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(3aR,5S,6S,7aS)-2-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-octahydro-1H-isoindole-5,6-diol
4-(4-methyl-1H-pyrazol-1-yl)-1-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxylic acid
1-{4-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]piperidin-1-yl}ethan-1-one
[(2S,4R)-1-methyl-4-{[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}pyrrolidin-2-yl]methanol
3-(1-butyl-1H-imidazol-2-yl)-1-(5-chloro-2-fluorobenzoyl)piperidine
2-{2-[(4-cyanopiperidin-1-yl)methyl]-4-(thiophen-2-yl)phenoxy}acetic acid
N-(1,3-dihydro-2-benzofuran-5-yl)-2-phenylmorpholine-4-carboxamide
N-{[7-chloro-5-(thiophen-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(2-methyl-1,3-thiazol-4-yl)acetamide
1-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)-3-(4-fluorophenoxymethyl)piperidine
N-(pyridin-2-ylmethyl)-1-[1-(pyrimidin-2-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
3-amino-1-{1-[3-(trifluoromethyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}propan-1-one
5-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]pyrazin-2-ol
N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-N-{2-[(2-methylprop-2-en-1-yl)oxy]phenyl}piperidine-1-carboxamide
(3R,4R)-1-[(2-methoxy-4-methylphenyl)methyl]-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
5-{[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]methyl}-2,1,3-benzothiadiazole
1-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-4-methyl-1,2,3,6-tetrahydropyridine
N-[(4-fluorophenyl)methyl]-3-[1-(3-methylthiophene-2-carbonyl)piperidin-4-yl]propanamide
(4S)-3,3,4-trimethyl-1-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)piperidin-4-ol
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-[(dimethylcarbamoyl)methyl]acetamide
N-[2-(2-fluorophenyl)-1-[1-(quinolin-7-ylmethyl)piperidin-4-yl]ethyl]-N,2-dimethylfuran-3-carboxamide
3-[(3S,7S,8aS)-3-(hydroxymethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-chloro-2-methylphenyl)urea
3-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}pyrrolidin-3-ol
2-cyclopropyl-8-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
2-methyl-2-[4-(morpholin-4-yl)-2-[(1-propylpyrrolidin-3-yl)amino]pyrimidin-5-yl]propanoic acid
N-[4-(2-methoxyphenyl)phenyl]-3-(2-methylpiperidin-1-yl)azetidine-1-carboxamide
1-{1-[(2R)-2-aminopropanoyl]piperidin-4-yl}-N-(2-phenylethyl)piperidine-4-carboxamide
5-{5-[2-(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)ethyl]-1,2,4-oxadiazol-3-yl}-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
2-(2-{[(2-methoxyethyl)(methyl)amino]methyl}phenyl)-6-(pentafluoroethyl)-3,4-dihydropyrimidin-4-one
2,6-dimethyl-4-{3-[1-(oxolan-2-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyridine
7-[(3-methylphenyl)methyl]-2-(pyrimidin-2-yl)-2,7-diazaspiro[4.5]decane
2-{2-[(3R,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-2-oxoethyl}-3-phenylcyclopent-2-en-1-one
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-1-[(2-fluorophenyl)methyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
(3E)-N-benzyl-N-(3-hydroxy-2-methylpropyl)hex-3-enamide
4-{5-[(4-methanesulfonyl-1,4-diazepan-1-yl)methyl]-1,2,4-oxadiazol-3-yl}benzoic acid
N-[(4-fluorophenyl)methyl]-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
2-({5-[2-amino-3-cyano-6-(2,4-dimethylphenyl)pyridin-4-yl]pyrimidin-2-yl}amino)acetic acid
1-[1-(3-aminopropyl)-1H-1,2,3-triazole-4-carbonyl]-4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-5-one
5-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine-1-carbonyl}-2-(pyridin-3-yl)pyrimidine
N-[(5-chlorothiophen-2-yl)methyl]-1-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
3-[1-({2-[3-(1H-imidazol-1-yl)propoxy]-3-methoxyphenyl}methyl)pyrrolidin-2-yl]-4-methyl-1,2,5-oxadiazole
(1s,4s)-4-{4-[(2S)-2-(piperidine-1-carbonyl)pyrrolidine-1-carbonyl]-1H-1,2,3-triazol-1-yl}cyclohexan-1-amine
(2S,4R)-4-(4-{2-[(4-cyanophenyl)formamido]propan-2-yl}-1H-1,2,3-triazol-1-yl)-N-methylpyrrolidine-2-carboxamide
1-(2-chloropyridin-3-yl)-3-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)urea
methyl 4-{1-[(1-methanesulfonylpiperidin-3-yl)methyl]-1H-imidazol-2-yl}benzoate
methyl 3-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]-7-oxo-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}(methyl)(oxolan-3-ylmethyl)amine
3-(2-methoxyphenyl)-N-methyl-N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-1H-pyrazole-5-carboxamide
(1S,5R)-6-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-{5-[(ethylcarbamoyl)amino]-2-methoxyphenyl}-2-methoxyacetamide