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2-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[3-(3-fluorophenyl)phenyl]-1-(1H-pyrrole-3-carbonyl)piperidine-4-carboxamide
1-(5-{[3-(methoxymethyl)piperidin-1-yl]methyl}imidazo[2,1-b][1,3]thiazole-6-carbonyl)azocane
N-ethyl-5-{2-[2-(pyridin-2-yl)ethyl]piperidine-1-carbonyl}pyrimidin-2-amine
2-(3-methylbut-2-en-1-yl)-8-(3-phenyl-1,2,4-oxadiazol-5-yl)-2,8-diazaspiro[4.5]decan-3-one
methyl 3-[(4-methoxy-2,3-dimethylphenyl)methyl]-9-[(1-methyl-5-oxopyrrolidin-3-yl)methoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(2S)-2-amino-1-(3,3-diphenylpiperidin-1-yl)propan-1-one
9-(isoquinoline-5-carbonyl)-1,4,9-triazaspiro[5.5]undecan-5-one
3-cyclohexyl-2-oxo-1-(pyrimidin-2-ylmethyl)-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[2-(4-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]piperidin-2-one
N-[(5-chloro-2-propoxyphenyl)methyl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxamide
2-cyclopropyl-5-(3-{[4-(propan-2-yl)phenyl]amino}piperidine-1-carbonyl)-3,4-dihydropyrimidin-4-one
N-[4-chloro-3-({methyl[(4-methyl-1H-imidazol-2-yl)methyl]carbamoyl}amino)phenyl]-2-methoxyacetamide
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-2-(2,5-dioxoimidazolidin-1-yl)acetamide
{3-[(3-methoxyphenyl)methyl]-1-{[2-(trifluoromethyl)phenyl]methyl}piperidin-3-yl}methanol
2-methoxy-N-[3-(8-methoxyquinolin-5-yl)phenyl]acetamide
{[4-(difluoromethoxy)phenyl]methyl}({[2-(2-methylphenoxy)pyridin-3-yl]methyl})amine
methyl 1-ethoxy-8-{2-[(5-methyl-1H-1,3-benzodiazol-2-yl)sulfanyl]acetyl}-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
3-cyclohexyl-1-(2-hydroxyethyl)-2-oxo-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
(2-methoxyethyl)[(4-methyl-1H-imidazol-5-yl)methyl][(1-methyl-1H-pyrazol-4-yl)methyl]amine
2-{4-[2-(2-methoxyphenyl)acetamido]-1H-pyrazol-1-yl}-N-[1-(thiophen-2-yl)propyl]acetamide
1-(4-ethylpiperazin-1-yl)-3-[2-methoxy-4-({methyl[(3-methylpyridin-2-yl)methyl]amino}methyl)phenoxy]propan-2-ol
4-{[4-(2-phenylpropyl)-1H-1,2,3-triazol-1-yl]methyl}-1,3-thiazol-2-amine
(3S)-4-(2-chloropyridine-4-carbonyl)-3-ethylmorpholine
propan-2-yl (1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonane-6-carboxylate
1-{4-[4-(2-hydroxypropan-2-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-2-(4-methylphenyl)ethan-1-one
7-[2-(7-chloro-2,3-dihydro-1,4-benzodioxin-6-yl)acetyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
3-chloro-N-[2-(dimethylamino)ethyl]-4-({1-[3-(methylsulfanyl)propanoyl]piperidin-4-yl}oxy)benzamide
7-(3,3-diphenylpiperidin-1-yl)-[1,2,4]triazolo[4,3-c]pyrimidin-5-amine
N-[(3,4-dimethoxyphenyl)methyl]-N-(pyridin-2-ylmethyl)propanamide
ethyl 2-(1-{2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]acetamido}cyclohexyl)acetate
(4aS,8aR)-2-{4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]benzoyl}-decahydroisoquinoline
3-(4-methyl-1,3-thiazol-5-yl)-N-[2-(pyrrolidin-1-yl)ethyl]propanamide
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-4-(1H-pyrazol-1-yl)benzene-1-sulfonamide
2-{4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine
{4-[(dimethylamino)methyl]-1-(5-propyl-1,3,4-oxadiazol-2-yl)piperidin-4-yl}methanol
5-[(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)methyl]-2,1,3-benzothiadiazole
1-(4-methoxybenzoyl)-4-(thiophen-3-ylmethyl)piperazine
9-methoxy-4-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(2S)-1-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(methylamino)propan-1-one
N-(furan-2-ylmethyl)-1-(5,6,7,8-tetrahydroquinoline-3-carbonyl)piperidine-4-carboxamide
4-(1-{[5-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-3-yl]methyl}-1H-imidazol-2-yl)pyridine
[(3-ethyl-1,2-oxazol-5-yl)methyl]({[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl})methylamine
N-(2-{[(8-fluoro-4-hydroxyquinolin-2-yl)methyl]amino}ethyl)-N-methylmethanesulfonamide
5-{3-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-3-oxopropyl}-5-{[4-(methylsulfanyl)phenyl]methyl}pyrrolidin-2-one
5-[(4-hydroxyphenyl)methyl]-N-(2-methoxyethyl)-1-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-(2-methylpyridin-4-yl)pyrrolidin-3-yl]-1-(methoxymethyl)cyclobutane-1-carboxamide
N-(2H-1,3-benzodioxol-5-yl)-4-{2-[benzyl(methyl)carbamoyl]ethyl}piperidine-1-carboxamide
2-[4-({4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}methyl)phenyl]ethan-1-amine
3-(2-{[4-(methylsulfanyl)phenyl]methyl}-5-oxopyrrolidin-2-yl)-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]propanamide