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N-[2-hydroxy-3-(3-methoxyphenoxy)propyl]-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
3-ethyl-1-(2-fluorophenyl)-3-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)urea
N-ethyl-5-(morpholin-4-ylmethyl)-N-(propan-2-yl)-1,2-oxazole-3-carboxamide
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-2-(pyridin-3-yl)acetamide
methyl 3-{methyl[(1-methylpiperidin-2-yl)methyl]carbamoyl}benzoate
(2E)-3-(2-chlorophenyl)-N-[(5-{[(4-fluorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]prop-2-enamide
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-4-methoxy-N,3-dimethylbenzamide
5-(1H-imidazol-1-ylmethyl)-N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]pyridin-2-amine
7-cyclopropanecarbonyl-N-methyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-[(3R,4S)-4-cyclopropyl-1-(2-methanesulfonylethyl)pyrrolidin-3-yl]-4-methylbenzamide
5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-(oxan-4-ylmethyl)pyridin-2-amine
N-{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-1,1-dioxo-1λ6-thiane-4-carboxamide
3-chloro-2-{3-[1-(2-ethoxyethyl)-1H-pyrazol-3-yl]phenyl}pyridine
(4aS,7aR)-N-(4-acetylphenyl)-4-ethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
2-{1-benzyl-4-[2-(methylamino)-1,3-thiazole-4-carbonyl]piperazin-2-yl}ethan-1-ol
1-cyclopentanecarbonyl-N-[1-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]piperidine-4-carboxamide
5-[2-(2,6-dichlorophenyl)-1H-imidazol-1-yl]pentan-1-amine
7-chloro-N-(5-methyl-1,3,4-thiadiazol-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carboxamide
4-[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]-1-(pyridin-2-ylmethyl)pyrrolidin-2-one
1-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidin-1-yl]-3-(5-methyl-1H-pyrazol-1-yl)propan-1-one
4-(1-{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}piperidine-3-carbonyl)morpholine
5-[2-(2,4,5-trimethoxyphenyl)-1H-imidazol-1-yl]-1H-1,2,3-benzotriazole
2-cyclohexyl-1-[3-(pyrrolidin-1-ylmethyl)piperidin-1-yl]ethan-1-one
(1S,5R)-6-[4-(morpholin-4-yl)benzoyl]-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
4-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]-2-methoxypyridine-3-carbonitrile
1-(1,4-dioxan-2-ylmethyl)-2-[3-(1H-pyrazol-1-ylmethyl)phenyl]-1H-imidazole
N-{4-[2-(4-hydroxypiperidin-1-yl)acetamido]phenyl}pentanamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N,2-dimethyl-1-benzofuran-5-carboxamide
2-benzyl-8-[(3E)-pent-3-enoyl]-2,8-diazaspiro[5.5]undecan-3-one
3-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-N-methylpyridin-2-amine
5-(2-chloro-6-fluorophenyl)-3-cyclopropyl-1-[(4-methoxyphenyl)methyl]-1H-1,2,4-triazole
4-[(dimethylamino)methyl]-N-[1-(methoxymethyl)cyclopentyl]benzamide
N-({3-methyl-7-[2-(2-phenyl-1,3-thiazol-4-yl)acetyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)propane-1-sulfonamide
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N-methyl-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
4-{3-[1-(4-fluorobutyl)-1H-pyrazol-3-yl]phenyl}pyridine
2-amino-6-(4-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperazin-1-yl)pyrimidin-4-ol
4-(3-cyano-1H-pyrazol-4-yl)benzamide
1-(cyclohex-1-en-1-ylmethyl)-3-[4-(3-methylpiperidine-1-carbonyl)phenyl]urea
N-[(1-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}piperidin-3-yl)methyl]cyclobutanecarboxamide
8-fluoro-2-[4-(2-methylphenyl)-1,4-diazepane-1-carbonyl]quinoline
1-[3-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-3-oxopropyl]azepan-2-one
2-(4-methyl-1,4-diazepan-1-yl)-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}acetamide
2-[(4-{2-[3-(methoxymethyl)pyrrolidine-1-carbonyl]phenoxy}piperidin-1-yl)methyl]pyridine
2-(3-{[2-(pyridin-3-ylmethyl)pyrrolidin-1-yl]methyl}phenyl)-3H,4H,5H,6H,7H-cyclopenta[d]pyrimidin-4-one
4-{[(4aS,7aR)-4-(carboxymethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]methyl}-5-methyl-1,2-oxazole-3-carboxylic acid
4-{1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carbonyl}piperazin-2-one
N-{1-[1-(cyclohex-3-ene-1-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methylbenzamide
N-methyl-4-sulfamoyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)butanamide
(1R,5R)-3-(2H-1,3-benzodioxole-5-carbonyl)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonane
1-{1-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}piperidin-4-ol