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N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-3-phenyl-3-(pyridin-2-yl)propanamide
(1R,5R)-3-methanesulfonyl-6-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(pyrrolidin-1-yl)ethane-1,2-dione
1-{2-[ethyl(methyl)amino]acetyl}-4-(2-methoxyphenoxy)piperidine-4-carboxylic acid
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
3-[(3R,4S)-1-[(3-chlorophenyl)carbamoyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
(2E)-N-[(7S,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-phenylprop-2-enamide
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-2-hydroxy-4-(methylsulfanyl)butanamide
4-(2,3-difluoro-4-methoxybenzoyl)-1-[(3,5-dimethylphenyl)methyl]piperazin-2-one
N-[(2,5-dichlorophenyl)methyl]-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
1-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propan-1-one
5-[5-(1-cyclopentanecarbonylpiperidin-4-yl)-1,2,4-oxadiazol-3-yl]-1H-1,3-benzodiazole
1-amino-N-(2-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)cyclopropane-1-carboxamide
N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)-2-(1H-1,2,4-triazol-1-yl)acetamide
N-(2-benzamido-5-methylphenyl)-N'-cyclohexylethanediamide
3-{4-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperazin-1-yl}-1,2-dihydropyrazin-2-one
N-[(1-ethyl-1H-indazol-3-yl)methyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
7-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-2-oxa-7-azaspiro[4.5]decan-8-one
3-(dimethyl-1H-1,2,4-triazol-1-yl)-1-[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-methylpropan-1-one
1-cyclopentyl-4-[2-(trifluoromethyl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
methyl (2S)-1-{7-acetamido-1-[2-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazole-5-carbonyl}pyrrolidine-2-carboxylate
(3R,4R)-1-[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]-4-methyl-3-(propan-2-yl)pyrrolidin-3-ol
2-({6-hydroxy-4-[1-(hydroxymethyl)cyclopropanecarbonyl]-1,4-diazepan-1-yl}methyl)-3,5-dimethyl-1,4-dihydropyridin-4-one
N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
2-[4-methyl-3-(5-methylthiophen-2-yl)-1H-pyrazol-1-yl]-N-(1-propyl-1H-1,2,3-triazol-4-yl)acetamide
(3S,4R)-1-[(4-methanesulfonylphenyl)methyl]-N,N-dimethyl-4-(4-methylphenyl)pyrrolidin-3-amine
5-ethyl-3-[2-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)ethyl]-1,2,4-oxadiazole
7-(4-fluorophenyl)-2-[4-(hydroxymethyl)phenyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-(5-fluoro-2-methoxybenzoyl)-1-[(5-methylthiophen-2-yl)methyl]piperidine
(4aS,7aR)-1-[(4-methylphenyl)methyl]-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(1R,3S)-3-(2-aminoethoxy)-7-[3-(trifluoromethyl)benzoyl]-7-azaspiro[3.5]nonan-1-ol
1-[2-(4-fluorophenyl)piperidin-1-yl]-2-(2-phenyl-1H-imidazol-1-yl)ethan-1-one
4-[4-(3,5-dimethyl-1H-pyrazol-1-yl)butanoyl]-1-methylpiperazine-2-carboxylic acid
N-ethyl-2-{2-[3-oxo-3-(pyrrolidin-1-yl)propyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}propanamide
N-(1-{1-[1-(4-methylpyridin-2-yl)propan-2-yl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-phenylacetamide
2-({[(3R,4R)-4-(hydroxymethyl)-1-[(4-methylphenyl)methyl]pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
1-[2-(2-chlorophenyl)acetyl]-4-propyl-1,4-diazepan-5-one
N-[(2-fluorophenyl)methyl]-2-{4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}acetamide
N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}-1,9-dioxaspiro[5.5]undecan-4-amine
N-{[6-(3-chlorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-N-(2-methoxyethyl)furan-3-carboxamide
methyl[(1-{[1-(1-methyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]amine
6-methyl-2-(4-methylphenoxymethyl)-1-[2-(morpholin-4-yl)ethyl]-4-oxo-N-[1-(thiophen-2-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
3-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-1-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]propan-1-one
5-[(2-hydroxy-3-methylphenyl)methyl]-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-(4-{[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}phenoxy)ethan-1-ol
2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-N-methyl-N-(oxolan-2-ylmethyl)-1,3-oxazole-4-carboxamide
N-{[6-chloro-4-(pyrrolidin-1-yl)quinazolin-2-yl]methyl}methanesulfonamide
1-[(1S,3R)-1-[2-(dimethylamino)ethoxy]-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-3-(thiophen-3-yl)propan-1-one
1-methyl-8-[(1-methyl-1H-indol-3-yl)methyl]-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-benzyl-3-[1-(2-methylpyrimidine-5-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one