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2-hydroxy-N-[(1S,3S)-3-{[4-(pyridin-2-yl)pyrimidin-2-yl]amino}cyclopentyl]pyridine-3-carboxamide
4-hydroxy-1-(5-phenyl-1,2,4-oxadiazol-3-yl)piperidine-4-carboxylic acid
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-6-(1,4-oxazepan-4-yl)pyridine-3-carboxamide
5-chloro-N-[2-(1H-indol-1-yl)ethyl]-N-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
methyl (2S)-2-{[5-(tert-butylcarbamoyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridin-3-yl]formamido}-3-phenylpropanoate
[(3R,4R)-4-(pyrrolidin-1-ylmethyl)-1-(thiophene-3-carbonyl)pyrrolidin-3-yl]methanol
3-[5-({4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}methyl)thiophen-2-yl]prop-2-yn-1-ol
N-(5-phenyl-1H-1,2,4-triazol-3-yl)spiro[indene-1,4'-piperidine]-1'-carboxamide
(4aR,7aS)-1-(2-methoxyacetyl)-4-[5-(methoxymethyl)thiophene-2-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
3-[(2-fluorophenyl)formamido]-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}propanamide
6-[2-(1-ethylpiperidin-3-yl)-1H-imidazol-1-yl]-1H-indazole
N-(2-{[5-(phenoxymethyl)-1H-pyrazol-3-yl]formamido}ethyl)acetamide
2-methoxy-6-{[({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)(pyridin-3-ylmethyl)amino]methyl}phenol
(benzylsulfamoyl)[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]amine
N,N-dimethyl-2-{[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}ethane-1-sulfonamide
5-{2-benzyl-3-oxo-2,9-diazaspiro[5.5]undecane-9-carbonyl}-1-methyl-1H-pyrrole-3-carbonitrile
3-[(4,6-dimethylpyrimidin-2-yl)methyl]-1-{3-[(dimethylsulfamoyl)amino]phenyl}urea
2-(4-fluorophenyl)-4-(2-methyl-1-benzofuran-7-carbonyl)morpholine
(3S,4R)-4-methyl-3-(2-methylpropyl)-1-[5-(propan-2-yl)-1,3-oxazole-4-carbonyl]piperidin-4-ol
N-[(4-chlorophenyl)(pyridin-4-yl)methyl]-2-hydroxypyridine-3-carboxamide
5-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-3-(phenoxymethyl)-1-(propan-2-yl)-1H-1,2,4-triazole
2-[3-(2,4-dimethoxybenzoyl)piperidin-1-yl]-N-(1-methyl-1H-pyrazol-4-yl)acetamide
1-(2-chlorophenyl)-3-(1-{1-[2-(methylsulfanyl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
N-methyl-2-(methylamino)-N-[(4-phenoxyphenyl)methyl]pyrimidine-5-carboxamide
1-{6-[4-(1H-imidazol-2-yl)piperidin-1-yl]pyridin-2-yl}ethan-1-ol
3-(1-propyl-1H-1,2,3-triazol-4-yl)-1-{2-[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]ethyl}urea
N-(furan-2-ylmethyl)-2-hydroxy-N-(1-hydroxybutan-2-yl)-3-methylbenzamide
(2S)-2-amino-3-(1H-imidazol-4-yl)-1-{4-[6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}propan-1-one
2-(2H-1,3-benzodioxol-5-yl)-N-[(5-{[(3-methylphenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl]acetamide
9-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
7-[2-(2-methoxyphenyl)acetyl]-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
7-[3-(4-chloro-1H-pyrazol-1-yl)propanoyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
5-[3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-2-(pyridin-4-yl)pyrimidine
(3R,4R)-3,4-dimethyl-1-[3-(pyrrolidine-1-carbonyl)pyridin-2-yl]pyrrolidin-3-ol
N-[(1-cycloheptylpyrrolidin-3-yl)methyl]-2-(2,4-dioxoimidazolidin-1-yl)acetamide
N-(1-carbamoylcyclopentyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
8-[2-(4-chlorophenoxy)ethyl]-2-methyl-2,8-diazaspiro[4.5]decan-3-one
1-{3,3-dimethyl-2-methylidenebicyclo[2.2.1]heptane-1-carbonyl}-3-(2-fluorophenyl)pyrrolidine
2-{1-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-1H-imidazol-2-yl}quinoline
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
5-acetyl-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}thiophene-3-carboxamide
N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}-1H-1,2,4-triazole-5-carboxamide
4-[(2-benzyl-1,3-thiazol-4-yl)methyl]-1,4-oxazepane
2-[(3-fluorophenyl)methyl]-4-[4-(5-methylthiophene-2-carbonyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-5-methylthiophene-2-carboxamide
methyl 3-[4-(7-fluoro-2-methylquinoline-4-carbonyl)-2-oxo-6-(pyridin-4-ylmethoxy)-1,4-diazepan-1-yl]propanoate
6-(4-fluorophenyl)-2-(3-hydroxyazetidine-1-carbonyl)-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
N-{4-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}quinoxaline-5-carboxamide
N-[(5-chlorothiophen-2-yl)methyl]-2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide