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1-ethyl-4-{[4-(pyridin-4-yl)piperidin-1-yl]methyl}-1H-pyrrole-2-carbonitrile
(2S,4S)-1-cyclohexyl-N-ethyl-4-[2-(5-methyl-1H-pyrazol-1-yl)acetamido]pyrrolidine-2-carboxamide
3-{4-[2-(dimethylamino)phenyl]-1H-pyrazol-1-yl}propanamide
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]amine
3-(1-ethyl-1H-imidazol-2-yl)-1-[1-(4-fluorophenyl)cyclopropanecarbonyl]piperidine
N,N-dimethyl-1-{2-phenylimidazo[1,2-a]pyridine-6-carbonyl}pyrrolidin-3-amine
3-{2-[4-(3-methoxypropyl)piperidin-1-yl]-2-oxoethyl}-4-[(2-methylphenyl)methyl]piperazin-2-one
2-({4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)-6-methylpyridine
1-[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-1-yl]-2-(pyridin-3-yl)ethan-1-one
N-[(4-fluorophenyl)methyl]-5-(morpholin-4-ylmethyl)-N-(prop-2-en-1-yl)furan-3-carboxamide
4-(1-ethylpiperidin-4-yl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-ethyl-3-(4-methyl-4H-1,2,4-triazol-3-yl)-N-(pyridin-4-ylmethyl)propanamide
N-(4-{4-[(1H-indol-2-ylmethyl)amino]piperidin-1-yl}phenyl)cyclopentanecarboxamide
5-({3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}methyl)-2-methoxyphenol
(3S,4S)-1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]-4-(morpholin-4-yl)pyrrolidin-3-ol
2-[1-(4-chlorophenyl)-5-(3,3,3-trifluoropropyl)-1H-1,2,4-triazol-3-yl]acetamide
1-[2-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
2-(3,4-dichlorophenyl)-5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]pyridine
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[2-(4-hydroxypiperidin-1-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}thiophene-2-carboxamide
(3-benzyl-1-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}piperidin-3-yl)methanol
2-(4-fluorophenyl)-N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)acetamide
1-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-4-(2-fluorophenyl)piperazine
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-1-[(2-chlorophenyl)methyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
6-{1-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]piperidin-3-yl}pyrimidin-4-ol
(3aS,6aR)-5-(2,3-dihydro-1H-inden-2-yl)-3-[2-(pyridin-2-yl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-{2-methoxy-4-[(3,3,4-trimethylpiperazin-1-yl)methyl]phenoxy}-3-(pyrrolidin-1-yl)propan-2-ol
N-{[2-(4-acetylpiperazin-1-yl)-6-methylquinolin-3-yl]methyl}-N-[2-(cyclohex-1-en-1-yl)ethyl]furan-2-carboxamide
4-[6-(2,4-dimethoxyphenyl)pyrimidin-4-yl]morpholine
ethyl 1-{[2-(methoxycarbonyl)phenyl]carbamoyl}-4-(oxan-2-ylmethyl)piperidine-4-carboxylate
(1S,5R)-3-[(5-ethylpyridin-2-yl)methyl]-3,9-diazabicyclo[3.3.2]decan-10-one
(3S,4R)-4-(hydroxymethyl)-1-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}piperidin-3-ol
N-[2-ethoxy-5-(4H-1,2,4-triazol-4-yl)phenyl]-2-(pyrrolidin-3-yl)benzamide
N-[(3-methoxyphenyl)methyl]-6-methyl-2-oxo-N-(prop-2-en-1-yl)-1,2-dihydropyridine-3-carboxamide
2-[3-(hydroxymethyl)-3-propylpiperidin-1-yl]propane-1,3-diol
9-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(4-methoxypyrimidin-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-{2-[(4-methylpyridin-2-yl)amino]ethyl}-3-[3-(piperidine-1-carbonyl)phenyl]urea
2-methyl-N-{[1-(2-phenylethyl)piperidin-4-yl]methyl}imidazo[1,2-a]pyridine-6-carboxamide
2-amino-4-{3-[1-(dimethylamino)ethyl]phenyl}-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
(1R,2R,3R,4S)-N-cyclopropyl-3-(3-phenyl-1H-1,2,4-triazol-5-yl)bicyclo[2.2.1]hept-5-ene-2-carboxamide
N-(1,3-benzothiazol-2-ylmethyl)-N-methyl-2-[(4S)-2-oxo-4-(propan-2-yl)-1,3-oxazolidin-3-yl]acetamide
3-(2H-1,3-benzodioxol-5-yl)-1-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]propan-1-one
3-[4-(2-methoxyphenyl)-1,3-dimethyl-1H-pyrazol-5-yl]-1-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]urea
4-[4-(2-methylphenyl)-1H-imidazol-2-yl]-1-(propan-2-yl)pyrrolidin-2-one
(4aS,8aR)-1-(2-aminoethyl)-6-[3-(1H-1,2,4-triazol-1-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
5-(2,6-difluorophenoxymethyl)-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-1,2-oxazole-3-carboxamide
1-{7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}propane-1,2-dione
2-[1-(1H-imidazol-4-ylmethyl)piperidin-4-yl]-1,3-benzoxazole
1-(3-{[methyl(1,2-oxazol-5-ylmethyl)amino]methyl}phenoxy)-3-(morpholin-4-yl)propan-2-ol
4-[2-(4-chlorophenyl)morpholin-4-yl]butanoic acid