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1-({1-[(3-methoxyphenyl)methyl]-1H-1,2,4-triazol-5-yl}methyl)-1,2-dihydropyridin-2-one
3-{1-[3-(4H-1,2,4-triazol-4-yl)benzoyl]pyrrolidin-2-yl}pyridine
N-(oxolan-2-ylmethyl)-1-propyl-N-(pyridin-2-ylmethyl)-1H-pyrazole-5-carboxamide
3-(cyclobutylmethoxy)-5-(1,1-dioxo-1λ6-thiomorpholine-4-carbonyl)benzoic acid
N-[1-(2-methoxyphenyl)-5-oxopyrrolidin-3-yl]-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-5-oxo-1-phenyl-2,5-dihydro-1H-pyrazole-3-carboxamide
3-{[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]methyl}pyridin-2-amine
methyl 3-({[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}carbamoyl)propanoate
2-{5-[(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)methyl]-1-(2-methylphenyl)-1H-1,2,4-triazol-3-yl}acetamide
2,3-dimethyl-6-[3-(3-methylphenyl)piperidine-1-carbonyl]-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
(2S,4R)-4-amino-N-ethyl-1-[5-(3-methoxyphenyl)furan-2-carbonyl]pyrrolidine-2-carboxamide
5-{[3-(1H-1,3-benzodiazol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,3-dimethylimidazolidine-2,4-dione
2-{[2-(2-butyl-4-methyl-3-oxopiperazine-1-carbonyl)phenyl]amino}acetic acid
3-({2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}carbonyl)-4,5,6,7-tetrahydro-1-benzofuran-4-one
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-1-(oxan-4-yl)piperidine-4-carboxamide
5-{1-[(2,4-difluorophenyl)methyl]-4-hydroxypiperidin-4-yl}-N-(oxolan-2-ylmethyl)-1-benzofuran-2-carboxamide
1-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]-4-(3-methylpyridin-4-yl)-1,4-diazepane
5-{[butyl(furan-2-ylmethyl)amino]methyl}-4-chloro-N,N-dimethyl-1,3-thiazol-2-amine
4-(hydroxymethyl)-1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}piperidin-4-ol
dimethyl({2-[2-(1-{2-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-yl)-1H-imidazol-1-yl]ethyl})amine
3-methoxy-1-{2-[3-(3-methylthiophene-2-carbonyl)piperidin-1-yl]-2-oxoethyl}-1,2-dihydropyridin-2-one
8-fluoro-6-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)-3,4-dihydro-2H-1,4-benzoxazin-3-one
1-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-[5-(4-fluorophenyl)-2H-1,2,3,4-tetrazol-2-yl]ethan-1-one
4-(3-hydroxy-3-methylbutyl)-N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]benzamide
2-(2,3-dihydro-1-benzofuran-5-carbonyl)-6-methyl-5-(5-methyl-1,2,4-oxadiazol-3-yl)-1,2,3,4-tetrahydro-2,7-naphthyridine
N-[2-(pyridin-4-yl)ethyl]-2,3-dihydro-1,4-benzodioxine-5-carboxamide
[2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl]{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}amine
4-(piperidin-3-yl)-N-[2-(trimethyl-1H-pyrazol-1-yl)ethyl]benzamide
2-[4-(3-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-3-methylpyridine
[(2-chloro-6-fluorophenyl)methyl](ethyl){[2-(methylsulfanyl)pyrimidin-5-yl]methyl}amine
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-1-[3-(4-fluorophenyl)phenyl]piperidin-4-amine
3-[1-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperidin-3-yl]-N-[(5-methylfuran-2-yl)methyl]propanamide
N-methyl-3-{[(4-methylphenyl)methyl]amino}-N-[2-(oxan-4-yl)ethyl]benzamide
1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-4-cyclopentyl-1,4-diazepane
1-[3-(3-fluorophenyl)phenyl]-3-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}urea
3-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-1-[3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]urea
(4aR,7aS)-1-(cyclopropylmethyl)-4-[2-(3-methyl-6-oxo-1,6-dihydropyridazin-1-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-6-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
N-methyl-1-[5-(propan-2-yl)thiophene-3-carbonyl]-N-[2-(pyridin-2-yl)ethyl]piperidin-3-amine
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetamide
3-[4-(4-chlorophenyl)-1H-pyrazol-5-yl]-1-[(2,3,4-trimethoxyphenyl)methyl]piperidine
1-(3-chloro-2-methylphenyl)-3-{[2-(dimethylamino)pyridin-3-yl]methyl}urea
N-[1-(4-methanesulfonylphenyl)ethyl]-1-(methoxymethyl)cyclobutane-1-carboxamide
1-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(thiophen-2-yl)propan-1-one
(1S,5R)-6-(2,6-dimethylpyrimidine-4-carbonyl)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-[2-(2-methylpiperidin-1-yl)ethyl]pyridin-2-amine
2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)acetamide
N-{2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}pyrimidin-4-amine
5-[(2-amino-5-ethylpyrimidin-4-yl)amino]-2,2-dimethylpentan-1-ol
2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-methyl-N-[(4-phenoxyphenyl)methyl]acetamide