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2-(1-ethylpiperidin-4-yl)-1-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethan-1-one
(3aS,6aS)-1-oxo-2-(prop-2-en-1-yl)-5-[(5-propylfuran-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]-2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane
3-(5-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl)pyridine
2-[3-(dimethylamino)propyl]-9-[(4-methoxy-2-methylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
2-[(2E)-3-phenylprop-2-en-1-yl]-8-(pyridine-2-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
6-{4-[hydroxy(thiophen-2-yl)methyl]piperidine-1-carbonyl}-2-methyl-2,3-dihydropyridazin-3-one
1-(2-{4-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrol-2-ylmethyl]-2-methoxyphenoxy}ethyl)pyrrolidine
N-[(3R,4R)-3-hydroxy-1-[3-(pyridin-2-yl)propanoyl]piperidin-4-yl]pyrazine-2-carboxamide
2-(4-methanesulfonylphenyl)-1-[3-(1H-pyrazol-1-yl)phenyl]-1H-imidazole
N-[1-(4-cyclopentyl-4H-1,2,4-triazol-3-yl)ethyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
1-({1-[(3-fluorophenyl)methyl]-6-methyl-2-oxo-1,2-dihydroquinolin-3-yl}methyl)-4-(piperidin-1-yl)piperidine-4-carboxamide
2-(2-methoxyphenyl)-1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
9-(2-propoxypropanoyl)-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
(3S,7S,8aS)-7-({[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)-3-(2-methylpropyl)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
(4aR,7aS)-1-ethyl-4-(2-methyl-1,3-benzothiazole-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-6-methylquinoline-4-carboxamide
5-(2,6-difluorophenoxymethyl)-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1,2-oxazole-3-carboxamide
2-cyclopropyl-8-[3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
(2R,6R)-10-methoxy-4-(pent-2-yn-1-yl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
3-[(1R,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propanoic acid
6-{4-[(2,4-dimethoxyphenyl)methyl]piperazin-1-yl}pyridine-3-carboxylic acid
3-[1-(8-fluoroquinolin-2-yl)-N-(2-phenylethyl)formamido]propanamide
2-(5-ethylfuran-2-yl)-1-[2-(1H-imidazol-4-yl)ethyl]-1H-imidazole
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-1,5-dimethyl-1H-pyrazole-4-carboxamide
N-[3-(2-methoxyacetamido)phenyl]-4-(pyridin-4-yl)piperazine-1-carboxamide
1-{1-[2-(1H-1,2,4-triazol-3-yl)benzoyl]piperidin-3-yl}pyrrolidin-2-one
N-[(5-ethylpyridin-2-yl)methyl]-N,2,5-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
N-{4-[(furan-2-ylmethyl)sulfanyl]phenyl}-2-(3-methyl-1,2-oxazol-5-yl)pyrrolidine-1-carboxamide
3-{1-[(4-acetamidophenyl)methyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)propanamide
2-{1-[1-(furan-2-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-2-ol
N-[(3,4-dimethylphenyl)(pyridin-3-yl)methyl]-1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-(ethylamino)-N,4-dimethyl-N-[1-(thiophen-2-yl)ethyl]-1,3-thiazole-5-carboxamide
(1R,5R)-3-[1-(4-fluorophenyl)cyclopropanecarbonyl]-3,9-diazabicyclo[3.3.2]decan-10-one
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-6-methylimidazo[2,1-b][1,3]thiazole-3-carboxamide
{3-[(1-{2-[(dimethylamino)methyl]-1,3-thiazole-4-carbonyl}pyrrolidin-3-yl)methyl]phenyl}methanol
N-[2-(cyclohex-1-en-1-yl)ethyl]-2-{[3-(pyridin-3-yl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]sulfanyl}acetamide
N-{1-[2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]piperidin-4-yl}methanesulfonamide
6-(2-methoxyphenyl)-N-methyl-N-[2-(morpholin-4-yl)propyl]pyridazin-3-amine
[1-({[4-(1-methyl-1H-1,2,4-triazol-5-yl)pyrimidin-2-yl]amino}methyl)cyclobutyl]methanol
N4-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]pyrimidine-4,6-diamine
(3S,4S)-1-(5-amino-4-chloro-1H-pyrazole-3-carbonyl)-4-cyclopropylpyrrolidine-3-carboxylic acid
2-(2,4-dichlorophenoxy)-N-[2-(methylsulfamoyl)ethyl]acetamide
4-[1-(2-phenoxyacetyl)piperidin-3-yl]benzoic acid
3-[2-(2,5-dioxoimidazolidin-1-yl)acetamido]-N-(2-ethylphenyl)benzamide
1-(oxolane-2-carbonyl)-4-[3-(4H-1,2,4-triazol-4-yl)benzoyl]-1,4-diazepane
2-methyl-N-[3-(pyrrolidin-1-yl)butyl]thieno[2,3-d]pyrimidin-4-amine
N-butyl-4-[(3-methoxypropyl)amino]-N,5-dimethylthieno[2,3-d]pyrimidine-6-carboxamide
[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl](methyl)[3-(methylsulfanyl)butyl]amine