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(3R,4R)-4-(azepan-1-yl)-1-[(2-chloro-3,4-dimethoxyphenyl)methyl]piperidin-3-ol
(1R,5R)-6-benzyl-3-[4-(trifluoromethyl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
N-cyclopentyl-3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]propanamide
5-(2-methoxyphenoxymethyl)-N-(2,2,6,6-tetramethylpiperidin-4-yl)-1H-pyrazole-3-carboxamide
[(3R,4R)-1-[(5-cyclopentylthiophen-2-yl)methyl]-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
N-[2-(2-fluorophenyl)ethyl]-2-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidine-1-carboxamide
(2S,4S)-4-amino-N,N-diethyl-1-[2-(4-methyl-2-oxo-1,2-dihydroquinolin-1-yl)acetyl]pyrrolidine-2-carboxamide
{1-[(1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidin-3-yl)methyl]-1H-1,2,3-triazol-4-yl}methanol
ethyl 1-(1-acetylpiperidin-4-yl)-4-(2-phenoxyethyl)piperidine-4-carboxylate
1-[2-({2-[1-(4-methoxyphenyl)-1H-imidazol-2-yl]-1H-imidazol-1-yl}methyl)morpholin-4-yl]ethan-1-one
1'-[5-(morpholin-4-ylmethyl)furan-3-carbonyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
3-cyclopropyl-5-[2-(3-methoxyphenyl)ethyl]-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
N-methyl-N-[3-(oxolan-2-yl)propyl]imidazo[1,2-a]pyridine-6-carboxamide
4-(naphthalen-2-ylmethyl)-3-[2-oxo-2-(4-phenylpiperazin-1-yl)ethyl]piperazin-2-one
2-(3-methoxyphenyl)-1-[3-(3-methoxypropyl)piperidin-1-yl]ethan-1-one
6-ethyl-N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-methyl-N-(4-methyl-1-phenylpentyl)-1,2,3-thiadiazole-4-carboxamide
(3R)-1-{[2-(2,5-dimethoxyphenyl)-8-methylquinolin-3-yl]methyl}pyrrolidin-3-ol
8-(1-methyl-1H-pyrazole-4-carbonyl)-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
3-[4-(4-methoxyphenyl)-3,3-dimethylpiperazine-1-carbonyl]-1,5,6-trimethyl-1,2-dihydropyridin-2-one
(1-{[2-(furan-2-yl)phenyl]methyl}piperidin-4-yl)methanamine
1-[(2-hydroxy-3-methoxyphenyl)methyl]-3-(2-methylphenyl)pyrrolidin-3-ol
N-[2-(3-benzyl-1,2,4-oxadiazol-5-yl)ethyl]-2-ethylpyrimidine-5-carboxamide
1-[(1-ethylpyrrolidin-2-yl)methyl]-3-methyl-1,2-dihydroquinoxalin-2-one
2-(3-chlorophenyl)-1-(4-cyclopentyl-1,4-diazepan-1-yl)-2-hydroxyethan-1-one
(3-{2-[1-(1-benzofuran-5-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)dimethylamine
(1S,5R)-6-[(2-ethoxyphenyl)methyl]-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-[3-(morpholin-4-yl)propyl]-3-(1H-pyrazol-4-yl)propanamide
N-[(5-ethylpyridin-2-yl)methyl]-N-methyl-5-[3-(trifluoromethyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
4-[(2-ethylpyrimidin-5-yl)methyl]-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-(4-{4-[(2,2-dimethyloxan-4-yl)amino]piperidin-1-yl}phenyl)-2-(4-methoxyphenyl)acetamide
ethyl 4-(dimethyl-1,3-oxazole-5-amido)piperidine-1-carboxylate
2-(butylsulfanyl)-N4-[(1-methylpyrrolidin-3-yl)methyl]pyrimidine-4,6-diamine
N-methyl-2-{8-methylimidazo[1,2-a]pyridin-3-yl}-N-[1-(pyridin-3-yl)pentyl]acetamide
5-(2-methoxyquinolin-3-yl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-ethyl-N-methyl-2-{[1-(morpholin-4-yl)hex-5-en-2-yl]oxy}pyrimidin-4-amine
5-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyrazin-2-ol
2-cyclopentyl-N-[1-(4-methyl-5-{[(2-methylphenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl)ethyl]acetamide
N-[(4-methoxynaphthalen-1-yl)methyl]-N,2-bis(propan-2-yl)pyrimidine-5-carboxamide
2-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
1-methyl-N-[6-(propan-2-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]-1H-imidazole-2-carboxamide
methyl (2R,4S)-4-hydroxy-1-[2-methyl-2-(phenylamino)propanoyl]piperidine-2-carboxylate
2-(adamantan-1-yl)-5-(3-ethylpiperazine-1-carbonyl)pyrimidin-4-ol
6-[4-(3-methylpyridin-4-yl)-1,4-diazepane-1-carbonyl]quinoxaline
N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
1-(2-methoxyethyl)-N-{[1-(4-methoxyphenyl)cyclopentyl]methyl}-6-oxopiperidine-3-carboxamide
4-{2-propyl-3H-imidazo[4,5-b]pyridin-3-yl}-1-[4-(trifluoromethyl)benzenesulfonyl]piperidine
2-ethyl-4-{[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}pyrimidine
8-fluoro-2-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]quinoline
N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-4-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]butanamide