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(2S,4S)-1-[(2-chlorophenyl)methyl]-N-methyl-4-({[2-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-5-(1H-pyrazol-1-ylmethyl)furan-2-carboxamide
5-({4-[(1S,4S)-2-azabicyclo[2.2.1]heptane-2-carbonyl]-1,3-oxazol-2-yl}methoxy)-2-methyl-1,3-benzothiazole
3-(azepane-1-carbonyl)-1-ethyl-N-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-{[1-(6-methoxypyridin-3-yl)-1H-1,3-benzodiazol-2-yl]methoxy}acetic acid
{3-cyclobutanecarbonyl-9-[(2-fluorophenyl)methyl]-3,9-diazaspiro[5.5]undecan-1-yl}methanol
2-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}quinoline
N-[(2R,4R,6S)-2-cyclohexyl-6-[2-(morpholin-4-yl)pyridin-3-yl]oxan-4-yl]acetamide
N-(3-methylbutyl)-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
{[4-(1-{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl)phenyl]methyl}dimethylamine
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-hydroxypiperidin-1-yl)methyl]pyrrolidin-1-yl]-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethan-1-one
methyl 5-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
(1R,5S,8S)-3-[4-(3-fluorophenyl)benzoyl]-N,N-dimethyl-3-azabicyclo[3.2.1]octan-8-amine
2-[4-(2-methoxyphenyl)-3-oxopiperazin-1-yl]-N-[(2-methoxyphenyl)methyl]acetamide
(3S,4R)-N,N-dimethyl-4-(4-methylphenyl)-1-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}pyrrolidin-3-amine
N-(2-cycloheptylethyl)thian-4-amine
[(3R,4R)-1-(4-aminopyrimidin-2-yl)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)pyrrolidin-3-yl]methanol
(3R,9aR)-3-(2-methylpropyl)-8-(4-phenylbenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
8-[(2R)-2-hydroxy-2-phenylethyl]-2-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
ethyl 1-(5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carbonyl)piperidine-4-carboxylate
4-(1H-imidazol-1-yl)-N-{[3-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}benzamide
2-[(1-benzofuran-5-ylformamido)methyl]-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
(2R,3S,6R)-3-(3-methoxyphenyl)-5-(oxane-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-amino-3-ethyl-N-(2-phenoxyethyl)-3H-imidazo[4,5-b]pyridine-6-carboxamide
3,6-dimethyl-N-[2-(pyrazin-2-yl)ethyl]-1-benzofuran-2-carboxamide
1-methyl-1'-(6-methyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
6-{[1-(1,4-oxazepan-4-yl)hex-5-en-2-yl]oxy}pyridine-2-carbonitrile
5-[4-(4-butyl-1H-1,2,3-triazol-1-yl)piperidine-1-carbonyl]pyrimidine
3-(2H-1,3-benzodioxol-5-ylmethyl)-1-[(4-methanesulfonylphenyl)methyl]-3-methylpiperidine
2-(1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}pyrrolidin-2-yl)pyridine
1-(carbamoylmethyl)-N-[3-(4-fluorophenyl)propyl]piperidine-3-carboxamide
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-1-(pyrrolidin-1-yl)cyclopentane-1-carboxamide
7-(cyclopropylmethyl)-2-{2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}-2,7-diazaspiro[4.5]decan-6-one
N-[2-fluoro-5-({[3-(pyridin-2-yl)propyl]carbamoyl}amino)phenyl]-2-methylpropanamide
1-{5,7-dimethyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carbonyl}-2-(3-methoxyphenyl)piperidine
methyl 3-{[1-(cyclopropylmethyl)-5-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]formamido}propanoate
4-({1-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]piperidin-2-yl}methyl)morpholine
(1H-imidazol-2-ylmethyl)(methyl){[8-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}amine
[(3R,4R)-1-(4-chlorobenzoyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
4-[2-(propan-2-yl)pyrimidine-5-carbonyl]-1λ6-thiomorpholine-1,1-dione
(1R,5R)-6-benzyl-3-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
5-cyclopropanecarbonyl-1'-(1H-imidazol-2-ylmethyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-(pyridin-3-ylmethyl)-4-[(3-{[1-(1,3-thiazole-5-carbonyl)piperidin-4-yl]oxy}phenyl)methyl]piperazine
5-methyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(1S,5R)-6-(2-methoxyethyl)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
2,6-diamino-4-[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]-5,6,7,8-tetrahydroquinoline-3-carbonitrile
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-2-(5-oxopyrrolidin-2-yl)acetamide
N-cyclopropyl-4-(2-phenoxyethyl)benzamide
N,5-dimethyl-N-(1-methylpyrrolidin-3-yl)-1-propyl-1H-pyrazole-4-carboxamide
2-ethyl-5-[4-(oxolan-2-ylmethyl)piperazine-1-carbonyl]pyrimidine