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[({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)sulfamoyl](ethyl)methylamine
4-{1-[(2,3-difluoro-6-methoxyphenyl)methyl]piperidin-4-yl}pyrimidine
3-methoxy-1-{1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}propan-1-one
{[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[4-(trifluoromethyl)phenyl]methyl}amine
N-benzyl-6-[4-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
2-{[5-(propane-2-sulfonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-2,3-dihydro-1H-isoindole
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
5-(3,6-dimethyl-1-benzofuran-2-yl)-3-(oxan-4-yl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
2-[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]quinoxaline
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[(1-ethylpyrrolidin-3-yl)methyl]-N-methyl-1,3-oxazole-4-carboxamide
2-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-1,2,3,4-tetrahydroisoquinoline
4-{[1-(but-3-enoyl)piperidin-4-yl]oxy}-3-chloro-N-cyclopentylbenzamide
2-(2-chlorophenyl)-N-ethyl-3-methyl-N-propyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
(5S)-5-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-2-one
2-(3-fluorophenyl)-1-[(3R,4R)-3-hydroxy-4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]ethan-1-one
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-{2-[(4-methoxynaphthalen-1-yl)methyl]-5-oxopyrrolidin-2-yl}-N-methylpropanamide
2-(3-fluoro-4-hydroxyphenyl)-1-[2-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]ethan-1-one
{7-[6-(propan-2-yl)pyridazin-3-yl]-2,3-dihydro-1-benzofuran-2-yl}methanamine
N-[4-(1H-pyrazol-1-yl)phenyl]-6-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)-6-azaspiro[2.5]octane-1-carboxamide
(1S,5R)-6-benzyl-3-[2-(2-methylphenoxy)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{4-chloro-3-[3-(hydroxymethyl)-3-(2-methylpropyl)piperidine-1-carbonyl]phenyl}acetamide
[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl](methyl)(thiophen-3-ylmethyl)amine
1,3-dimethyl-N-[2-(1H-pyrazol-4-yl)ethyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
(2S)-N-(8-chloroquinolin-5-yl)-2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carboxamide
3-[2-methyl-6-(4H-1,2,4-triazol-4-yl)pyridin-3-yl]-5-[2-(piperidin-2-yl)ethyl]phenol
4-(5-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)-1-methylpiperazin-2-one
N3-ethyl-1-(2-methylpropyl)-4-oxo-N5-(2-phenylpropyl)-1,4-dihydropyridine-3,5-dicarboxamide
4-chloro-N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-1H-pyrazole-3-carboxamide
4-(2-methoxyethyl)-1-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}-1,4-diazepan-5-one
1-({[3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]amino}methyl)cyclohexan-1-ol
1-{2-cyclopentyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-1,4-diazepan-5-one
3-(2-fluorophenyl)-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]propanamide
N-tert-butyl-3-(cyclopentylamino)-5-(4-methyl-1,4-diazepane-1-carbonyl)benzene-1-sulfonamide
2-{[5-(2-methylpropyl)-4-(1-phenylethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
(1S,5R)-3-[3-(pyridin-4-yl)propanoyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-(5-amino-1H-1,2,4-triazol-3-yl)-1-(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)propan-1-one
5-{1-[2-methoxy-2-(thiophen-2-yl)ethyl]-1H-1,2,3-triazol-4-yl}pyrimidine
9-(6-methylpyridine-3-carbonyl)-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[3-({7-methyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}sulfonyl)phenyl]acetamide
N-[phenyl(pyridin-2-yl)methyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
(3aS,6aS)-2-[(4-chloro-3-fluorophenyl)methyl]-5-(2-methoxyacetyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
8-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)sulfonyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
3-({2-[1-(2H-1,3-benzodioxol-5-yl)propan-2-yl]-1H-imidazol-1-yl}methyl)-5-(propan-2-yl)-1,2,4-oxadiazole
N-(7-{6-azabicyclo[3.2.1]octane-6-carbonyl}-1-cyclopentyl-1H-1,3-benzodiazol-5-yl)benzamide
N-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]cyclopentanecarboxamide
3-[5-oxo-3-(pyridin-3-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-4-yl]propanoic acid
4-methyl-N-(2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(piperidine-4-carbonyl)piperidin-3-ol
3-{3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}-N-methylpropanamide
5-benzyl-3-(3-methylbut-2-en-1-yl)-5-(piperidin-4-yl)imidazolidine-2,4-dione