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2-(1-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}pyrrolidin-2-yl)-6-methyl-1H-1,3-benzodiazole
(3aR,6aR)-2-acetyl-5-(1-benzothiophen-2-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(dimethyl-1,3-thiazol-5-yl)-N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}acetamide
N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-{[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]amino}acetamide
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}({[2-(methylsulfanyl)pyrimidin-5-yl]methyl})(pyridin-4-ylmethyl)amine
N-(1-{3-[(dimethylamino)methyl]-3-hydroxypiperidin-1-yl}-2-methyl-1-oxopropan-2-yl)thiophene-2-carboxamide
methyl 2-(1-{10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}pyrrolidin-3-yl)acetate
N-[4-(furan-2-yl)phenyl]-1-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperidine-3-carboxamide
1-[4-({3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}sulfonyl)phenyl]ethan-1-one
1-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(prop-2-en-1-ylsulfanyl)ethan-1-one
4-(3-fluoropyridine-4-carbonyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N-methyl-1H-pyrrolo[2,3-b]pyridin-6-amine
2-[methyl(1-{[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)amino]ethan-1-ol
1-[5-(ethylsulfanyl)thiophene-2-carbonyl]-3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
(2S)-3-(4-hydroxyphenyl)-2-{[6-(4H-1,2,4-triazol-4-yl)pyridin-3-yl]formamido}propanamide
N-butyl-N-(furan-2-ylmethyl)-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
1-(furan-3-ylmethyl)-4-[4-(naphthalen-2-yl)-1H-pyrazol-5-yl]piperidine
{4-[4-(4-methylphenyl)-2-[(pyrimidin-4-ylmethyl)amino]pyrimidin-5-yl]phenyl}methanol
4-[(4S)-4-hydroxy-3,3,4-trimethylpiperidin-1-yl]butanoic acid
4-phenyl-5-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]pyrimidin-2-amine
7-(9H-fluorene-9-carbonyl)-2,7-diazaspiro[4.4]nonane-1,3-dione
3-[1-(but-2-ynoyl)piperidin-3-yl]-N-[(2-fluorophenyl)methyl]propanamide
2-(6-methoxynaphthalen-2-yl)-4-(pyridine-3-carbonyl)morpholine
[(3R,4R)-4-[(dimethylamino)methyl]-1-[(3-fluoro-5-methylphenyl)methyl]pyrrolidin-3-yl]methanol
1-(3-fluorophenyl)-4-[3-(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-2-one
5-(2-chloro-4-methoxyphenoxymethyl)-N-(pyridin-3-ylmethyl)-1,2-oxazole-3-carboxamide
2-{2-[1-(2-ethoxybenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
[(3,4-dimethoxyphenyl)methyl](methyl){[5-methyl-2-(5-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}amine
(3S,4S)-4-cyclopropyl-1-[2-(4-ethylpiperazin-1-yl)acetyl]pyrrolidine-3-carboxylic acid
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-ethyl-N-(2-hydroxyethyl)acetamide
2-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-5-fluoro-N-methylpyrimidin-4-amine
3-[1-(5-methoxypyrimidin-2-yl)piperidin-3-yl]propanamide
3-({[1-(4-chlorophenyl)cyclopropyl]formamido}methyl)-N-(2-methoxyethyl)piperidine-1-carboxamide
3-ethyl-N-{4-[(2-phenylethyl)carbamoyl]phenyl}piperazine-1-carboxamide
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-2-(pyrrolidin-3-yl)benzamide
[(4-cyclopropyl-5-{1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
1-cyclopentanecarbonyl-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}piperidine-4-carboxamide
ethyl 4-{2-[4-(3-phenoxypropanamido)-1H-pyrazol-1-yl]acetyl}piperazine-1-carboxylate
2-{4-[3-(2,3-dihydro-1H-isoindol-2-yl)benzoyl]morpholin-3-yl}acetamide
N-[3-({[(4-phenylphenyl)methyl]amino}methyl)-5-(pyrrolidine-1-carbonyl)phenyl]acetamide
methyl 4-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}-4-oxobutanoate
2-[(4aS,7aR)-6,6-dioxo-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-1-carbonyl]benzonitrile
N-(2,3-dihydro-1-benzofuran-3-yl)-1-{2-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-amine
methyl 6-({[3-(furan-2-yl)propyl]carbamoyl}amino)-1,2,3,4-tetrahydroquinoline-1-carboxylate
N-cyclopentyl-5-(furan-2-ylmethyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
3-(1-methylcyclopropyl)-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)propanamide
4-benzyl-3-ethyl-N-(4-methoxyphenyl)-5-oxo-1,4-diazepane-1-carboxamide
2-[6-oxo-4-(piperidin-1-yl)-1,6-dihydropyridazin-1-yl]-N-(3-phenyl-1,2-oxazol-5-yl)acetamide
7-(6-ethyl-1,5-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide