(3-fluorophenyl)phenyl]-1-(1,2,4-oxadiazol-3-ylmethyl)pyrrolidine-2-carboxamide
3-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-1-(2-phenylethyl)urea
3-(azepan-1-ylmethyl)-N-[(1-methylpyrrolidin-3-yl)methyl]benzamide
4-methoxy-6-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
(2E)-N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(pyridin-2-yl)prop-2-enamide
4-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-N,N-dimethylpiperazine-1-sulfonamide
N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)oxane-2-carboxamide
5-phenyl-N-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)pyrazolo[1,5-a]pyrimidin-7-amine
5-methoxy-N-[(2-methyl-1,3-thiazol-4-yl)methyl]furan-2-carboxamide
6-methyl-2-(4-{[methyl({[2-(1H-pyrazol-1-yl)phenyl]methyl})amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
ethyl 3-{[5-(4-chloro-3,5-dimethylphenoxymethyl)-1,2-oxazol-3-yl]formamido}propanoate
2-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrazine
4-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-5-methyl-1-(4-methylphenyl)piperazin-2-one
1-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-[(cyclopropylmethyl)sulfanyl]ethan-1-one
5-(1-benzylpyrrolidin-2-yl)-3-(propan-2-yl)-1,2,4-oxadiazole
N-[(5-methylpyrazin-2-yl)methyl]-5-[1-(piperidin-1-yl)ethyl]furan-2-carboxamide
N-{[2-(3-chlorophenyl)-7-methylquinolin-3-yl]methyl}-2-(dimethyl-1H-1,2,4-triazol-1-yl)-N-(3-methoxypropyl)acetamide
N-benzyl-3-(3-chlorobenzoyl)piperidine-1-carboxamide
N-[1-(4-methyl-5-{[(2-methylphenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl)ethyl]-3-(4-methylphenyl)propanamide
1-[(1-{[4-(5-methylpyridin-2-yl)piperidin-4-yl]methyl}piperidin-3-yl)methyl]pyrrolidin-2-one
4-(1H-imidazol-1-yl)-N-(2-methanesulfonamidoethyl)benzamide
2-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
2-[(2S,3R)-2-amino-3-hydroxybutanoyl]-N-benzyl-N-methyl-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-(naphthalen-2-ylmethyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
(3R,5S)-1-benzyl-N3-(4-fluorophenyl)-N5-(3-methoxypropyl)piperidine-3,5-dicarboxamide
3-[4-(2,4-dimethylphenyl)piperazine-1-carbonyl]-1-[2-(2-methoxyphenyl)ethyl]-2,6-dimethyl-1,4-dihydropyridin-4-one
3-(1-ethyl-1H-1,2,4-triazol-3-yl)-1-[(8-methoxyquinolin-5-yl)methyl]-1-methylurea
N3-(2,1,3-benzothiadiazol-5-ylmethyl)-N1,N1,N3-trimethylpiperidine-1,3-dicarboxamide
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethylbenzamide
5,7-dimethyl-N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
3-chloro-N-[2-(diethylamino)ethyl]-4-[(1-methanesulfonylpiperidin-4-yl)oxy]benzamide
7-(5-methylthiophen-2-yl)-4-[6-(propan-2-yl)pyrimidin-4-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-hydroxyethan-1-one