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1-{[1-(2H-1,3-benzodioxol-5-yl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-{2-[(1R,5S,8S)-8-hydroxy-3-azabicyclo[3.2.1]octan-3-yl]-4-(morpholin-4-yl)pyrimidin-5-yl}-2-methylpropanoic acid
3-{5-[(3-methyl-1,2-oxazol-5-yl)methyl]-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-1-yl}-1λ6-thiolane-1,1-dione
N-(3,5-dimethoxyphenyl)-3-[1-(2-hydroxy-6-methylpyridine-3-carbonyl)piperidin-3-yl]propanamide
(3S,9aR)-3-[(1R)-1-(benzyloxy)ethyl]-8-{[1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-ethylpyridine-4-carboxamide
2-(thiophen-2-yl)-N-(5,7,8-trimethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)azetidine-1-carboxamide
N-methyl-5-oxo-1-phenyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-2,5-dihydro-1H-pyrazole-3-carboxamide
3-[1-cyclohexyl-3-(2-methyl-1,3-thiazol-4-yl)-1H-1,2,4-triazol-5-yl]piperidine-1-carboxamide
2-amino-N-[3-hydroxy-1-(4-methylphenyl)propyl]-4-phenylpyrimidine-5-carboxamide
2-{2-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]-1H-1,3-benzodiazol-1-yl}ethan-1-ol
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-3-yl)-5-methylpyrazolo[1,5-a]pyrimidin-7-amine
N-(pyridin-3-ylmethyl)-N-(thiophen-3-ylmethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
3-[3-methoxy-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-1-(piperidin-4-ylmethyl)urea
3-(5-{[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]methyl}furan-2-yl)-1H-pyrazole
2-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-N,N,5-trimethylpyrimidin-4-amine
N-ethyl-N-[1-(4-methoxyphenyl)propyl]-3-(2-oxopiperidin-1-yl)propanamide
1-[5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-amido]cyclopentane-1-carboxylic acid
1-benzyl-4-{[4-(3-propylpyrrolidine-1-carbonyl)-1,3-oxazol-2-yl]methyl}piperazine
1-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-2-(3-fluorophenoxy)ethan-1-one
(2S,4S)-N,N-diethyl-4-[2-(methylsulfanyl)acetamido]-1-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
2-hydroxy-S-{4-[4-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]phenyl}ethane-1-sulfonamido
4-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]-6-(propan-2-yloxy)pyrimidin-2-amine
(4-{[(1-ethylpyrrolidin-3-yl)methyl]sulfamoyl}phenyl)urea
1-methyl-4-{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-1,4-diazepane
6-{4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-4-amine
1-[(5-ethylfuran-2-yl)methyl]-4-(oxolane-2-carbonyl)-1,4-diazepane
9-[(5-fluoro-2-methoxyphenyl)methyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N,2-dimethyl-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
7-(pyridine-2-amido)-N-(thiophen-2-yl)-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
N-benzyl-N-methyl-1-(3-methylthiophene-2-carbonyl)piperidin-3-amine
1-(carbamoylmethyl)-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]piperidine-4-carboxamide
methyl 2-{[2-(cyclohex-1-en-1-yl)ethyl]sulfamoyl}-6-(1-methyl-1H-pyrazole-5-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(4aR,8aS)-1-[2-(dimethylamino)ethyl]-6-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-decahydro-1,6-naphthyridin-2-one
N-(2-methyl-1-{2-[(methylcarbamoyl)methyl]-3-oxopiperazin-1-yl}-1-oxopropan-2-yl)thiophene-2-carboxamide
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-[2-(dimethylamino)-2-(5-methylfuran-2-yl)ethyl]urea
3-methoxy-N-[2-(2-methoxyphenoxy)phenyl]pyrrolidine-1-carboxamide
9-ethyl-3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-9H-carbazole
4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)-1-(cyclopropanesulfonyl)piperidine
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-(propan-2-yl)thiophene-3-carboxamide
N-cyclopropyl-1-{1-[(2-methyl-1,3-thiazol-4-yl)methyl]piperidin-4-yl}piperidine-3-carboxamide
2-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidine-1-carbonyl]-5-methoxy-4H-pyran-4-one
3-(2-amino-1,3-thiazol-4-yl)-N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methylpropanamide
1-(1-cycloheptylpiperidin-4-yl)-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1-oxo-1,2-dihydroisoquinoline-4-carboxamide
(1S,5R)-3-[4-(4-fluorophenyl)-1,3-thiazol-2-yl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(2S,4R,6S)-2-benzyl-6-[2-(propylamino)pyrimidin-5-yl]oxan-4-yl]acetamide
2-(2,5-dimethoxyphenyl)-5-methyl-4-(pyrrolidin-1-ylmethyl)-1,3-oxazole
N-[1-(2-phenylethyl)piperidin-3-yl]-3-(1H-pyrazol-4-yl)propanamide