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1-(azepan-1-yl)-3-{3-[({[3-(methylsulfanyl)phenyl]methyl}amino)methyl]phenoxy}propan-2-ol
9-methoxy-4-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-(pyridin-2-yl)acetamide
(1S,9R)-11-{pyrazolo[1,5-a]pyridine-7-carbonyl}-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
N-(2-{4-[(2-methyl-1H-imidazol-4-yl)methyl]morpholin-2-yl}ethyl)cyclohexanecarboxamide
methyl 2-(diethylsulfamoyl)-6-(3-phenylpropanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-benzyl-3-methyl-4-(1H-pyrazole-4-carbonyl)piperazin-2-one
1-{2-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}-2-(morpholin-3-yl)ethan-1-one
3-hydroxy-N-{[1-(2-methylpropyl)piperidin-3-yl]methyl}pyridine-2-carboxamide
N-(adamantan-1-yl)-5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}-1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
ethyl 4-[1-(4-{2-[(2S)-2-(methoxycarbonyl)pyrrolidin-1-yl]-2-oxoethyl}phenyl)piperidin-4-yl]piperazine-1-carboxylate
N-(2H-1,3-benzodioxol-5-yl)-5-(1H-pyrazol-4-yl)furan-2-carboxamide
8-fluoro-2-{[(oxolan-2-ylmethyl)(pyridin-4-ylmethyl)amino]methyl}quinolin-4-ol
4-{[(2R,3S,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}phenol
2-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
2-[(3R,4S)-3-amino-4-(5-methylfuran-2-yl)pyrrolidin-1-yl]propane-1,3-diol
2-[3,5-dimethyl-4-(2-methyl-1,3-benzothiazole-6-sulfonamido)-1H-pyrazol-1-yl]acetic acid
2-[methyl({[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl})amino]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
4-{2-ethyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}butanamide
(3R,4R)-1-{[5-(3-chlorophenyl)furan-2-yl]methyl}-4-(4-methylpiperazin-1-yl)piperidin-3-ol
3-ethyl-4-methyl-5-{1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-ylmethyl}-1H-pyrazole
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(1-propylpiperidin-4-yl)pyrrolidine-3-carboxylic acid
(1S,5R)-6-(propane-1-sulfonyl)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(3R)-N-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-1-azabicyclo[2.2.2]octan-3-amine
4-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-6-ethyl-1,2-dihydropyridin-2-one
2-{5-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
5-[(3R,4S)-3-amino-4-propylpyrrolidine-1-carbonyl]pyrazin-2-ol
2-{2-[2-oxo-5-(trifluoromethyl)-1,2-dihydropyridin-1-yl]acetyl}-2,7-diazaspiro[4.5]decan-6-one
2-amino-8-(2-methoxypyridin-3-yl)-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
ethyl 1-(3-phenylpropyl)-5-(1,2,5-thiadiazole-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-{1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]piperidine-3-carbonyl}azepane
1-(3-chloro-4-methoxyphenyl)-4-(thiomorpholine-4-carbonyl)pyrrolidin-2-one
(3aR,6aR)-2-benzyl-N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
N-(dimethyl-1H-1,2,4-triazol-3-yl)-4-[2-oxo-2-(pyrrolidin-1-yl)ethyl]piperazine-1-carboxamide
N,N-dimethyl-2-[(1S,5R)-6-[3-(5-methyl-1H-pyrazol-1-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
[1-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-3-propylpiperidin-3-yl]methanol
6-(benzyloxy)-1-(2-methylpropyl)-4-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)-1,4-diazepan-2-one
[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl](methyl)({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)amine
(1S,5R)-6-[(2-butyl-1H-imidazol-4-yl)methyl]-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
2-{4-[(4-methyl-1,4-diazepan-1-yl)methyl]phenyl}-6-(pyridin-4-yl)-3,4-dihydropyrimidin-4-one
N-{2-[(2-chlorophenyl)formamido]ethyl}-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
methyl 2-(N-methyl-1-{2-[methyl(2-phenylethyl)amino]-2,3-dihydro-1H-inden-2-yl}formamido)acetate
4-{[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]sulfonyl}-3,5-dimethyl-1H-pyrazole
N-(1,4-dioxan-2-ylmethyl)-6-ethyl-2-(pyrrolidin-1-yl)pyrimidin-4-amine
6-chloro-2-(3,3,3-trifluoropropyl)-1H-1,3-benzodiazole
2-(3,5-dimethoxyphenyl)-5-fluoro-N-methylpyrimidin-4-amine
2-(2-phenylethyl)-8-(1,3-thiazol-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-(2-chloro-6-fluorophenyl)-1-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]ethan-1-one
N-benzyl-5-{[3-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]methyl}pyrimidin-2-amine