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N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]-2-(5-methyl-2H-1,2,3,4-tetrazol-2-yl)acetamide
1-(4-hydroxy-1,2,3,4-tetrahydroisoquinolin-2-yl)-3-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]propan-1-one
(5-{3-[2-methyl-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidine-1-carbonyl}furan-2-yl)methanol
(3S,4R)-1-[4-(1H-imidazol-1-yl)benzoyl]-4-methylpiperidine-3,4-diol
2-hydroxy-1-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}-2-phenylethan-1-one
(3S,9aR)-8-(4-methoxybenzoyl)-3-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(2R,3S,6R)-3-(3,5-difluorophenyl)-N-ethyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxamide
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-1H-pyrrole-2-carboxamide
3,5-dimethyl-1-(1-{2-phenylimidazo[1,2-a]pyridine-6-carbonyl}azetidin-3-yl)-1H-pyrazole
5-{4-[6-methyl-2-(pyridin-3-yl)pyrimidin-4-yl]piperazin-1-yl}-2,3-dihydropyridazin-3-one
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-3-[(1-methanesulfonylpiperidin-4-yl)oxy]benzamide
7-(cyclopropylmethyl)-2-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-2,7-diazaspiro[4.5]decan-6-one
4-{5-butyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-6-methoxypyrimidin-2-amine
5-[(isoquinolin-5-yloxy)methyl]-N-[1-(3-methylpyridin-2-yl)propan-2-yl]-1,2-oxazole-3-carboxamide
4-(1H-imidazol-1-ylmethyl)-1-{pyrazolo[1,5-a]pyridine-7-carbonyl}piperidin-4-ol
1-{4-[6-(1-hydroxyethyl)pyridin-2-yl]phenyl}-3-(propan-2-yl)urea
1-[5-(7-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)-2-methylphenyl]imidazolidin-2-one
1-[1-(oxan-4-yl)piperidine-3-carbonyl]-4-(pyridin-3-yl)piperidin-4-ol
2,6,8-trimethyl-N-[(3R,4R)-4-(morpholin-4-yl)oxolan-3-yl]quinoline-4-carboxamide
3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-(1-methyl-5-oxopyrrolidin-3-yl)benzamide
N-[3-(methylsulfanyl)butyl]-N-(pyridin-4-ylmethyl)cyclopropanamine
N-(4-methoxyphenyl)-5-(pyrimidin-5-yl)furan-2-carboxamide
{2-[2-(methoxymethyl)-1,3-benzoxazol-5-yl]phenyl}methanol
N-tert-butyl-3-{[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]amino}-5-(4-methyl-1,4-diazepane-1-carbonyl)benzene-1-sulfonamide
9-[(4-fluorophenyl)methyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-({5-[(1-methyl-1H-indol-6-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)methanesulfonamide
7-[(2-aminopyridin-3-yl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
2-(furan-2-yl)-5-({4-[1-(4-methylpiperazin-1-yl)ethyl]piperidin-1-yl}methyl)pyrimidine
2-(2,4-dichlorophenoxy)-N-methyl-N-[2-(oxan-2-yl)ethyl]acetamide
(1S,5R)-6-(dimethyl-1,2-oxazole-4-carbonyl)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
methyl (2S)-1-{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}pyrrolidine-2-carboxylate
2-{5-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1H-pyrazol-3-yl}phenol
3-(3-hydroxyquinoxalin-2-yl)-N-methyl-N-(quinolin-5-ylmethyl)propanamide
1-(methoxymethyl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]cyclobutane-1-carboxamide
(3S,4S)-1-cyclopentyl-4-(naphthalen-2-yl)piperidin-3-ol
9-[(3,5-difluorophenyl)methyl]-2-[2-(dimethylamino)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
(4aR,7aS)-1-acetyl-4-[2-(ethylamino)pyrimidine-5-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
1-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]-3-(naphthalene-2-carbonyl)piperidine
N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-3-methoxypropanamide
5-{1-[2-(phenylsulfanyl)acetyl]pyrrolidin-2-yl}thiophene-2-carboxamide
3-({methyl[2-(1H-pyrazol-4-yl)ethyl]amino}methyl)-7-(methylsulfanyl)-1,2-dihydroquinolin-2-one
N-methyl-2-(morpholin-3-yl)-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)acetamide
1-{4-[({1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}amino)methyl]thiophen-2-yl}ethan-1-one
4-{[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]sulfonyl}benzoic acid
1-{3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}pent-4-en-1-one
N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-[6-oxo-4-(piperidin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
5-[1-(2-methanesulfonylethyl)-4-phenyl-1H-imidazol-5-yl]-2,1,3-benzoxadiazole
N-(2-{5-[(cyclohexylmethyl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}ethyl)-4-methylbenzamide
6-[(diethylamino)methyl]-N-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide