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(3R,9aR)-8-(4-chlorobenzoyl)-3-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
9-(cyclopropylmethyl)-4-[4-(hydroxymethyl)benzoyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-methyl-4-(4-{[4-(pyridin-4-yl)piperazin-1-yl]methyl}phenyl)butan-2-ol
1'-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)spiro[indene-1,4'-piperidine]
6-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)-5,6-dihydro-1,6-naphthyridin-5-one
3-(1-methyl-1H-pyrrol-2-yl)-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]-1H-pyrazole-5-carboxamide
2-{1-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]pyrrolidin-2-yl}-6-methyl-1H-1,3-benzodiazole
(4aR,7aS)-1-methyl-4-(1,3,7-trimethyl-1H-indole-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(7S,9aR)-N-cyclohexyl-7-ethyl-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
2-(5-fluoro-1-methyl-1H-indole-2-carbonyl)-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
2-({[(2-methoxyphenyl)methyl](propyl)amino}methyl)benzoic acid
4-({[7-(furan-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}methyl)-1,3-thiazol-2-amine
(3S,4R)-4-(2-methoxyphenyl)-1-[3-(pyridin-2-yl)propanoyl]pyrrolidine-3-carboxylic acid
N-({7-fluoro-2-[4-(3-methoxyphenyl)piperazin-1-yl]quinolin-3-yl}methyl)-N-(2-methoxyethyl)acetamide
2-[(2S)-2-amino-3-hydroxypropanoyl]-N-(5-methyl-1,3,4-thiadiazol-2-yl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
3-(4-methoxyphenyl)-3-phenyl-N-(pyrimidin-4-ylmethyl)propanamide
(2R,3S,6R)-3-phenyl-5-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}-1,5-diazatricyclo[5.2.2.02,6]undecane
1-{1-[1-(pyridin-2-yl)propan-2-yl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
N-{2-chloro-4-[2-(2-hydroxyphenoxy)acetamido]phenyl}propanamide
4-hydroxy-2-{[methyl(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)amino]methyl}quinoline-6-carboxamide
4-(2-cyclopropyl-1H-imidazol-1-yl)-N-ethyl-N-phenylbenzamide
3-methyl-5-[4-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)phenyl]-4H-1,2,4-triazole
5-(2-fluorophenyl)-N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
2-[(2R,3R)-2-hydroxy-3-(pyrrolidin-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]pyridine-3-carbonitrile
1-{4-oxo-4-[3-(2-phenylethyl)piperidin-1-yl]butyl}piperidin-2-one
2-{4-[benzyl(methyl)amino]-6-oxo-1,6-dihydropyridazin-1-yl}-N-(1-ethyl-1H-1,2,3-triazol-4-yl)acetamide
5-(2H-1,3-benzodioxol-5-ylmethyl)-3-[3-(4-fluorophenyl)oxolan-3-yl]-1,2,4-oxadiazole
2-({7-hydroxy-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}sulfanyl)-1-[(1R,3S,5S)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl]ethan-1-one
N-methyl-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
3-({4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridin-2-amine
3-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]propan-1-one
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-2-(2,5-dioxoimidazolidin-1-yl)acetamide
2-methyl-N-(2-{2-methyl-1-azatricyclo[6.3.1.04,12]dodeca-2,4,6,8(12)-tetraen-3-yl}ethyl)-1,3-thiazole-4-carboxamide
N-[2-(1H-indol-1-yl)ethyl]-N-methyl-2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
5-[(2-fluoro-3-methylphenyl)methyl]-2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
2-butyl-5-[4-(2-fluorophenoxy)piperidine-1-carbonyl]-1,3-benzoxazole
(1S,5R)-3-(5-chloro-2-methoxybenzoyl)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{[1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}-5-(trifluoromethyl)-1,2-dihydropyridin-2-one
N-methyl-2-{5-[3-(3-methylbutoxy)phenyl]-4-phenyl-1H-imidazol-1-yl}acetamide
1-[(1-ethyl-1H-imidazol-5-yl)methyl]-2-oxo-3-[2-(pyridin-2-yl)ethyl]-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
(2S,4S,5R)-5-(4-chlorophenyl)-4-(cyclopropylcarbamoyl)-1,2-dimethylpyrrolidine-2-carboxylic acid
N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxamide
2-[4-methyl-2-(1H-pyrazol-1-yl)phenyl]-2-(morpholin-4-yl)acetic acid
4-[(4-methyl-5-{1-[(2-methylphenyl)methyl]piperidin-3-yl}-4H-1,2,4-triazol-3-yl)methyl]morpholine
N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-2,3-dihydro-1,4-benzodioxine-2-carboxamide
{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}(methyl)[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amine
3-(4-methoxyphenyl)-N-methyl-N-(2-methylpropyl)-3-phenylpropanamide
N-[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]-6-methoxy-1-methyl-1H-indole-2-carboxamide
N,N-dimethyl-5-({7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}methyl)-1,3-thiazol-2-amine
1-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-2-[methyl(pyridin-4-ylmethyl)amino]ethan-1-one