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4-methyl-3-{[methyl({[3-(methylsulfanyl)phenyl]methyl})carbamoyl]amino}-N-(propan-2-yl)benzamide
N-[5-(dimethylamino)-2-methylphenyl]-4-[(3-fluorophenyl)methyl]-3-oxopiperazine-1-carboxamide
1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4-[(2-fluorophenyl)methyl]-1,4-diazepane
{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}(methyl)[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amine
N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
7-{4-[(3-fluorophenyl)methyl]-1,4-diazepane-1-carbonyl}-1,3-diazepane-2,4-dione
4-(1H-pyrazol-1-yl)-1-(pyrrolidine-1-sulfonyl)piperidine-4-carboxylic acid
(3aS,6aS)-5-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]-1-methyl-octahydropyrrolo[3,4-b]pyrrole
3-(2-{8-cyclopropyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}-2-oxoethyl)imidazolidine-2,4-dione
5-{[(2-methoxynaphthalen-1-yl)methyl]amino}-1-methyl-N-(pyridin-4-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-(2-methoxy-5-methylphenyl)-3-(1H-pyrazol-4-yl)-4H-1,2,4-triazole
5-{10,10-dichlorotricyclo[7.1.0.04,6]decan-5-yl}-3-ethyl-1,2,4-oxadiazole
(1R,3S)-7-[2-(4-fluorophenoxy)ethyl]-3-methoxy-3-methyl-7-azaspiro[3.5]nonan-1-ol
(3aS,6aS)-N-[5-chloro-2-(1H-1,2,4-triazol-1-yl)phenyl]-octahydropyrrolo[2,3-c]pyrrole-1-carboxamide
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)amine
ethyl 2-{[7-(2-methoxybenzamido)-1,2,3,4-tetrahydroisoquinoline-2-carbonyl]amino}acetate
N-[(1-{[1-(propan-2-yl)-1H-pyrrol-3-yl]methyl}piperidin-4-yl)methyl]cyclopropanesulfonamide
1-cyclopropyl-N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
4-{[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]methyl}-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
4-{3-[1-(but-3-en-1-yl)-1H-pyrazol-3-yl]phenyl}-3-methylpyridine
(1S,5R)-3-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(4-{[(1R,2R,4S)-bicyclo[2.2.1]heptan-2-yl]amino}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
3-(4-methoxyphenoxymethyl)-1-(4-methyl-1,3-thiazol-2-yl)piperidine
2-[4-(1H-pyrazol-5-yl)phenyl]pyridine-4-carboxamide
2-(5,5-dimethyl-2,4-dioxo-1,3-oxazolidin-3-yl)-N-[1-(4-fluorophenyl)ethyl]-N-methylacetamide
1-[(3S,4R)-1-(2-aminopyridine-4-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
2-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]methyl}-5-ethylpyridine
N,N-diethyl-5-{1-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]pyrrolidin-2-yl}thiophene-2-carboxamide
3-(3-hydroxy-3-methylbutyl)-N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}benzamide
2-{9-[(2E)-2-methylbut-2-en-1-yl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}propanoic acid
(4S)-3-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(propan-2-yl)-1,3-oxazolidin-2-one
N-[(2-chloro-6-fluorophenyl)methyl]-1-methyl-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carboxamide
3-hydroxy-3-({[2-(4-methyl-1H-pyrazol-1-yl)ethyl]amino}methyl)-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
4-(1-{[3-(dimethylamino)phenyl]methyl}-1H-imidazol-2-yl)phenol
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-6-(piperidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
3-[(3R,4S)-1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
1,4-dimethyl-9-[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]-1,4,9-triazaspiro[5.5]undecane
1-(4-{2-[5-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]-1H-imidazol-1-yl}-2-methylphenyl)pyrrolidin-2-one
N,1,3-trimethyl-N-(1,3-thiazol-2-ylmethyl)-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
1-[2-methoxy-4-({[3-(pyridin-3-yloxy)propyl]amino}methyl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
5-(3,4-dimethylphenoxymethyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
3-hydroxy-3-({methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amino}methyl)-1-(3-phenylpropyl)piperidin-2-one
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]isoquinoline-5-carboxamide
1-(2,1-benzoxazole-3-carbonyl)-4-benzyl-3-ethyl-1,4-diazepan-5-one
(1-{1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-3-yl}piperidin-4-yl)methanol
3-amino-1-{[3-(3,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidine-3-carboxylic acid
1-[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-N-[1-(pyrimidin-4-yl)ethyl]piperidin-4-amine
(2R,3S,6R)-3-(3,5-difluorophenyl)-5-(6-methylpyrimidin-4-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
6-(2-methylpropyl)-4-(3-propylmorpholine-4-carbonyl)-1,2-dihydropyrimidin-2-one
(3S,4R)-4-(4-fluorophenyl)-1-[3-(methylsulfanyl)propyl]pyrrolidine-3-carboxylic acid