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3-(1H-imidazol-2-yl)-1-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]piperidine
2-{1-methyl-4-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-10-oxo-1,4,9-triazaspiro[5.6]dodecan-9-yl}acetic acid
N-(3-methoxypropyl)-4-{[(1-methyl-1H-pyrazol-4-yl)methyl]sulfamoyl}benzamide
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-3-(pyrazin-2-yl)propanamide
(2S,4R)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-(2-methylpropyl)-4-({[4-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
2-ethyl-4-methyl-5-({4-[2-(methylsulfanyl)ethyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)-1H-imidazole
[2-(4-methoxyphenyl)ethyl][(4-methylphenyl)methyl][(1-methylpiperidin-4-yl)methyl]amine
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)oxolane-3-carboxamide
N-[(3S,4R)-1-{[2-(methylsulfanyl)phenyl]methyl}-4-propylpyrrolidin-3-yl]acetamide
6-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-yl]-N,N-dimethylpyrazine-2-carboxamide
2-[(1,1-dioxo-1λ6-thiolan-3-yl)(methyl)amino]-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}acetamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-2-{3-oxo-1-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}acetamide
2-[2-({methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]amino}methyl)phenoxy]-1-(piperidin-1-yl)ethan-1-one
N-ethyl-5-({[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl](methyl)amino}methyl)pyrimidin-2-amine
2-fluoro-N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-5-sulfamoylbenzamide
1-(3-methylpiperidin-1-yl)-3-{[2-(pyridin-2-yl)ethyl]amino}propan-1-one
1-methyl-4-{[3-(methylsulfanyl)phenyl]methyl}-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
3-(2,2-difluoro-2H-1,3-benzodioxol-5-yl)-1-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)urea
N-{[4-(butan-2-yloxy)phenyl]methyl}-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
N-(1,3-benzothiazol-2-ylmethyl)-2-tert-butyl-4-hydroxy-N-methylpyrimidine-5-carboxamide
2-[5-(ethoxymethyl)-3-(oxan-4-yl)-1H-1,2,4-triazol-1-yl]ethan-1-ol
{4-[(4-fluoro-3-methoxyphenyl)methyl]morpholin-3-yl}methanol
(2,1,3-benzoxadiazol-4-ylmethyl)(methyl){[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}amine
1-(butane-1-sulfonyl)-4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
(2S,4S)-N-ethyl-4-(2-methoxyacetamido)-1-[3-(2-methylphenyl)propanoyl]pyrrolidine-2-carboxamide
8-methoxy-2-(1H-pyrazol-3-yl)quinoline
2-{2-[3-(6-methoxynaphthalene-2-carbonyl)piperidin-1-yl]ethyl}pyridine
N-cyclohexyl-N-[2-(dimethylamino)ethyl]-4-(3-hydroxy-3-methylbutyl)benzamide
9-(6-methylpyridine-2-carbonyl)-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
2-chloro-4-[1-(2-fluoroethyl)-4-phenyl-1H-imidazol-5-yl]-6-methoxyphenol
(3aR,7aS)-5-methyl-2-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)-2,3,3a,4,7,7a-hexahydro-1H-isoindole
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-N-(prop-2-en-1-yl)acetamide
3-(diphenylmethyl)-4-(4-methoxyphenyl)-4H-1,2,4-triazole
4-{2-[1-(3-methoxybenzenesulfonyl)piperidin-2-yl]ethyl}morpholine
N-[2-(3-methoxy-4-propoxyphenyl)ethyl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
[1-(2-aminopyrimidin-4-yl)-4-(3-phenylpropyl)piperidin-4-yl]methanol
(1-benzothiophen-2-ylmethyl)(methyl)({4-methyl-5-[(2-phenoxyethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)amine
methyl 2-hydroxy-6-(1H-imidazol-1-yl)quinoline-4-carboxylate
(3S,4S)-4-[4-(3-methyl-1-propyl-1H-pyrazol-4-yl)-1H-1,2,3-triazol-1-yl]-1-(propan-2-yl)pyrrolidin-3-ol
2-(4-{[1-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-1-(3-methylbut-2-en-1-yl)piperazin-2-yl)ethan-1-ol
(5S,9aS,9bS)-2-cyclopentyl-5-[1-(3-fluorophenyl)-1H-pyrazol-4-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-(methoxymethyl)-6-[5-(thiophen-2-yl)thiophen-2-yl]pyrimidine
(3S,9aR)-3-(1H-imidazol-4-ylmethyl)-8-(quinolin-6-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-(5-cyclopropyl-1,2-oxazole-3-carbonyl)-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
4-{[1-(1H-pyrazol-3-ylmethyl)piperidin-4-yl]oxy}-N-(pyridin-2-ylmethyl)benzamide
3-{1-[5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carbonyl]piperidin-4-yl}-1,3-oxazolidin-2-one
1-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-3-(3,5-dimethyl-1H-pyrazol-4-yl)propan-1-one
[1-(azepan-1-yl)propan-2-yl][(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]amine