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5-{[benzyl(methyl)amino]methyl}-N-methyl-N-(pyridin-3-ylmethyl)-1,2-oxazole-3-carboxamide
4-[4-(azetidine-1-carbonyl)-2-chlorophenoxy]-1-methanesulfonylpiperidine
N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]-3-phenoxypropanamide
N-[1-(5-methyl-1,3,4-oxadiazol-2-yl)ethyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}cyclobutanamine
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-(naphthalen-2-yloxy)propanamide
3-{1-[2-(dimethylamino)-6-ethylpyrimidin-4-yl]piperidin-3-yl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(2S)-2-amino-1-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propan-1-one
4-(4-fluorophenyl)-1-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidin-4-ol
N-[2-(4-methylmorpholin-2-yl)ethyl]isoquinoline-5-carboxamide
2-chloro-4-{[({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)amino]methyl}phenol
3-amino-1-{[2-(4-methoxyphenyl)imidazo[1,2-a]pyridin-3-yl]methyl}pyrrolidine-3-carboxylic acid
N-(2,3-difluorophenyl)-2-(5-methyl-1,2-oxazol-3-yl)piperidine-1-carboxamide
N'-(3-chloro-4-fluorophenyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-propylbutanediamide
(2S,4S)-4-cyclopentaneamido-N,N-diethyl-1-[(4-methyl-1H-imidazol-5-yl)methyl]pyrrolidine-2-carboxamide
{[6-chloro-2-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}(1H-imidazol-2-ylmethyl)methylamine
methyl 3-chloro-4-[(cyclobutylcarbamoyl)amino]benzoate
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}acetamide
[(3R,4R)-1-(3,6-dimethyl-1-benzofuran-2-carbonyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-2-(pyridin-3-yl)acetamide
dimethyl({[5-(3-phenoxyphenyl)-1,2,4-oxadiazol-3-yl]methyl})amine
1-{2-[2-(2-butyl-5-chloro-1H-imidazol-4-yl)-1H-imidazol-1-yl]ethyl}imidazolidin-2-one
4-(1-butyl-1H-imidazol-2-yl)-1-[3-(thiophen-3-yl)-1H-pyrazole-5-carbonyl]piperidine
4-hydroxy-N-[2-(5-methylthiophen-2-yl)ethyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
1-{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidine-4-carbonitrile
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}benzamide
5-methyl-1-phenyl-4-[1-(thiophen-2-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1H-pyrazole
2-{4-[3-(2-hydroxyethyl)-4-methylpiperazin-1-yl]-6-methylpyrimidin-2-yl}phenol
5-[benzyl(methyl)amino]-2-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-2,3-dihydropyridazin-3-one
N-ethyl-2-(1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-{[2-(prop-2-en-1-yloxy)phenyl]methyl}acetamide
methyl 3-({[2-(methylsulfanyl)-1,3-thiazol-4-yl]formamido}methyl)-5-propanamidobenzoate
1-[5-(5-ethyl-1,3,4-oxadiazol-2-yl)-2-methoxyphenyl]-3-(oxolan-2-ylmethyl)urea
4-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]butan-1-one
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-7-fluoro-2-methylquinoline-4-carboxamide
N-[(3R,4R)-3-hydroxy-1-[4-(thiophen-2-yl)butanoyl]piperidin-4-yl]pyridine-2-carboxamide
2-tert-butyl-5-[4-(pyridin-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]pyrimidin-4-ol
1-(4-chloro-1H-pyrazole-3-carbonyl)-3-(4-methoxy-3,5-dimethylbenzoyl)piperidine
N4-{[1-(4-fluorophenyl)cyclopentyl]methyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
5-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidine-1-carbonyl]-1-phenyl-1H-1,2,3-triazole
N-methyl-N-[2-(pyridin-4-yl)ethyl]-7H-pyrrolo[2,3-d]pyrimidin-4-amine
8-fluoro-2-{4-[2-(methylsulfanyl)ethyl]piperazine-1-carbonyl}quinoline
2-[4-(1-phenylpiperidin-4-yl)-1-(thiophen-2-ylmethyl)piperazin-2-yl]ethan-1-ol
3-[3-(1-methoxyethyl)phenyl]-5-(morpholine-4-sulfonyl)benzoic acid
1'-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
2-(1-benzyl-1H-pyrazol-4-yl)-2-{[2-(1H-imidazol-1-yl)ethyl](methyl)amino}acetic acid
6-methyl-2-(2-methylpyrimidin-4-yl)-5-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
6-ethyl-N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-2-methylquinoline-4-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-4-(2,4-dioxoimidazolidin-1-yl)benzamide
2-(3-fluoropyridine-4-carbonyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
2-{2-[1-(2-cyclopentylacetyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide