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4-(2-ethoxypyridine-3-carbonyl)-1-(4-methoxyphenyl)-3-methylpiperazin-2-one
1-(6-methyl-1,2,3,4-tetrahydroquinolin-1-yl)-2-({2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}amino)ethan-1-one
1-(4-{[bis(2-hydroxyethyl)amino]methyl}phenoxy)-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
(4aS,7aR)-1-(1-tert-butyl-1H-pyrrole-3-carbonyl)-4-(2-methoxyacetyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}phenoxy)ethan-1-ol
2-{8-[(5-methylpyrazin-2-yl)methyl]-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}pyridine-4-carboxamide
1-[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]-N-[2-(morpholin-4-yl)ethyl]piperidin-4-amine
3-chloro-N-[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]thiophene-2-carboxamide
(1S,5R)-6-methyl-3-[3-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
6-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-3-cyclopropyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
8-(4-chloro-1-methyl-1H-indazol-3-yl)-2H,5H,6H,7H,8H-[1,3]dioxolo[4,5-g]quinolin-6-one
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}acetamide
3-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
N-(4-fluoro-2-methylphenyl)-3-(2-hydroxyethyl)-4-(2-methylpropyl)piperazine-1-carboxamide
1-[(2-chloro-5-fluorophenyl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
3-(2-aminoethyl)-4-[(3-methylphenyl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[(4aR,8aR)-1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-decahydro-1,6-naphthyridin-6-yl]-2-(2-methoxyphenyl)ethan-1-one
8-(2,6,8-trimethylquinoline-4-carbonyl)-1,3-dioxa-8-azaspiro[4.5]decan-2-one
N-{[4-(2-methoxyethoxy)phenyl]methyl}-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
2-ethyl-8-(3-methoxybenzenesulfonyl)-2,8-diazaspiro[5.5]undecan-3-one
1-[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethan-1-one
3-[methyl({5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-yl})amino]propane-1,2-diol
1-(1,3-benzoxazol-2-yl)-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}piperidin-4-amine
2-{1-[(2-chloro-4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-cyclohexylacetamide
4-(2-methoxy-2-phenylacetyl)-1-(3-methoxyphenyl)piperazin-2-one
1-(3-methanesulfonamido-4-methoxyphenyl)-3-methyl-3-[(5-methylfuran-2-yl)methyl]urea
2-[1-(cyclohexylmethyl)-4-[1-(2-methylphenyl)piperidin-4-yl]piperazin-2-yl]ethan-1-ol
4-[(3R,4S)-3-amino-4-(5-methylfuran-2-yl)pyrrolidine-1-carbonyl]oxane-4-carbonitrile
1-benzyl-3-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-3-methylurea
5-{1-cyclohexyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-3-methyl-1,2-oxazole
2-cyclopentyl-N-{2-[4-(4-fluorophenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]ethyl}acetamide
1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-3-(thiophen-2-yl)propan-1-one
3-(azepane-1-carbonyl)-1-methyl-5-(pyrrolidin-1-yl)-4,5,6,7-tetrahydro-1H-indazole
N-(4-{1-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-1H-imidazol-2-yl}phenyl)acetamide
(3-{5-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}phenyl)methanol
5-{2-[(3R,4S)-3-amino-4-propylpyrrolidin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}propan-1-one
2-{[6-(3,5-difluorophenyl)quinazolin-4-yl]amino}ethan-1-ol
2-[(2-fluoro-4-methoxyphenyl)methyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
7-cyclohexyl-2-[4-(1H-imidazol-1-yl)butanoyl]-2,7-diazaspiro[4.5]decan-6-one
3-{9-methyl-3,9-diazaspiro[5.6]dodecan-3-yl}-N-(4-methylphenyl)-3-oxopropanamide
1-[(4-fluorophenyl)methyl]-4-(4-methylpyridine-3-carbonyl)-2-(propan-2-yl)-1,4-diazepane
2-(4-methoxyphenoxymethyl)-N-[(2-methylphenyl)methyl]-1,3-oxazole-4-carboxamide
N-(2,3-dihydro-1H-inden-2-yl)-2-(2-oxo-1,2-dihydropyrimidin-1-yl)-N-propylacetamide
3-oxo-N-[1-(pyrazin-2-yl)propan-2-yl]-1,2,3,4-tetrahydroquinoxaline-6-carboxamide
methyl 4-[7-(2-cyclohexylethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-4-oxobutanoate
3-(carbamoylmethoxy)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)benzamide
2,7-dimethyl-N-(1,2-oxazol-3-ylmethyl)pyrazolo[1,5-a]pyrimidine-5-carboxamide
2-(furan-2-yl)-N-{[1,2,4]triazolo[4,3-a]pyridin-8-yl}azepane-1-carboxamide
4-[2-(pyrazin-2-yl)ethyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one