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[(3S,5R)-1-(2-methoxypyridine-4-carbonyl)-5-(pyrrolidin-1-ylmethyl)piperidin-3-yl]methanol
2-methoxy-N-{[5-(piperidin-3-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}acetamide
N-[4-(propan-2-yl)phenyl]-1-(thian-4-yl)piperidin-3-amine
N-methyl-5-{2-oxo-1-oxaspiro[4.5]decane-4-carbonyl}-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-[4-(2-methylpropyl)benzoyl]pyrrolidin-3-yl]methanol
dimethyl({2-[1-(pyridine-3-sulfonyl)piperidin-2-yl]ethyl})amine
4-(2-aminopyrimidin-4-yl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propan-1-one
2-[1-(azepan-1-yl)-2-methylpropan-2-yl]-5-(1H-1,2,3,4-tetrazol-1-yl)-1H-1,3-benzodiazole
4-phenyl-1-{1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}-1,2,3,6-tetrahydropyridine
1-[(2,3-difluoro-6-methoxyphenyl)methyl]-2-(5-methyl-1,2-oxazol-3-yl)piperidine
N,5-dimethyl-4-phenyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}thiophene-3-carboxamide
1-(1-methyl-1H-pyrazole-5-carbonyl)-3,3-diphenylpiperidine
4-[2-(methylsulfanyl)phenyl]-3-(1H-1,2,3,4-tetrazol-5-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
5-[4-(3-cyanopyridin-2-yl)piperazin-1-yl]-1-ethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
2-(4,6-dimethyl-1-benzofuran-3-yl)-1-{5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethan-1-one
2-(4,7-dimethyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}acetamide
3-methyl-4-(2-methyl-1,3-thiazole-5-carbonyl)-1-(2-methylpropyl)piperazin-2-one
ethyl 1-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-3-(2-phenoxyethyl)piperidine-3-carboxylate
N-(2-{4-methyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)-3-(4-methylphenyl)propanamide
8-fluoro-N,N-bis(1,3-oxazol-4-ylmethyl)quinoline-2-carboxamide
2-[(1-methylpiperidin-4-yl)(pyridin-3-ylmethyl)amino]-1-(morpholin-4-yl)ethan-1-one
2-({[(3R,4R)-4-(hydroxymethyl)-1-(1-phenylcyclohexanecarbonyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
(3R,5S)-1-benzyl-5-[(2,3-dihydro-1H-inden-5-yloxy)methyl]-N-[3-(dimethylamino)propyl]piperidine-3-carboxamide
3-[(1-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]-2,3-dihydro-1,3-benzoxazol-2-one
N-[1-(3-methylpyridin-2-yl)propan-2-yl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
2-(2-methyl-1,3-thiazol-4-yl)-N-{3-[(pyridin-3-yl)amino]propyl}acetamide
N-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]-3,5-dimethyl-1H-pyrazole-4-sulfonamide
{5-[3-(5-methylfuran-2-yl)butyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}methanol
2-(trifluoromethyl)-6-(2,3,4-trimethoxyphenyl)pyridine
methyl (2S,4R)-1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-4-(4-methoxybenzamido)pyrrolidine-2-carboxylate
5-[2-(3-methoxyphenyl)azetidine-1-carbonyl]-3-propyl-1H-pyrazole
1-cyclopentyl-5-{4-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine-1-carbonyl}piperidin-2-one
2-(5,5-dimethyl-2,4-dioxo-1,3-oxazolidin-3-yl)-N-[1-(2-methoxyphenyl)propan-2-yl]-N-methylacetamide
2,3-dimethyl-5-[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidine-1-carbonyl]benzene-1-sulfonamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[2-(1H-imidazol-1-yl)ethyl]benzamide
{4-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-1-methylpiperazin-2-yl}methanol
4-[(2,4-dimethoxyphenyl)methyl]-9-methoxy-7-[4-(methylsulfanyl)phenyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(1-{1-[(5-ethylfuran-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)acetamide
6-methyl-5-({3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}methyl)quinoline
N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-5-phenylpentanamide
(3S,4R)-1-(4-carboxybutanoyl)-4-phenylpyrrolidine-3-carboxylic acid
2-(2-hydroxyethyl)-8-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
1-{6-[(2-hydroxyethyl)amino]pyrimidin-4-yl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-(1-benzylpyrrolidin-3-yl)-3-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]propanamide
2-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-6-(piperidin-3-yl)pyrimidin-4-amine
4-[4-(3-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-2-(trifluoromethyl)pyrimidine
N-[phenyl(pyridin-4-yl)methyl]-2-[(propan-2-yl)amino]pyrimidine-5-carboxamide
N-[(5-methylfuran-2-yl)methyl]-2-(oxolane-2-carbonyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]acetamide