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(3R,9R)-11-(3-methoxybenzoyl)-5-thia-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
1-(4-{2-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrol-1-yl]-2-oxoethyl}phenyl)imidazolidin-2-one
5-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridin-2-amine
N-[3,5-difluoro-4-(trifluoromethyl)phenyl]-1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole-5-carboxamide
N-[2-(3-phenylpiperidin-1-yl)ethyl]-4-(4H-1,2,4-triazol-4-yl)benzamide
methyl (2S)-1-{1-[4-(4-methoxybenzamido)phenyl]piperidin-4-yl}pyrrolidine-2-carboxylate
4-[(1S,5R)-6-(3-methylbut-2-en-1-yl)-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1,2-dihydrophthalazin-1-one
2-benzyl-9-(butane-1-sulfonyl)-2,9-diazaspiro[5.5]undecan-3-one
dimethyl[(4-{1-[(1-methyl-1H-pyrazol-4-yl)sulfonyl]piperidin-2-yl}phenyl)methyl]amine
[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl](methyl)[(2,3,6-trifluorophenyl)methyl]amine
2-[N-(4-methylphenyl)methanesulfonamido]-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}acetamide
N-(1-{1-[2-(pyridin-3-yl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopropanecarboxamide
11-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}-7-methyl-3,7,11-triazaspiro[5.6]dodecane
5-[(1R,3S,5S)-3-(4-fluoro-3-methylphenyl)-8-azabicyclo[3.2.1]octane-8-carbonyl]-1-methyl-1H-1,3-benzodiazole
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-3-(1H-imidazol-2-yl)-N-methylbenzamide
2-(2-{2-amino-3-cyano-5H,7H,8H-pyrano[4,3-b]pyridin-4-yl}-6-methoxyphenoxy)propanoic acid
6-[1-(furan-2-ylmethyl)piperidine-3-carbonyl]-5,6,7,8-tetrahydro-1,6-naphthyridine
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-phenylacetamide
N-ethyl-5-({3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyrimidin-2-amine
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-5-(propan-2-yl)-1,3,4-thiadiazol-2-amine
1-ethyl-4-{4-[(3-methylphenyl)sulfanyl]piperidine-1-carbonyl}pyrrolidin-2-one
2-cyclobutanecarbonyl-6-methyl-5-[5-(thiophen-2-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
(3S,4R)-N,N-dimethyl-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-4-(4-methylphenyl)pyrrolidin-3-amine
4-[(1R,5S,8S)-8-methoxy-3-azabicyclo[3.2.1]octan-3-yl]-6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaene
{[2-(cycloheptanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)(1,2-oxazol-3-ylmethyl)amine
2-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-3-carboxamide
4-(morpholine-4-carbonyl)-N-(1,2-oxazol-3-ylmethyl)benzene-1-sulfonamide
2-[4-(2-methyl-1,3-benzothiazole-5-carbonyl)-2-oxopiperazin-1-yl]benzonitrile
3-{1-[(3-fluoro-2-methoxyphenyl)methyl]piperidin-3-yl}propanoic acid
4-{[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}morpholine
2-({2-[5-(methylcarbamoyl)thiophen-2-yl]pyrrolidin-1-yl}methyl)pyridine-3-carboxylic acid
(4aS,8aR)-1-[3-(1H-imidazol-1-yl)propyl]-6-(2-methoxy-2-methylpropanoyl)-decahydro-1,6-naphthyridin-2-one
N-cyclopropyl-N-(3-phenylprop-2-yn-1-yl)-2-[(prop-2-en-1-yl)amino]benzamide
N'-(3-ethylphenyl)-N-(1H-imidazol-2-ylmethyl)butanediamide
2-amino-6-(1,3-dimethyl-1H-pyrazol-4-yl)-4-[4-(1H-pyrazol-1-yl)phenyl]pyridine-3-carbonitrile
2-phenyl-4-[3-(1H-pyrazol-5-yl)piperidine-1-carbonyl]quinoline
N-(1-methoxypropan-2-yl)-3-{methyl[(3-methyl-1,2-oxazol-5-yl)methyl]sulfamoyl}benzamide
2-({4-[(3R,4S)-3-amino-4-propylpyrrolidine-1-carbonyl]phenyl}sulfanyl)ethan-1-ol
3-(4-fluorophenyl)-4-{[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methyl}-1H-pyrazole
2-[3-(2,6-dimethoxyphenyl)benzoyl]-1-methyl-1H-imidazole
3-{1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]azetidin-3-yl}pyridine
5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-methyl-N-(pyridin-3-ylmethyl)-1H-pyrazole-3-carboxamide
1-(4-methoxy-2-methylphenyl)-3-{[1-(methoxymethyl)cyclopentyl]methyl}urea
N-(1-{[4-(5-methylfuran-2-yl)phenyl]methyl}piperidin-3-yl)acetamide
N-[2-(dimethylamino)ethyl]-5-(2-hydroxypyridine-3-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
4-ethyl-3-{1-[(3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
(4aS,8aR)-1-butyl-6-[2-(3-oxo-2,3-dihydro-1H-indazol-2-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
2-{[4-(2,3-dichloro-4-methylphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1H-imidazole
N-{[2-(4-acetylpiperazin-1-yl)pyridin-3-yl]methyl}-4-(methylsulfanyl)benzamide
(3aS,6aS)-2-(2-aminopyrimidin-4-yl)-5-cyclopentanecarbonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid