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8-cyclopropanecarbonyl-2-[(3-methylthiophen-2-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-(ethylamino)-5-methyl-N-[2-(pyridin-4-yl)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide
2-{4-[(4-ethylphenyl)methyl]-1-(propan-2-yl)piperazin-2-yl}ethan-1-ol
3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-1,2,5,6,7,8-hexahydroquinolin-2-one
1-(furan-2-ylmethyl)-4-[2-(pyridin-2-yl)pyrimidin-5-yl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
3-(1-methyl-1H-1,3-benzodiazol-6-yl)-1-[1-(pyrimidin-2-yl)piperidin-3-yl]urea
5-[4-(2-ethylpyrimidine-5-carbonyl)piperazin-1-yl]-6-phenyl-2,3-dihydropyridazin-3-one
1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-(3-methylphenoxy)piperidine
N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)-2H-1,3-benzodioxole-5-carboxamide
8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-butyl-N-methyl-1-{2-[(4-methyl-1,3-thiazol-2-yl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}piperidine-3-carboxamide
5-(3-{1-[(2,4-difluorophenyl)methyl]-1H-pyrazol-3-yl}phenyl)pyrimidine
3-butanamido-4-methyl-N-[2-(1-methylpyrrolidin-2-yl)ethyl]benzamide
(1S,5R)-3-benzyl-6-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
5-benzyl-5-[1-(5-ethyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]-3-[2-(pyrrolidin-1-yl)ethyl]imidazolidine-2,4-dione
[(3R,4R)-1-(7-chloroquinolin-4-yl)-4-[(4-ethylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
N-tert-butyl-6-ethyl-2-(morpholin-4-yl)pyrimidin-4-amine
1-(1-benzyl-1H-pyrazole-4-carbonyl)-4-(hydroxymethyl)piperidin-4-ol
4-benzyl-1-[(4-methoxypyridin-2-yl)methyl]-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-cyclopropyl-5-{1-[(4-methoxyphenyl)methyl]-1H-pyrazol-4-yl}-1H-1,2,4-triazole
1-(furan-2-carbonyl)-4-[(3-{[1-(4-methylbenzoyl)piperidin-4-yl]oxy}phenyl)methyl]piperazine
N-methyl-N-[(3-methyl-1H-indol-2-yl)methyl]piperidin-4-amine
2-(adamantan-1-yl)-5-(3-hydroxy-3-methylpiperidine-1-carbonyl)pyrimidin-4-ol
5-[4-(2-methoxyphenyl)piperazine-1-carbonyl]-1,3-benzothiazol-2-amine
1-(2,4-dimethoxybenzoyl)-4-[2-(oxolan-2-yl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidine
5-[1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1H-1,2,3-triazol-4-yl]-3-(propan-2-yl)-1,2,4-oxadiazole
1-{4-[(3-chlorophenyl)methyl]piperazin-1-yl}-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
2-{[(4-tert-butylphenyl)formamido]methyl}-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
2-hydroxy-1-(3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)ethan-1-one
N-(5-chloro-2-methoxyphenyl)-3-(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-3-yl)propanamide
N-[2-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
3-(4-fluorophenyl)-N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-1H-pyrazole-5-carboxamide
(1R,5R)-3-benzoyl-6-[(4-fluoro-3-methylphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
4-{2-[1-(morpholine-4-carbonyl)piperidin-2-yl]ethyl}phenol
N-{2-[4-(hydroxymethyl)piperidin-1-yl]-5,6,7,8-tetrahydroquinazolin-5-yl}cyclohexanecarboxamide
N4-[(8-methoxyquinolin-5-yl)methyl]-N2,N2,N4-trimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
2-[(6-hydroxy-1,4-oxazepan-4-yl)methyl]-3,5-dimethyl-1,4-dihydropyridin-4-one
6-methyl-3-{[3-(pyridin-3-ylmethoxy)piperidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
2-{4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-N-methylacetamide
N-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-5-propylpyrazolo[1,5-a]pyrimidin-7-amine
ethyl 3-{[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carbonyl]amino}propanoate
N-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]-1,4-dithiepan-6-amine
1-{4-[4-(thiophen-2-ylmethyl)-1,4-diazepane-1-carbonyl]thiophen-2-yl}ethan-1-one
5-methyl-1-{2-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-[1-(cyclohexylmethyl)-3-(1-phenylcyclopropyl)-1H-1,2,4-triazol-5-yl]morpholine
N-(1-hydroxybutan-2-yl)-N-(pyridin-2-ylmethyl)-1-benzofuran-2-carboxamide
{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[2-(furan-2-yl)ethyl]amine
1-methyl-N-{[4-(methylsulfanyl)phenyl]methyl}-2-oxo-N-propyl-1,2-dihydropyridine-3-carboxamide
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-[2-(1H-imidazol-1-yl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
{2-[3-(pyrrolidin-1-ylmethyl)phenyl]phenyl}methanol