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2-methyl-5-(4-{[5-(oxan-2-yl)furan-2-yl]methyl}piperazin-1-yl)-2,3-dihydropyridazin-3-one
4-cyclopentanecarbonyl-2-(4-methylpentyl)morpholine
3-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-3-methyl-1-(1-methyl-1H-1,3-benzodiazol-6-yl)urea
methyl 2-({methyl[3-(1-methyl-1H-imidazol-2-yl)propyl]amino}methyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxylate
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)acetamide
3-(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepine-3-carbonyl)-1-methyl-1,2-dihydroquinoxalin-2-one
1-[(3-chloro-2-fluorophenyl)methyl]-4-(pyrrolidin-1-ylmethyl)piperidine
N4-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-6-methylpyrimidine-2,4-diamine
1-[(5-chloro-3-methyl-1H-indol-2-yl)methyl]azepan-4-ol
3-{[methyl({[2-(1H-pyrazol-1-yl)phenyl]methyl})amino]methyl}benzonitrile
(2-{7-cyclopentyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}-2-oxoethyl)urea
1-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}azepan-3-amine
N-cyclopentyl-N-{[4-methoxy-3-(propan-2-yloxy)phenyl]methyl}-2-methyl-1,3-thiazole-4-carboxamide
1-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-(pyridin-3-yl)piperazine
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
2-{[2-(pyridin-2-yl)pyrrolidin-1-yl]methyl}quinolin-8-ol
4-{3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}-3-(3-fluorophenyl)piperazin-2-one
1-[2-(4-chlorophenyl)ethyl]-N-(3-hydroxy-3-methylbutyl)-N-methyl-6-oxopiperidine-3-carboxamide
1-{2-[2-(1-methyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]propyl}-1H-indole
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-(pyridin-4-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
7-methyl-4-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}-3,4-dihydro-2H-1,4-benzothiazin-3-one
N-[2-(furan-2-yl)-2-(pyrrolidin-1-yl)ethyl]-1-phenyl-1H-1,2,3-triazole-5-carboxamide
2-(4-methyl-6-{[2-(2-methylpropanesulfonyl)ethyl]amino}pyrimidin-2-yl)phenol
2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-(2-methylpropyl)-N-(thiophen-3-ylmethyl)acetamide
N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]imidazo[1,2-a]pyrimidine-2-carboxamide
(5-{4-phenyl-1-[(3-propyl-1,2-oxazol-5-yl)methyl]-1H-imidazol-5-yl}furan-2-yl)methanol
2-methoxy-N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-4-carboxamide
(2S)-2-(methylamino)-1-{3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}pentan-1-one
3-[1-(5-cyclopropyl-1,3-oxazole-4-carbonyl)piperidin-3-yl]-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}(methyl){[3-(1H-pyrazol-1-yl)phenyl]methyl}amine
1,3,6-trimethyl-4-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]-1H-pyrazolo[3,4-b]pyridine
3-(2-ethylbutyl)-8-[2-(2-oxo-1,2-dihydropyridin-1-yl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-{1'-[(2-fluoro-5-methylphenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}-2-methoxyethan-1-one
N-{2-[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]ethyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
1-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
N-[(2-ethoxypyridin-3-yl)methyl]-4-hydroxy-2-(2-methyl-1,3-thiazol-4-yl)pyrimidine-5-carboxamide
1'-(3,6-dimethyl-1-benzofuran-2-carbonyl)-3,4-dihydrospiro[1-benzopyran-2,3'-pyrrolidine]-4-one
(2E)-N-{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-3-(pyridin-4-yl)prop-2-enamide
1-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecan-4-yl]-3-(dimethyl-1,2-oxazol-4-yl)propan-1-one
N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-6-(morpholin-4-yl)pyridine-3-carboxamide
9-(2H-1,3-benzodioxol-4-yl)-4-ethyl-2H,3H,4H,6H,7H,8H,9H-[1,4]oxazino[2,3-g]quinoline-3,7-dione
N-[(2-methyl-1H-indol-5-yl)methyl]-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide
2-ethyl-4-methyl-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-1,3-thiazole-5-carboxamide
methyl 3-{[(1R,2R,4R)-bicyclo[2.2.1]hept-5-en-2-ylformamido]methyl}-5-cyclohexaneamidobenzoate
2-methoxy-6-{[methyl({[5-(methylsulfanyl)-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl})amino]methyl}phenol
N-(2-{[(3S,4S)-3-hydroxy-4-(4-methylpiperazin-1-yl)pyrrolidin-1-yl]methyl}quinolin-6-yl)acetamide
5-[2-(dimethyl-1,3-thiazol-5-yl)acetyl]-N-(3-methoxypropyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-[(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)methyl]-4-(pyridin-3-yl)phenol
8-[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazole-4-carbonyl]-1-oxa-8-azaspiro[4.5]decane
1-(furan-2-ylmethyl)-N-[2-(pyridin-3-yloxy)propyl]piperidine-4-carboxamide