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(3aR,6aR)-2-(3-chlorobenzoyl)-5-cyclobutanecarbonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(2R,6R)-4-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-(3-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-3-oxopropyl)acetamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-1-(methoxymethyl)-N-methylcyclobutane-1-carboxamide
2-[4-(furan-3-ylmethyl)-1-(3-methylbutyl)piperazin-2-yl]ethan-1-ol
N-[(3R,4S)-1-{[4-(methylsulfamoyl)phenyl]methyl}-4-propylpyrrolidin-3-yl]acetamide
dimethyl[2-({[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}(oxolan-2-ylmethyl)amino)ethyl]amine
2-(3-hydroxypropyl)-9-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
5-(4-butyl-3-oxopiperazin-1-yl)-1-ethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-2-(2-methylpiperidin-1-yl)-2-oxoacetamide
N-cyclopentyl-7-(pyrrolidine-1-sulfonyl)-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
[(3R,4R)-1-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-4-yl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methoxypyridine-3-carboxamide
1-(2-methoxyethyl)-2-oxo-3-(4-phenoxybutyl)-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
(2S)-2-amino-1-[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propan-1-one
2-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
4-(2,3-difluoro-6-methoxybenzoyl)-1-phenylpiperazin-2-one
3-{[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methoxy}pyridine
(2R,3R,6R)-5-(6-chloropyridazin-3-yl)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-(3-oxo-1,3-dihydro-2-benzofuran-5-yl)-1-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]urea
5-[(1-methyl-1H-pyrrol-3-yl)methyl]-3-[3-(pyrrolidin-1-yl)propyl]-1,2,4-oxadiazole
4-[2-(3-acetyl-1H-indol-1-yl)butanoyl]piperazin-2-one
3-(but-2-yn-1-yl)-5-{1-[(3-methylthiophen-2-yl)methyl]piperidin-4-yl}-5-(3-phenylpropyl)imidazolidine-2,4-dione
2-(2H-1,3-benzodioxol-5-yl)-N-[(3S,4S)-4-methoxy-1,1-dioxo-1λ6-thiolan-3-yl]acetamide
9-[(dimethyl-1,2-oxazol-4-yl)methyl]-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-3-one
5-[1-(cyclopent-1-ene-1-carbonyl)piperidin-4-yl]-5-propyl-3-[2-(pyridin-2-yl)ethyl]imidazolidine-2,4-dione
4-{4-[methyl(2-phenylethyl)amino]piperidin-1-yl}-N-[2-(morpholin-4-yl)ethyl]benzamide
N,6-dimethyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}pyridazin-3-amine
(3R,4S)-1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-4-phenylpyrrolidin-3-amine
3-benzyl-5-(2-phenoxyethyl)-1H-1,2,4-triazole
[(3-methylthiophen-2-yl)methyl][(3-phenyl-1,2,4-oxadiazol-5-yl)methyl](prop-2-en-1-yl)amine
3-(2-aminoethyl)-1-[3-(2-ethoxyethoxy)phenyl]urea
9-[(2R)-2-amino-3-methoxypropanoyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-{[4-fluoro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(3-methoxyphenyl)acetamide
2-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
N-[2-(3-benzyl-1H-1,2,4-triazol-5-yl)ethyl]acetamide
N-{[4-(dimethylsulfamoyl)phenyl]methyl}-3-(trimethyl-1H-pyrazol-4-yl)propanamide
6-ethyl-2-oxo-N-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]-1,2-dihydropyridine-4-carboxamide
4-(4-methoxyphenoxy)-1-(1,3-thiazol-4-ylmethyl)piperidine
3-[1-(2-methoxy-5-methylbenzenesulfonyl)piperidin-3-yl]-N-[(5-methylfuran-2-yl)methyl]propanamide
1-(2-cyclohexylethyl)-3-hydroxy-3-({[2-(3-methyl-1H-pyrazol-1-yl)ethyl]amino}methyl)piperidin-2-one
5-(oxolan-2-yl)-N-{[3-(pyrrolidin-1-ylmethyl)phenyl]methyl}thiophene-2-carboxamide
(3aR,6aS)-1-oxo-5-(5-phenyl-1,3,4-thiadiazol-2-yl)-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
7-methyl-6-oxo-N-(2-phenylphenyl)-2,7-diazaspiro[4.5]decane-2-carboxamide
5-(1-{2-[4-(methylsulfanyl)phenyl]acetyl}piperidin-4-yl)-5-propyl-3-[2-(pyridin-2-yl)ethyl]imidazolidine-2,4-dione
N-(2-cyclopentylethyl)-2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-1H-1,3-benzodiazole-5-carboxamide
2-ethyl-N,4-dimethyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1,3-oxazole-5-carboxamide
methyl 2-{methyl[(1-phenyl-1H-pyrazol-4-yl)methyl]carbamoyl}piperidine-1-carboxylate
(1S,4S)-5-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-2-(2,5-dimethoxyphenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
1-[1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-4-(2-ethoxyethyl)piperazine