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3-{1-[3-(morpholin-4-yl)propanoyl]piperidin-3-yl}benzoic acid
5-[3-({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)propyl]-1,3,4-thiadiazol-2-amine
N-methyl-5-{4-oxo-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-2-yl}furan-2-carboxamide
9-(1-ethyl-1H-pyrazole-4-carbonyl)-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(dimethyl-1,2-oxazol-4-yl)-N-[2-methoxy-5-(4H-1,2,4-triazol-4-yl)phenyl]pyrrolidine-1-carboxamide
1-(4-benzylpiperazin-1-yl)-3-{1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-3-yl}propan-1-one
9-[(2,6-difluoro-4-methoxyphenyl)methyl]-3-oxa-9-azaspiro[5.5]undecane
(9aR)-2-methyl-8-(3-phenylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}[3-(2-methyl-1H-imidazol-1-yl)-1-phenylpropyl]amine
1-{2-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
N-[(1-ethyl-5-oxopyrrolidin-3-yl)methyl]-N-methyl-1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
3-{[(2-chloro-5-fluorophenyl)carbamoyl]amino}-N-cyclohexylpropanamide
4-[5-({[3-(dimethylamino)propyl](methyl)amino}methyl)-1,2,4-oxadiazol-3-yl]benzoic acid
1-[2-({[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}amino)ethyl]imidazolidin-2-one
3-(3-methyl-1H-pyrazol-1-yl)-N-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]propanamide
{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
2-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]phenol
2-amino-6-[1-(4-chlorophenyl)-1H-pyrazol-4-yl]-4-(pyridin-3-yl)pyridine-3-carbonitrile
2-[3-(hydroxymethyl)-3-[(3-methoxyphenyl)methyl]piperidin-1-yl]pyridine-3-carboxamide
1-(2,4-difluorobenzoyl)-3-(2,5-dimethoxyphenyl)pyrrolidine
N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-6-[2-methyl-2-(morpholin-4-ylmethyl)propyl]-3,6-diazabicyclo[3.2.2]nonane
3-(2-chlorophenyl)-1-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]pyrrolidine
N-[(2-methoxyphenyl)methyl]-4,5-dimethyl-N-(prop-2-en-1-yl)-2-(1H-1,2,3,4-tetrazol-1-yl)thiophene-3-carboxamide
3-{5-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
3-(4-methyl-1,3-thiazol-5-yl)-1-[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]propan-1-one
2,3-dimethyl-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}quinoxaline-6-carboxamide
5-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decane-4-carbonyl]-4-phenylpyrimidin-2-amine
5-(3-fluorophenoxymethyl)-N-[(1R)-2-hydroxy-1-phenylethyl]-1H-pyrazole-3-carboxamide
[(3R,4R)-1-(1-benzofuran-2-ylmethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
2-{4-chloro-2-[(2,4-dimethyl-1,4-diazepan-1-yl)methyl]phenoxy}acetic acid
1-ethyl-4-{2-[3-(methoxymethyl)pyrrolidine-1-carbonyl]-2,3-dihydro-1H-inden-2-yl}piperazine
2-[5-(3,4-dihydro-2H-1-benzopyran-3-yl)-3-(oxan-4-yl)-1H-1,2,4-triazol-1-yl]ethan-1-ol
N-[(3-methyl-7-{2-oxo-1-oxaspiro[4.5]decane-4-carbonyl}-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]thiophene-2-carboxamide
4-(3-methylphenoxy)-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine-4-carboxylic acid
1-(2-ethoxyphenyl)-4-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine
2-(2-{[(3-hydroxy-3-phenylpropyl)(methyl)carbamoyl]amino}phenyl)-N,N-dimethylacetamide
2-amino-4,6-bis(3-hydroxyphenyl)pyridine-3-carbonitrile
{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}(methyl)[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]amine
(1S,5R)-6-(cyclopropylmethyl)-3-{[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
(2S,4R)-4-{[(3-chlorophenyl)methyl]amino}-N-(2-methoxyethyl)-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
methyl 6-[(4-acetamidophenyl)methyl]-2-[(3-methylbutyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-{2-[(4,6-dimethoxypyrimidin-2-yl)oxy]hex-5-en-1-yl}thiomorpholine
3-fluoro-4-{2-[2-(propan-2-yl)pyrimidin-4-yl]-1H-imidazol-1-yl}benzoic acid
N-({1-[(6-chloropyridin-3-yl)methyl]piperidin-3-yl}methyl)cyclopropanesulfonamide
3-(2-fluoro-4-methoxyphenyl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]urea
N,N,3-trimethyl-2-{[4-(propan-2-yl)pyrimidin-2-yl]amino}butanamide
2-fluoro-N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)-5-sulfamoylbenzamide
2-{2-[3-(cyclopentylcarbamoyl)propanamido]ethyl}-1,3-thiazole-4-carboxylic acid
4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-methanesulfonylpiperidine