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3-(3-fluorophenyl)-N-[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]-1H-pyrazole-4-carboxamide
2-[2-(dimethylamino)-6-methylpyrimidin-4-yl]-7-propyl-2,7-diazaspiro[4.5]decan-6-one
5-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-2-methylphenol
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
5-(1-{8-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carbonyl}pyrrolidin-2-yl)thiophene-2-carboxamide
N-methyl-4-(4-methylphenyl)-5-[3-(morpholin-4-ylmethyl)phenyl]pyrimidin-2-amine
1-[1-(2-aminoethyl)-1H-1,2,3-triazole-4-carbonyl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
1-cyclobutanecarbonyl-N-[3-(pyridin-3-yloxy)propyl]piperidine-4-carboxamide
2-[methyl(pyridin-4-ylmethyl)amino]-1-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}ethan-1-one
3-{[(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}benzonitrile
N-[2-(3-hydroxy-4-methoxyphenyl)ethyl]-4-(4-methylpiperazin-1-yl)benzamide
N-{[2-(diethylamino)pyridin-3-yl]methyl}-1H-indole-3-carboxamide
N-[(2,5-dimethoxyphenyl)methyl]-2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]acetamide
4-[(1-acetylpiperidin-4-yl)oxy]-3-methoxy-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(propan-2-yl)benzamide
2-benzyl-N-[(2-chloropyridin-3-yl)methyl]-N-methyl-1,3-thiazole-4-carboxamide
1-(3-{[3-(hydroxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}phenoxy)-3-(morpholin-4-yl)propan-2-ol
2-{1-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]pyrrolidin-2-yl}pyridine
1-[3-ethyl-3-(hydroxymethyl)piperidin-1-yl]-2-[4-(3-methylphenyl)piperazin-1-yl]ethan-1-one
N-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-1H-indazol-5-amine
(3R,4S)-1-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-4-(5-methylfuran-2-yl)pyrrolidin-3-amine
methyl[(1-methyl-1H-imidazol-5-yl)methyl][(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]amine
(2R,6R)-4-(2-ethoxyethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
(2R)-2-methyl-1-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)piperazine
N3-ethyl-N5-({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
N-[2-(1H-indol-3-yl)ethyl]-2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carboxamide
[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl][(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]methylamine
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N-methyl-1-benzothiophene-5-carboxamide
8-(3-methoxypropyl)-N-(2-methylphenyl)-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxamide
2-[(2,3-dihydro-1,4-benzodioxin-2-ylformamido)methyl]-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
(1S,5R)-6-[2-methyl-2-(morpholin-4-yl)propyl]-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-[(2-fluorophenyl)methyl]-N-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidin-3-amine
2-[2-ethoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]pyridine-4-carbonitrile
5-{[benzyl(methyl)amino]methyl}-N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N-methyl-1,2-oxazole-3-carboxamide
{4-[(1-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}pyrrolidin-3-yl)methyl]phenyl}methanol
methyl 2-[1-(2,8-dimethylquinoline-3-carbonyl)-3-oxopiperazin-2-yl]acetate
N-{2-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-en-2-ylformamido]ethyl}-2,2,2-trifluoroacetamide
(butan-2-yl)[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl](pyridin-4-ylmethyl)amine
(3aR,6aR)-2-methyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
2-(3-hydroxypropyl)-9-[5-(propan-2-yl)pyrimidin-4-yl]-2,9-diazaspiro[5.5]undecan-3-one
(2S,4R)-N,N-diethyl-4-(2-oxo-2-phenylacetamido)-1-(propan-2-yl)pyrrolidine-2-carboxamide
N-methyl-N'-[2-(methylsulfanyl)phenyl]-N-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}butanediamide
N-[(2-chloro-6-fluorophenyl)methyl]-N-cyclopropyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
N-(3-chloro-4-methoxyphenyl)-3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidine-1-carboxamide
2-[(3-chlorophenyl)methyl]-N-[1-(pyrazin-2-yl)propan-2-yl]-1,3-benzoxazole-6-carboxamide
1-({5-[(3-fluoro-5-methylphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3,3-dimethylurea
N-phenyl-1-({4-[2-(pyrimidin-5-yl)ethynyl]phenyl}methyl)piperidin-3-amine
1-butyl-3-(8-fluoro-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-1-(pyridin-3-ylmethyl)urea
{[2-(cyclopentyloxy)phenyl]methyl}[2-methoxy-1-(pyridin-2-yl)ethyl]methylamine
2-(4-methylpiperidin-1-yl)-5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]pyridine
3-(pentan-2-yl)-8-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one