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1-{1-[3-(2-methylpropyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]ethyl}-2-(propan-2-yl)-1H-imidazole
1-{4-[4-(2-chlorophenyl)piperidin-4-yl]pyrimidin-2-yl}piperidin-4-ol
2-[(5-methylpyrazin-2-yl)methyl]-9-[2-(thiophen-3-yl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[(6-methylpyridin-2-yl)methyl]-6-(3-phenyl-1,2-oxazole-5-carbonyl)-6-azaspiro[2.5]octane-1-carboxamide
N-cyclopropyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-phenylpyrimidine-5-carboxamide
6-(piperidin-4-yl)-2-(thiophen-2-yl)-3,4-dihydropyrimidin-4-one
1-[(3,4-dimethoxypyridin-2-yl)methyl]-2-(furan-2-yl)azepane
(1R,2R)-2-[3-(2-methyl-1,3-thiazol-4-yl)-5-(pyridin-3-ylmethyl)-1H-1,2,4-triazol-1-yl]cyclohexan-1-ol
3-(4-chloro-1H-pyrazol-1-yl)-1-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]propan-1-one
(3R,4R)-4-amino-1-(1-ethyl-3,5-dimethyl-1H-pyrazole-4-carbonyl)piperidin-3-ol
1-[2-(4-chlorophenyl)ethyl]-5-(3-ethyl-1,2,4-oxadiazol-5-yl)piperidin-2-one
N-[(3S,4R)-1-(1,1-dioxo-1λ6-thiane-4-carbonyl)-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
2-[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]-1-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-1H-imidazole
5,6-dimethyl-2-[2-(3-methyl-3-phenylpiperidin-1-yl)-2-oxoethyl]-2,3-dihydropyridazin-3-one
2-(5-chloro-6-methyl-1-benzofuran-3-yl)-N-[2-(dimethylsulfamoyl)ethyl]acetamide
3-[1-methyl-3-(pyridin-2-yl)-1H-pyrazol-5-yl]-1-[2-(pyrrolidine-1-sulfonyl)ethyl]urea
2-{[7-(2-cyclopropylpyrimidine-5-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}ethan-1-ol
2-(2-ethyl-1H-1,3-benzodiazol-1-yl)-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]butanamide
5-cyclopropyl-N-[2-(diethylamino)ethyl]-N-ethyl-1-[4-(2-fluorophenyl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
3-methoxy-1-{2-oxo-2-[4-(piperidine-1-carbonyl)piperidin-1-yl]ethyl}-1,2-dihydropyridin-2-one
1-cyclohexyl-5-[(2-methoxyethoxy)methyl]-3-methyl-1H-1,2,4-triazole
2-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)pyridin-3-ol
8-(2-cyclopropylpyrimidine-5-carbonyl)-2-[2-(dimethylamino)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
(4aR,8aS)-1-(2H-1,3-benzodioxol-5-ylmethyl)-6-(furan-2-carbonyl)-decahydro-1,6-naphthyridine
N-[2-(1-methylpyrrolidin-2-yl)ethyl]-6-(morpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
1,3,6-trimethyl-N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-pyrazolo[3,4-b]pyridine-4-carboxamide
ethyl 3-(2-methoxyethyl)-1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidine-3-carboxylate
3-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-4-[(5-methylfuran-2-yl)methyl]piperazin-2-one
5-[2-(aminomethyl)morpholine-4-carbonyl]-N-phenylpyrimidin-2-amine
[1-(2,6-diaminopyrimidin-4-yl)-4-[(3-fluorophenyl)methyl]piperidin-4-yl]methanol
1'-(2,1,3-benzoxadiazol-4-ylmethyl)-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-[2-({1-[3-(1H-pyrazol-1-yl)phenyl]piperidin-4-yl}amino)ethyl]-1,3-oxazinan-2-one
2-(7-methyl-1H-indol-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
(2S,4R)-1-[(2-chlorophenyl)methyl]-N-(propan-2-yl)-4-({[4-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
5-oxo-1-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}pyrrolidine-3-carboxylic acid
7-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-N,N,2-trimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-methyl-3-{[4-(pyridin-3-ylmethoxy)piperidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
4-{3-[1-(3-methylpyridin-4-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]pyridin-2-yl}morpholine
N-[(5-ethylpyridin-2-yl)methyl]-2,6-dihydroxy-N-methylbenzamide
{3-[(3-chlorophenyl)methyl]-1-(1-propylpiperidin-4-yl)piperidin-3-yl}methanol
4-[(dimethylamino)methyl]-1-[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperidin-4-ol
N-cyclopropyl-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]acetamide
N-(1,4-dioxan-2-ylmethyl)-1,3-dimethyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-1-{4-[(pyrimidin-2-yl)amino]piperidin-1-yl}ethan-1-one
N-[(3R,4S)-4-cyclopropyl-1-(2-methoxyethyl)pyrrolidin-3-yl]-3-methoxybenzene-1-sulfonamide
3-(2-amino-4-methyl-6-{methyl[2-(pyridin-4-yl)ethyl]amino}pyrimidin-5-yl)propanoic acid
2-[3-(4-methylphenyl)-1H-pyrazol-4-yl]-1H-1,3-benzodiazole-5-carbonitrile
1-(2,3-dihydro-1H-inden-2-yl)-4-(1H-1,2,4-triazole-5-carbonyl)-1,4-diazepan-6-ol
1-(4-fluoro-2-methylphenyl)-4-{4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}piperidine
4-(2-methyl-1-phenyl-1H-1,3-benzodiazole-5-carbonyl)-1,4-oxazepan-6-ol