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(1R,5S)-3-(1-benzofuran-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
{1-[(1-{7-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-3-yl)methyl]-1H-1,2,3-triazol-4-yl}methanol
4-({3-[(2H-1,3-benzodioxol-5-yl)amino]piperidin-1-yl}methyl)-5-chloro-2-methoxyphenol
2-[4-(5-chloropyridin-2-yl)-1-[(3,5-dimethoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
1-(5-ethylpyrimidin-2-yl)-4-(hydroxymethyl)piperidin-4-ol
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-ethyl-1H-indole-5-carboxamide
2-{[(3-fluoro-4-methylphenyl)formamido]methyl}-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
2-({1-[1-(4-hydroxyphenyl)propan-2-yl]piperidin-4-yl}oxy)-4-methoxy-N-(2-methoxyethyl)benzamide
2-[3-(dimethylamino)propyl]-9-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]-2,9-diazaspiro[5.5]undecan-3-one
1-(3,5-dimethylphenyl)-4-(2-methanesulfonylacetyl)piperazin-2-one
4-hydroxy-N-(2-methoxyethyl)-2-methyl-N-(pyridin-3-ylmethyl)pyrimidine-5-carboxamide
butyl (4aR,7aS)-4-[(3-methylthiophen-2-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxylate
7-(furan-3-ylmethyl)-3-(oxolan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
1-[(3R,4S)-3-amino-4-(3-methoxyphenyl)pyrrolidin-1-yl]-4-(2-methyl-1H-imidazol-1-yl)butan-1-one
3-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]quinoline
ethyl 4-[(3-methoxyphenyl)methyl]-1-(1-phenylpiperidin-4-yl)piperidine-4-carboxylate
(2-{4-[(4-ethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}-2-oxoethyl)urea
6-methyl-2-({2-oxo-2-[2-(pyridin-2-yl)pyrrolidin-1-yl]ethyl}sulfanyl)-3,4-dihydropyrimidin-4-one
4-{[3-(3-fluorophenoxymethyl)piperidin-1-yl]methyl}-1,5-dimethyl-1H-pyrrole-2-carbonitrile
2-ethoxy-5-{[3-(methanesulfonylmethyl)piperidin-1-yl]methyl}pyridine
3-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridin-2-ol
1-ethyl-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
4-(azocane-1-carbonyl)-7-fluoro-2-(2-methylpyrimidin-5-yl)quinoline
2-methoxy-1-(4-{[4-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}-1,4-diazepan-1-yl)ethan-1-one
4-methyl-N-{2-methyl-5-[2-(1H-1,2,3,4-tetrazol-1-yl)acetamido]phenyl}benzamide
N-cyclopropyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-(1-methylpiperidin-4-yl)piperidine-3-carboxamide
2-{6,8-dioxo-2,7-diazaspiro[4.4]nonane-2-carbonyl}benzonitrile
5,7-dimethyl-2-(2-methylpyrimidin-5-yl)-4-(2-methylpyrrolidine-1-carbonyl)quinoline
N-[1-(pyrazin-2-yl)propan-2-yl]-3-(pyrrolidine-1-sulfonyl)benzamide
N-[(2R,3R)-2-(pyridin-3-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-1,2-oxazole-3-carboxamide
2-(1-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-2-yl)pyridine
N-[1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-5-(3-hydroxy-3-methylbut-1-yn-1-yl)furan-2-carboxamide
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-(morpholine-4-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
(3aR,6aS)-5-[2-(3-methylphenoxy)acetyl]-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(4-phenyl-1H-pyrazol-5-yl)-1-(5-propyl-1,2-oxazole-3-carbonyl)piperidine
(4S)-3-[(3-methoxyphenyl)methyl]-4-(propan-2-yl)-1,3-oxazolidin-2-one
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-[(3S)-3-hydroxypyrrolidin-1-yl]-N,1-dimethyl-1H-1,3-benzodiazole-5-carboxamide
(2S)-1-(4-{[2-(4-methoxyphenyl)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carbonyl)pyrrolidine-2-carboxamide
1-(furan-2-carbonyl)-4-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperazine
2-[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-4-carboxylic acid
2-amino-N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}acetamide
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-N-[(4-methoxyphenyl)methyl]-2-(2-methyl-1,3-thiazol-4-yl)acetamide
7-[(3-methylphenyl)methyl]-2-(pyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
8-(1-benzothiophen-2-ylmethyl)-3-benzyl-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{4-[(2,5-dimethoxyphenyl)methyl]piperazin-1-yl}-2-[(2-fluorophenyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
2-[3-(dimethylamino)propyl]-9-(2-ethoxybenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(diethylamino)-3-{2-methoxy-5-[(4-methoxypiperidin-1-yl)methyl]phenoxy}propan-2-ol
7-[(3,4-difluorophenyl)methyl]-2-(1-methylcyclopropanecarbonyl)-2,7-diazaspiro[4.5]decan-6-one
6-(2,5-dichlorophenyl)-N,N-dimethylpyridine-3-carboxamide
3-[(3R,4S)-1-(2,3-dichlorobenzoyl)-4-(dimethylamino)piperidin-3-yl]propanoic acid