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N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]thieno[2,3-d]pyrimidin-4-amine
3-(4-{[4-(2-methylphenyl)phenyl]methyl}piperazin-1-yl)propanamide
2-{4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-4-carbonitrile
5-(3,4-dimethylphenoxymethyl)-3-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}-1,2-oxazole
2-methyl-4-[4-({[1-(pyrimidin-2-yl)piperidin-3-yl]amino}methyl)phenyl]but-3-yn-2-ol
N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-3-propyl-1H-pyrazole-5-carboxamide
(2,3-dihydro-1-benzofuran-5-ylmethyl)(methyl)[1-(4-methylpyridin-2-yl)propan-2-yl]amine
4-(1H-imidazol-1-ylmethyl)-1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidin-4-ol
8-[(2S)-2-amino-4-(methylsulfanyl)butanoyl]-3-ethyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-ethyl-2-methyl-4-{4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine
[(4-fluoro-2-methylphenyl)methyl](methyl){[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}amine
N-[1-(2,5-difluorophenyl)cyclopropyl]-2-fluoro-5-sulfamoylbenzamide
1-[(3-methyl-1H-1,2,4-triazol-5-yl)methyl]-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
N-(2,5-dimethoxyphenyl)-2-(morpholin-4-ylmethyl)piperidine-1-carboxamide
N-[1-(furan-2-carbonyl)piperidin-3-yl]-7-methylimidazo[1,2-a]pyridine-2-carboxamide
3-[(3R,4S)-1-[2-(2,5-dimethylphenyl)acetyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
N-{[3-(3-fluorophenyl)oxolan-3-yl]methyl}-2,3-dihydro-1H-inden-2-amine
5-[(6-methoxy-2H-chromen-3-yl)methyl]-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
1-[1-(4-fluorophenyl)-2,2-dimethylcyclopropanecarbonyl]-4-phenylpiperidin-4-ol
(2S,4S)-N-ethyl-4-[(3E)-hex-3-enamido]-1-(4-hydroxybenzoyl)pyrrolidine-2-carboxamide
3-(furan-2-yl)-N-{2-[6-(pyrrolidin-1-yl)pyrimidin-4-yl]ethyl}propanamide
2-(8-methoxy-2-methylquinolin-5-yl)-N-(prop-2-en-1-yl)pyridine-3-carboxamide
2-methyl-N-[2-(7-{2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]propanamide
3-[(3S,4R)-3-cyclopropyl-4-[(4-ethyl-5-methylpyrimidin-2-yl)amino]pyrrolidin-1-yl]propan-1-ol
1-ethyl-3-(1H-1,2,4-triazol-1-ylmethyl)-5-{[4-(trifluoromethyl)phenyl]methyl}-1H-1,2,4-triazole
methyl 4-{[2-(furan-2-ylmethoxy)phenyl]carbamoyl}piperazine-1-carboxylate
2,5-difluoro-N-{1-[1-(2-hydroxyethyl)-1,2,3,6-tetrahydropyridin-4-yl]propan-2-yl}benzamide
methyl 2-[(oxolan-2-ylmethyl)({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)sulfamoyl]benzoate
4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1-ethylpiperidin-4-yl)piperidine
4-methyl-7-(4H-1,2,4-triazol-4-yl)-3,4-dihydro-2H-1,4-benzoxazin-3-one
methyl 2-[3-(3-chlorophenyl)-3-phenylpropanamido]acetate
5-tert-butyl-N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-1,3,4-oxadiazol-2-amine
3-(6-aminopyridin-2-yl)benzoic acid
2-{1-[(4-ethoxyphenyl)methyl]-4-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]piperazin-2-yl}ethan-1-ol
(4aS,7aR)-1-[(2,5-difluorophenyl)methyl]-4-(2-methoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(1-benzylpyrrolidin-3-yl)methyl]-2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetamide
6-(2-chlorophenyl)-2-(4-{[(3R)-3-hydroxypiperidin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-1H-1,2,3-benzotriazole-5-carboxamide
N-(1-{1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopentanecarboxamide
2,4-dichloro-3-{[3-(morpholine-4-carbonyl)piperazin-1-yl]methyl}phenol
1-methyl-2-oxo-8-[4-(1H-pyrazol-4-yl)butanoyl]-1,8-diazaspiro[4.5]decane-4-carboxylic acid
6-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidine-1-carbonyl]-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-{[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyloxolan-3-amine
1-benzyl-5-(ethoxymethyl)-3-(oxan-4-yl)-1H-1,2,4-triazole
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl][3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]methylamine
(3R,4S)-3,4-dimethyl-1-[2-(1,1,2,2-tetrafluoroethoxy)benzoyl]piperidin-4-ol
(1R,5R)-3-cyclobutanecarbonyl-6-[(2-ethylphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-methyl-N-(1H-pyrazol-3-ylmethyl)-2-[4-(trifluoromethyl)phenyl]-1,3-thiazole-4-carboxamide
6-[(2S)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-[2-(4-ethylpiperazin-1-yl)ethyl]-8-(oxolan-3-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one