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5-[3-(1H-pyrazol-1-yl)phenyl]furan-2-carboxamide
4-[3-(benzyloxy)azetidine-1-carbonyl]-2,6-dimethylquinoline
N-{2-methyl-1-oxo-1-[2-(pyridin-2-yl)pyrrolidin-1-yl]propan-2-yl}thiophene-2-carboxamide
2-[4-(2-oxopyrrolidin-1-yl)piperidin-1-yl]-N-(pyridin-2-ylmethyl)acetamide
7-fluoro-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2-(1H-pyrazol-4-yl)quinoline-4-carboxamide
3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-1-[4-(3-phenylpropyl)-1,4-diazepan-1-yl]propan-1-one
N-[2-(1,3-thiazol-2-yl)ethyl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
3-methyl-N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
N-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-[3-(methylsulfanyl)propyl]-3-[(oxan-3-yl)sulfamoyl]benzamide
6-[(2H-1,3-benzodioxol-5-yloxy)methyl]-3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
10-methoxy-5-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-6-{[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amino}pyridine-3-carboxamide
{2-[4-(piperidin-1-ylmethyl)phenyl]phenyl}methanol
N-[2-(pyrrolidine-1-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]pyridine-2-carboxamide
2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]-N-[1-(2-phenylethyl)piperidin-3-yl]acetamide
4-ethyl-1-methyl-3-{[1-(thiophene-2-sulfonyl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
(2R,6R)-4-[3-(4-chloro-1H-pyrazol-1-yl)propanoyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
[3,3-dimethyl-1-(pyridin-3-yl)butyl]({[2-(3-methylphenyl)pyrimidin-5-yl]methyl})amine
7-(cyclopropylmethyl)-2-(1-methyl-4-phenylpiperidine-4-carbonyl)-2,7-diazaspiro[4.5]decane
3-[1-(4-chloro-1H-pyrazole-3-carbonyl)piperidin-3-yl]-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(2,6-dioxo-1,3-diazinan-1-yl)-N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]acetamide
ethyl 2-{[5-(2-amino-3-cyano-5,6,7,8-tetrahydroquinolin-4-yl)pyrimidin-2-yl]amino}acetate
5-(2-chloro-4-fluorophenoxymethyl)-N-cyclopentyl-1,2-oxazole-3-carboxamide
8-[1-(4-methoxyphenyl)cyclopropanecarbonyl]-2,8-diazaspiro[4.5]decan-3-one
4-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-methylpyridine
1-(2-cyclopropylacetyl)-4-(2-fluorophenoxy)piperidine-4-carboxylic acid
2-(4-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1-(thiophen-2-ylmethyl)piperazin-2-yl)ethan-1-ol
3-amino-1-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}pyrrolidine-3-carboxylic acid
1-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}-4-(piperidin-1-yl)piperidine-4-carboxamide
N-[(3R,4R)-3-hydroxy-1-[2-(2-methoxyphenyl)acetyl]piperidin-4-yl]pyrazine-2-carboxamide
1'-benzyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,3'-pyrrolidine]
1-{1-[(3-methylphenyl)methyl]-3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl}cyclopropane-1-carboxamide
4-{3-[3-methyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]phenyl}-1λ6-thiomorpholine-1,1-dione
(1R,3S)-3-(2-aminoethoxy)-7-(4-fluorobenzenesulfonyl)-7-azaspiro[3.5]nonan-1-ol
N-(furan-2-ylmethyl)-N,1-dimethyl-5-{[(5-phenyl-1,2-oxazol-3-yl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[3-(pyrrolidin-1-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
{2-propoxy-5-[3-(1H-pyrazol-3-yl)phenyl]phenyl}methanol
2-(dimethyl-1,3-thiazol-5-yl)-N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]acetamide
1-(3-{[(3-acetamido-4-fluorophenyl)carbamoyl]amino}propyl)piperidine-4-carboxamide
1-[4-(3-methylphenyl)phenyl]-3-[(5-oxopyrrolidin-2-yl)methyl]-3-(propan-2-yl)urea
3-{2-[(4-methylphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[1-(thiophen-2-yl)propyl]propanamide
2-(2-chloro-6-methoxyphenyl)-5-methylpyrimidin-4-amine
2-(2-ethyl-4-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]acetamide
N-cyclohexyl-3-(2,5-dioxoimidazolidin-4-yl)-N-(pyridin-2-ylmethyl)propanamide
[4-({1-[4-(morpholine-4-carbonyl)pyridin-2-yl]pyrrolidin-3-yl}methyl)phenyl]methanol
N-{1-[1-(3,5-dimethyl-1H-pyrrole-2-carbonyl)piperidin-4-yl]-2-(3-methoxyphenyl)ethyl}-N-methylfuran-2-carboxamide
2-(2-hydroxyethyl)-8-(7-methyl-1-benzofuran-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-2-(3-methyl-5-oxo-1-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl)acetamide
1-{2-[3-(benzyloxy)azetidin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydroquinolin-2-one