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methyl 2-(4-{[3-(3-methylphenoxy)azetidin-1-yl]methyl}phenoxy)acetate
2-(2-aminopyridine-4-carbonyl)-7-(cyclobutylmethyl)-2,7-diazaspiro[4.5]decan-6-one
1-(3-chloropyridin-2-yl)-4-{[4-(5-methylpyridin-2-yl)piperidin-4-yl]methyl}piperazine
(1R,2R,6S,7S)-4-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}-10-oxa-4-azatricyclo[5.2.1.02,6]decane
4-{1-[1-(4-methanesulfonylphenyl)ethyl]-1H-imidazol-2-yl}pyridine
N-[(4-fluorophenyl)methyl]-3-(1H-imidazol-2-yl)-N-(3-methoxypropyl)benzamide
2-{1-[5-(phenoxymethyl)-1H-pyrazole-3-carbonyl]piperidin-4-yl}propan-2-ol
1-{3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}-3-phenylprop-2-yn-1-one
4-ethyl-3-{1-[1-(1H-imidazol-1-ylmethyl)cyclopropanecarbonyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
4-methyl-N-[2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-1,3-oxazole-5-carboxamide
2-(dimethyl-1,3-thiazol-5-yl)-1-[(1S,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
ethyl 2-[(3-{[(2-amino-1,3-thiazol-4-yl)methyl]carbamoyl}phenyl)amino]acetate
3-{5-[2-(3-hydroxyphenyl)acetyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
2-[(4aS,7aR)-4-(2-methoxyacetyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N-(2-fluorophenyl)acetamide
N-[(2R,3R)-1'-(cyclohex-1-ene-1-carbonyl)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenylacetamide
(2S,4S)-4-(3-ethoxypropanamido)-N-ethyl-1-(6-methylpyridine-3-carbonyl)pyrrolidine-2-carboxamide
[(2-ethylpyrimidin-5-yl)methyl](methyl)(quinolin-6-ylmethyl)amine
dimethyl(3-{2-[1-(2-methylpyridin-4-yl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)amine
N-[3-(dimethylamino)-2,2-dimethylpropyl]-15-methyl-13-oxo-9-(thiophen-3-yl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carboxamide
3-(4-methoxyphenyl)-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-1H-pyrazole-5-carboxamide
5-[4-(2-chlorophenyl)piperazine-1-carbonyl]-1,3-benzothiazol-2-amine
N-(1-{1-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]piperidin-4-yl}-1H-pyrazol-5-yl)-2,2-dimethylpropanamide
3-ethyl-N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-1H-pyrazole-4-carboxamide
3-[5-(benzylsulfanyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-[(2-chloro-6-fluorophenyl)methyl]piperidine
(1S,5R)-6-(2-chloro-4-fluorobenzoyl)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-{1-[(2-fluorophenyl)methyl]-4-{4-[(propan-2-yl)amino]pyrimidin-2-yl}piperazin-2-yl}ethan-1-ol
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-3-methyl-1,2-oxazole-5-carboxamide
1-{1-[3-(2-methyl-1H-imidazol-1-yl)propyl]piperidin-4-yl}-3-(pyrrolidine-1-carbonyl)piperidine
5-(4-fluorophenyl)-N-(furan-2-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
1-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-[2-(1H-imidazol-1-yl)ethyl]piperidine
N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-1-(propan-2-yl)piperidine-3-carboxamide
1-{4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(1H-imidazol-1-yl)ethan-1-one
N-benzyl-5-(2-methylpiperidine-1-carbonyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
N-[(3-methyl-1H-pyrazol-5-yl)methyl]-2-(pyrrolidin-1-yl)benzamide
2-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]pyrazine
N-[3-(furan-2-yl)propyl]-2,6-dimethylpyridine-4-carboxamide
5-(4-methyl-1,4-diazepan-1-yl)-2-{[1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl}-2,3-dihydropyridazin-3-one
N-[(4-chlorophenyl)methyl]-8-cyclopropyl-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxamide
1,5-dimethyl-2-phenyl-4-{[3-(phenylamino)piperidin-1-yl]methyl}-2,3-dihydro-1H-pyrazol-3-one
N-{[1-(ethoxymethyl)cyclobutyl]methyl}-6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-{[3-(3-methoxybenzoyl)piperidin-1-yl]methyl}-2,6-dimethylphenol
2-[3-(piperidin-1-ylmethyl)piperidin-1-yl]pyrimidin-4-amine
N-[2-(benzyloxy)ethyl]oxane-2-carboxamide
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-amine
1-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridin-6-yl]-2-(2,4-dichlorophenoxy)ethan-1-one
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}pyrrolidin-3-yl]methanol
N-(2-hydroxyethyl)-N-[(5-methylthiophen-2-yl)methyl]-5-(morpholin-4-ylmethyl)furan-3-carboxamide
3-methyl-N-{[5-methyl-7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}pentanamide
methyl (1S,3S,3aR,6aS)-1-(hydroxymethyl)-5-methyl-4,6-dioxo-3-[6-(trifluoromethyl)pyridin-3-yl]-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
9-[3-(4-ethylphenyl)-1H-pyrazole-5-carbonyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol