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6-{2-[(4-methoxyphenyl)methoxy]phenyl}-N,N-dimethylpyridine-3-carboxamide
N-{5-methoxy-2-[2-(1H-1,2,3,4-tetrazol-1-yl)acetamido]phenyl}-2-methylpropanamide
4-cyclobutyl-6-methyl-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}pyrimidin-2-amine
N-cyclopentyl-1-propyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2,2-dimethyl-1-(3-{[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)butan-1-one
4-{4-[3-(2-chlorophenoxy)azetidin-1-yl]piperidin-1-yl}-6-methylpyrimidin-2-amine
2-({4-[2-(3-methyl-1H-1,2,4-triazol-5-yl)pyrrolidine-1-carbonyl]phenyl}sulfanyl)ethan-1-ol
2-[4-(2,2-dimethylpropyl)-1-[(4-methylphenyl)methyl]piperazin-2-yl]ethan-1-ol
2-(dimethylamino)-2-(2-methylphenyl)-1-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]ethan-1-one
1-[(2-amino-1,3-thiazol-4-yl)methyl]-3-(5-tert-butyl-1,3,4-thiadiazol-2-yl)urea
2-methoxy-4-{[3-(3-methoxyphenoxymethyl)piperidin-1-yl]methyl}phenol
N-[(2,4-difluorophenyl)methyl]-2-(1H-1,2,4-triazol-3-yl)benzamide
2-[4-(2-methylpyridin-4-yl)-1,4-diazepane-1-carbonyl]benzonitrile
4-[4-(2,3-dihydro-1H-indene-1-carbonyl)piperazin-1-yl]quinazoline
4-(1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl)pyrimidin-2-amine
7-amino-4-(trimethyl-1H-pyrazol-4-yl)-1,2,3,4-tetrahydro-1,8-naphthyridin-2-one
2-(ethylamino)-4-methyl-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1,3-thiazole-5-carboxamide
N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
(3S,4S)-1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-(4-fluorophenyl)piperidin-3-ol
3,3,3-trifluoro-1-{7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}propan-1-one
(3R)-1-(2-amino-6-methoxypyrimidin-4-yl)-3,4,4-trimethylpyrrolidin-3-ol
5-(4-{imidazo[1,2-b]pyridazin-6-yl}piperazine-1-carbonyl)-1H-1,2,3-benzotriazole
2-[3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propanoyl]-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
2-(2-cyclopropylacetyl)-N-methyl-N-(1,3-thiazol-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
1-(furan-2-ylmethyl)-N-methyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidine-3-carboxamide
2-{3-[2-methyl-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}-N-(propan-2-yl)acetamide
5-{[(1,4-dioxan-2-ylmethyl)(methyl)amino]methyl}-2-oxo-2,3-dihydro-1H-imidazole-4-carboxylic acid
N-{5-[(5S,9aS,9bS)-2-(1-methylpiperidin-4-yl)-1-oxo-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-5-yl]thiophen-2-yl}acetamide
(3S,4R)-4-(4-fluorophenyl)-1-(1,3-thiazol-2-ylmethyl)pyrrolidine-3-carboxylic acid
2-(furan-2-yl)-N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
ethyl 5-[(3-methylquinoxalin-2-yl)methyl]-1-(prop-2-en-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-[4-(5,6-dimethylpyrimidin-4-yl)piperazin-1-yl]-4-(piperidin-1-yl)butan-1-one
[2-({1-[(2-methoxy-3,5-dimethylphenyl)methyl]piperidin-4-yl}oxy)ethyl]dimethylamine
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-(4-hydroxy-3,5-dimethylphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-[(2-{7,7-dimethyl-4-oxo-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-2-yl}phenyl)methyl]pyrrolidin-2-one
2-benzyl-8-(3-propyl-1H-pyrazole-4-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
1-(2-methoxyethyl)-N-[2-(5-methylthiophen-2-yl)ethyl]-6-oxopiperidine-3-carboxamide
4-[(1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-2-yl)methyl]morpholine
1-[(4-fluorophenyl)methyl]-2-(propan-2-yl)-4-(pyrrolidine-1-carbonyl)-1,4-diazepane
(2R)-2-cyclohexyl-2-hydroxy-N-[(5-methoxy-1H-indol-2-yl)methyl]acetamide
1-{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-ol
methyl (2R,4S)-4-hydroxy-1-[(2-hydroxyphenyl)methyl]piperidine-2-carboxylate
[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl](methyl)[3-(1H-pyrazol-1-yl)propyl]amine
N-(propan-2-yl)-4-{[1-(pyridin-2-yl)propan-2-yl]sulfamoyl}benzamide
2-cyclopropyl-8-(5-ethyl-2,6-dimethylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
1-[(4-methoxy-2-methylphenyl)methyl]-3-(piperidin-1-ylmethyl)pyrrolidin-3-ol
2-(2H-1,3-benzodioxol-5-yl)-1-[3-(hydroxymethyl)-3-(2-phenoxyethyl)piperidin-1-yl]ethan-1-one
4-(5-{4-[(2-fluorophenyl)methyl]piperidine-1-carbonyl}-1H-pyrazol-3-yl)pyridine
N-methyl-4-[(1S,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridin-2-amine
3-[(1-acetylpiperidin-4-yl)oxy]-N-cyclooctyl-4-methoxybenzamide