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2-acetyl-8-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-1-[4-(pyrimidin-2-yl)piperazin-1-yl]propan-1-one
2-[(3E)-hex-3-enamidomethyl]-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
3-(2-methylphenyl)-1-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}pyrrolidin-3-ol
3-{[(cyclohexylmethyl)amino]methyl}-1-[(4-fluorophenyl)methyl]-3-hydroxypiperidin-2-one
4-amino-2-(2,3-dihydro-1,4-benzodioxin-6-yl)pyrimidine-5-carbonitrile
1-benzyl-8-[(3-methylthiophen-2-yl)methyl]-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-({2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}carbamoyl)benzoic acid
2-[(2-{octahydro-1H-pyrido[1,2-a]piperazin-2-ylmethyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl)methyl]-1H-imidazole
2-ethyl-5-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}pyrimidine
1-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]-4-phenylbutan-1-one
(1S,5R)-6-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
6-{2-[2-(propan-2-yl)pyrimidin-4-yl]-1H-imidazol-1-yl}-1H-indazole
methyl 1-({[3-ethyl-4-(4-fluorophenyl)-1-methyl-1H-pyrazol-5-yl]carbamoyl}methyl)-1H-pyrazole-3-carboxylate
1-{2-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]pyrimidin-4-yl}piperidin-4-ol
4-({4-[5-chloro-2-(piperidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)pyridine
N-[2-(morpholin-4-yl)ethyl]-5-[3-(trifluoromethyl)phenoxymethyl]-1H-pyrazole-3-carboxamide
1-cyclopentanecarbonyl-4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-ethyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-4-oxo-1,4-dihydroquinoline-2-carboxamide
3-(3-tert-butyl-1-methyl-1H-pyrazol-5-yl)-1-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]urea
5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-[1-(thiophen-2-yl)propyl]-1H-pyrazole-3-carboxamide
N-(3-chloro-4-methoxyphenyl)-3-{1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]piperidin-3-yl}propanamide
2-[4-(3-chlorophenyl)-3-oxopiperazin-1-yl]-N-[(2-methylphenyl)methyl]acetamide
N-(butan-2-yl)-4-fluoro-3-hydroxy-N-(pyridin-3-ylmethyl)benzamide
4-{3-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridine-1-carbonyl]phenyl}-2-methylbutan-2-ol
N-{2-[3-cyclopropyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]ethyl}-2-fluorobenzamide
3-(4-methyl-1,3-thiazol-5-yl)-1-[(1S,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
N-{1-[(2-methyl-1,3-oxazol-4-yl)methyl]piperidin-4-yl}methanesulfonamide
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-2-phenyl-2-(1H-1,2,3,4-tetrazol-1-yl)acetamide
N-(4-{[2-(2-methoxyphenyl)ethyl]carbamoyl}-2-methylphenyl)furan-2-carboxamide
1-(2-chlorophenyl)-3-{1-[1-(3-phenylprop-2-ynoyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
[(2S)-1-{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl]methanol
N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-1-benzothiophene-5-carboxamide
N-{2-[cyclopentyl(methyl)amino]ethyl}-1-ethyl-N-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
1-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(methylsulfanyl)ethan-1-one
3-(furan-2-yl)-1-[2-(3-phenylpropyl)morpholin-4-yl]propan-1-one
N'-cycloheptyl-N'-methyl-N-(1,3,4-thiadiazol-2-yl)butanediamide
1-{4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
2-(4-methylphenyl)-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]quinoline-4-carboxamide
9-[4-(hydroxymethyl)benzoyl]-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
N-cyclopropyl-4-{[(2,3-dimethoxyphenyl)methyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
6-[1-(7-methoxy-4-methylquinazolin-2-yl)piperidin-3-yl]-2-methylpyrimidin-4-ol
4-(1-methyl-1H-imidazol-2-yl)-1-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-1H-1,2,3-triazole
8-(1,4-dithiepan-6-yl)-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}-N-(2-methoxyethyl)-1H-pyrrole-3-carboxamide
2-(cyclohex-1-en-1-yl)-N-{[4-fluoro-7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
4-ethyl-3-(1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
8-[2-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)ethoxy]quinoline
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}({1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl})amine
3-{[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}-2-(4-methoxyphenyl)-7-methylquinoline