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4-(6-aminopyrimidin-4-yl)-7-(3,6-dimethylpyrazin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
6-methoxy-N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}pyrimidin-4-amine
[(3S,5R)-5-(morpholin-4-ylmethyl)-1-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]piperidin-3-yl]methanol
5-[2-(dimethylamino)-2-(2-methylphenyl)acetyl]-N,N-dimethyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide
1-[(3,5-dimethylphenyl)methyl]-4-{2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetyl}piperazin-2-one
3-(5-methylthiophen-2-yl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazole-5-carboxamide
N-{2-[4-(hydroxymethyl)piperidin-1-yl]-5,6,7,8-tetrahydroquinazolin-5-yl}furan-2-carboxamide
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N,2-dimethyl-6-(piperidin-3-yl)pyrimidin-4-amine
(1S,5R)-6-[(4-fluoro-3-methoxyphenyl)methyl]-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
5-acetyl-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N'-cyclopentyl-N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methylbutanediamide
N-{imidazo[1,2-a]pyridin-3-ylmethyl}-N-methyl-5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carboxamide
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-[3-(1H-1,2,4-triazol-1-yl)propyl]-1H-1,2,4-triazole
2-(1H-indol-2-ylmethyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
N-butyl-2-[1-(4-chlorophenyl)-3-(furan-2-yl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]acetamide
N-methyl-1-[2-(piperazin-1-yl)ethyl]-N-[2-(pyridin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-[(3-methoxyphenyl)methyl]-4-[2-(propylsulfanyl)acetyl]piperazin-2-one
3-{1-[(5-cyclopentylthiophen-2-yl)methyl]piperidin-4-yl}-1-(morpholin-4-yl)propan-1-one
(2R,3S,6R)-5-[(2-butyl-1H-imidazol-4-yl)methyl]-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[1-methyl-5-({methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]amino}methyl)-1H-pyrrol-3-yl]ethan-1-one
N,2-dimethyl-N-[3-(oxolan-2-yl)propyl]-2-(thiophen-2-ylformamido)propanamide
2-cyclopentyl-N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
1-[(1R,5R)-6-{[5-(4-ethoxyphenyl)furan-2-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
3-{2-[(2-butyl-6-methylpyrimidin-4-yl)amino]ethyl}-1-(6-methylpyridin-3-yl)urea
4-(4-methylphenyl)-2-[4-(propan-2-yl)piperazin-1-yl]-5-(pyrimidin-5-yl)pyrimidine
1-(4-methoxyphenyl)-3-methyl-4-(pyridin-4-ylmethyl)piperazin-2-one
6-(4-fluorophenyl)-N-[(5-phenyl-1H-pyrazol-3-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
(2R,6S)-4-{[1-benzyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}-2,6-dimethylmorpholine
N-[2-(2-fluorophenyl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]ethyl]-N-methylthiophene-2-carboxamide
N-benzyl-N-methyl-1-(thian-4-yl)piperidin-3-amine
3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-2-one
2-[1-(3,5,7-trimethyl-1H-indole-2-carbonyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
4-phenyl-1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperidine-4-carbonitrile
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-[(5-propylfuran-2-yl)methyl]piperidin-3-yl]propanoic acid
N-[1-methyl-4-(pyridin-3-yloxy)-1H-indazol-3-yl]-1-propyl-1H-pyrazole-5-carboxamide
N-{[2-(butan-2-yloxy)phenyl]methyl}-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
(2S,4S)-4-amino-1-[(3E)-hex-3-enoyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-propyl-1,3-thiazole-4-carboxamide
5-({5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}amino)-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-4-(1-methyl-1H-imidazol-2-yl)-1H-1,2,3-triazole
(2S,3S)-2-amino-3-methyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]pentanamide
2-{2-[3-(hydroxymethyl)-4-methylpiperazin-1-yl]-4-(morpholin-4-yl)pyrimidin-5-yl}-2-methylpropanoic acid
3-(3-tert-butyl-1-methyl-1H-pyrazol-5-yl)-1-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]urea
N-[(3S,4S)-4-methoxy-1,1-dioxo-1λ6-thiolan-3-yl]-2-(thiophen-2-yl)acetamide
N-[2-(4,5-dimethyl-1H-imidazol-1-yl)ethyl]-2-[(4-oxo-3,4-dihydroquinazolin-2-yl)sulfanyl]propanamide
1-(2,4-dichloro-3-methylphenyl)-3-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-3-methylurea
4-chloro-2-{[3-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]methyl}phenol
2-(1H-imidazol-4-yl)-1-(2-phenoxyethyl)-1H-imidazole
2-ethyl-5-(2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-2-oxoethyl)-6-methyl-3,4-dihydropyrimidin-4-one