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3-[4-(pyrimidin-2-yloxy)piperidin-1-yl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraene
N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-1-(propan-2-yl)piperidine-4-carboxamide
3-(1H-imidazol-1-ylmethyl)-1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidine
[2-ethoxy-5-({[(5-ethylpyridin-2-yl)methyl](methyl)amino}methyl)phenyl]methanol
N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}-3-oxo-3,4-dihydro-2H-1,4-benzoxazine-7-carboxamide
N-[2-methoxy-2-(thiophen-2-yl)ethyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
2-(3-methoxypyrazin-2-yl)-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
N-[2-(4-hydroxyphenyl)-2-oxoethyl]-N-methyl-3-(1-methylpiperidin-3-yl)propanamide
(2-methoxyethyl)(1-{1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-2-phenylethyl)(pyridin-3-ylmethyl)amine
methyl 4-(5-{[4-(thiomorpholin-4-yl)piperidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoate
2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-hydroxyethyl)-N-methylacetamide
3-(azetidine-1-carbonyl)-N-[2-(2-fluorophenoxy)ethyl]benzene-1-sulfonamide
(2S,3S)-3-methyl-2-{5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-6-yl}pentanamide
methyl N-{[methyl({[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl})carbamoyl]methyl}carbamate
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-3-(trimethyl-1H-pyrazol-1-yl)propanamide
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-(oxan-4-ylmethyl)acetamide
N-[(2-methylpyrimidin-5-yl)methyl]-4-(morpholin-4-yl)aniline
N-[(3S,5S,9S)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]-4-fluoro-3-(trifluoromethyl)benzamide
N-{3-[4-({[3-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]formamido}methyl)-5-methyl-1,3-oxazol-2-yl]phenyl}-2-methylfuran-3-carboxamide
1-methyl-2-(morpholin-4-yl)-N-[3-(1H-1,2,3-triazol-1-yl)propyl]-1H-1,3-benzodiazole-5-carboxamide
N-({1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl}methyl)-1H-indole-2-carboxamide
2-[(2E)-2-methylbut-2-en-1-yl]-2,8-diazaspiro[4.5]decane
2-[4-({3-[benzyl(methyl)amino]piperidin-1-yl}methyl)phenoxy]ethan-1-ol
5-[1-(2-ethylbutanoyl)piperidin-4-yl]-5-(pyridin-2-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
5-[1-methyl-5-(trifluoromethyl)-1H-pyrazol-3-yl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
N-[3-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)propyl]-5-propyl-1,3,4-oxadiazol-2-amine
[(1,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)(quinoxalin-2-ylmethyl)amine
(2-methoxyethyl)[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl](propan-2-yl)amine
N-[(3S,4R)-1-[(3-cyanophenyl)methyl]-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-6-{[methyl(oxan-2-ylmethyl)amino]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
N-(oxan-4-ylmethyl)-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
N-(adamantan-2-ylmethyl)-2-oxo-6-[(4-phenylpiperidin-1-yl)methyl]-1,2-dihydropyridine-3-carboxamide
4-{1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}benzoic acid
4-cyclopropyl-6-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}pyrimidine
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-[4-(1H-1,2,4-triazol-1-yl)butanoyl]pyrrolidin-3-yl]acetamide
2-methyl-N-(4-{[1-(pyridin-4-yl)propan-2-yl]carbamoyl}phenyl)furan-3-carboxamide
1-[6-(2-amino-2-methylpropyl)-2-(dimethylamino)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-4-yl]piperidin-4-ol
(1S,5R)-3-cyclobutanecarbonyl-6-(1,2-oxazole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[1-(2,3-dihydro-1H-inden-2-yl)-2-methylpropan-2-yl]-1-[2-(dimethylamino)ethyl]-5-oxopyrrolidine-3-carboxamide
1-(5-methoxyfuran-2-carbonyl)-3-(3-methoxypropyl)piperidine-3-carboxylic acid
4-[1-(2-aminoethyl)-1H-1,2,3-triazole-4-carbonyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-1-(propan-2-yl)piperidine-4-carboxamide
(1S,6R)-9-[3-(1H-pyrazol-4-yl)benzoyl]-3,9-diazabicyclo[4.2.1]nonane
methyl 4-[({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(oxolan-2-ylmethyl)carbamoyl]butanoate
2-butyl-8-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
1-benzyl-5-[(3-methoxyphenyl)methyl]-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-[2-oxo-4-(5-phenyl-1,2-oxazole-3-carbonyl)piperazin-1-yl]benzonitrile
5-{2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetyl}-1-(2-methylpropyl)-N-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[(2,3-dimethoxyphenyl)methyl]-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-4-ol
2-[benzyl({[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl})amino]ethan-1-ol